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List of works by Sébastien Albrecht

Alkynes as masked ylides: gold-catalysed intermolecular reactions of propargylic carboxylates with sulfides

scientific article published on 24 October 2007

Allosteric inhibition of aminopeptidase N functions related to tumor growth and virus infection.

scientific article

Amino-benzosuberone: a novel warhead for selective inhibition of human aminopeptidase-N/CD13

scientific article published on 11 January 2011

Aminobenzosuberone Scaffold as a Modular Chemical Tool for the Inhibition of Therapeutically Relevant M1 Aminopeptidases

scientific article published on 11 October 2018

Cyclin-dependent kinase 12 is a drug target for visceral leishmaniasis

scientific article published in Nature

Discovery of Indoline-2-carboxamide Derivatives as a New Class of Brain-Penetrant Inhibitors of Trypanosoma brucei

scientific article published on 29 September 2015

Exploring S1 plasticity and probing S1' subsite of mammalian aminopeptidase N/CD13 with highly potent and selective aminobenzosuberone inhibitors

scientific article published on 01 May 2015

Gold- or platinum-catalyzed synthesis of sulfur heterocycles: access to sulfur ylides without using sacrificial functionality

scientific article published on 01 January 2009

Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis

scientific article published on 20 December 2018

Insight into the remarkable affinity and selectivity of the aminobenzosuberone scaffold for the M1 aminopeptidases family based on structure analysis.

scientific article published on 6 April 2017

Rapid and efficient synthesis of a novel series of substituted aminobenzosuberone derivatives as potent, selective, non-peptidic neutral aminopeptidase inhibitors

scientific article published on 28 June 2012

Selective inhibition of PfA-M1, over PfA-M17, by an amino-benzosuberone derivative blocks malaria parasites development in vitro and in vivo

scientific article published on 21 September 2017

Synthesis and structure activity relationships of novel non-peptidic metallo-aminopeptidase inhibitors

scientific article published on 17 July 2006

Synthesis of amino-hydroxy-benzocycloheptenones as potent, selective, non-peptidic dinuclear zinc metalloaminopeptidase inhibitors.

scientific article

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