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List of works by Lucjusz Zaprutko

A facile synthesis and anticancer activity evaluation of spiro[thiazolidinone-isatin] conjugates

scientific article published on 3 October 2011

Anti-COVID drugs: repurposing existing drugs or search for new complex entities, strategies and perspectives

scientific article published on 23 July 2020

Anticancer effect of A-ring or/and C-ring modified oleanolic acid derivatives on KB, MCF-7 and HeLa cell lines

scientific article published on January 5, 2012

Hybrid Compounds Strategy in the Synthesis of Oleanolic Acid Skeleton-NSAID Derivatives.

scientific article

Methyl 3-hydroxyimino-11-oxoolean-12-en-28-oate (HIMOXOL), a synthetic oleanolic acid derivative, induces both apoptosis and autophagy in MDA-MB-231 breast cancer cells.

scientific article published on 27 November 2013

Microwave (MW), Ultrasound (US) and Combined Synergic MW-US Strategies for Rapid Functionalization of Pharmaceutical Use Phenols

scientific article published on 15 September 2018

Microwave assisted synthesis of fragrant jasmone heterocyclic analogues

scientific article published on 24 March 2006

Molecular Consortia-Various Structural and Synthetic Concepts for More Effective Therapeutics Synthesis.

scientific article published on 6 April 2018

Multidirectional Efficacy of Biologically Active Nitro Compounds Included in Medicines.

scientific article published on 29 May 2018

Oleanolic Acid A-lactams Inhibit the Growth of HeLa, KB, MCF-7 and Hep-G2 Cancer Cell Lines at Micromolar Concentrations.

scientific article published on 6 September 2015

Oleanolic Acid’s Semisynthetic Derivatives HIMOXOL and Br-HIMOLID Show Proautophagic Potential and Inhibit Migration of HER2-Positive Breast Cancer Cells In Vitro

scientific article published in 2021

Oleanolic acid derivative methyl 3,11-dioxoolean-12-en-28-olate targets multidrug resistance related to ABCB1.

scientific article

Proapoptotic activity and ABCC1-related multidrug resistance reduction ability of semisynthetic oleanolic acid derivatives DIOXOL and HIMOXOL in human acute promyelocytic leukemia cells

scientific article published on 8 September 2015

Recent advances in synthesis and biological activity of triterpenic acylated oximes.

scientific article published on 11 April 2014

Semisynthetic oleanane triterpenoids inhibit migration and invasion of human breast cancer cells through downregulated expression of the ITGB1/PTK2/PXN pathway.

scientific article

Simple amides of oleanolic acid as effective penetration enhancers

scientific article

Strong and Long-Lasting Antinociceptive and Anti-inflammatory Conjugate of Naturally Occurring Oleanolic Acid and Aspirin

scientific article published on 12 July 2016

Synthesis and antitumor activity of aminopropoxy derivatives of betulin, erythrodiol, and uvaol

scientific article published on 01 May 2011

Synthesis of novel thiazolone-based compounds containing pyrazoline moiety and evaluation of their anticancer activity.

scientific article

Synthesis of some N-substituted nitroimidazole derivatives as potential antioxidant and antifungal agents.

scientific article published on 28 May 2008

Synthesis, structure and biological evaluation of novel bicyclic nitroimidazole derivatives

scientific article published on 20 January 2012

The Structure and Activity of Double-Nitroimidazoles. A Mini-Review

scientific article published on 25 July 2018

The analgesic and anti-inflammatory effect of new oleanolic acid acyloxyimino derivative

scientific article published on 31 July 2012