List of works - Dawid Debowski

Antimicrobial Activity of Chimera Peptides Composed of Human Neutrophil Peptide 1 (HNP-1) Truncated Analogues and Bovine Lactoferrampin

scientific article published on 10 August 2018

Atomic resolution crystal structure of HV-BBI protease inhibitor from amphibian skin in complex with bovine trypsin

scientific article

Bladder cancer detection using a peptide substrate of the 20S proteasome.

scientific article published on 21 June 2016

Bowman-Birk Inhibitors: Insights into Family of Multifunctional Proteins and Peptides with Potential Therapeutical Applications

scientific article published on 25 November 2020

Conjugates of Ciprofloxacin and Levofloxacin with Cell-Penetrating Peptide Exhibit Antifungal Activity and Mammalian Cytotoxicity ⬇️

scientific article published on 30 June 2020

Convenient preparation of deuterium-labeled analogs of peptides containing N-substituted glycines for a stable isotope dilution LC-MS quantitative analysis.

scientific article

Cyclic Peptidic Furin Inhibitors Developed by Combinatorial Chemistry

scientific article published on 13 April 2023

Design and chemical syntheses of potent matriptase-2 inhibitors based on trypsin inhibitor SFTI-1 isolated from sunflower seeds.

scientific article published on 27 May 2017

Fluorescent analogs of trypsin inhibitor SFTI-1 isolated from sunflower seeds--synthesis and applications.

scientific article published on January 2014

Hybrid analogues of SFTI-1 modified in P1position by β- and γ-amino acids andN-substituted β-alanines

scientific article published on 01 April 2013

Implication of the disulfide bridge in trypsin inhibitor SFTI-1 in its interaction with serine proteinases.

scientific article published on 29 October 2010

Inhibition of human and yeast 20S proteasome by analogues of trypsin inhibitor SFTI-1

scientific article

Inhibitors of Matriptase-2 Based on the Trypsin Inhibitor SFTI-1

scientific article published on 19 June 2015

Inhibitory and antimicrobial activities of OGTI and HV-BBI peptides, fragments and analogs derived from amphibian skin

scientific article

Interactions between trypsin and its peptidic inhibitors studied by isothermal titration calorimetry (ITC)

Introduction of Pro and Its Analogues in the Conserved P1 Position of Trypsin Inhibitor SFTI-1 Retains Its Inhibitory Activity

scientific article published on 01 November 2011

Introduction of non-natural amino acid residues into the substrate-specific P1 position of trypsin inhibitor SFTI-1 yields potent chymotrypsin and cathepsin G inhibitors.

scientific article published on 27 March 2009

Investigation of Serine-Proteinase-Catalyzed Peptide Splicing in Analogues of Sunflower Trypsin Inhibitor 1 (SFTI-1)

scientific article

Investigation of peptide splicing using two-peptide-chain analogs of trypsin inhibitor SFTI-1.

scientific article

Matriptase-2: monitoring and inhibiting its proteolytic activity

Natural Proteinaceous Inhibitors of Serine Proteases

scientific article published on January 1, 2013

Noncovalent inhibitors of human 20S and 26S proteasome based on trypsin inhibitor SFTI-1.

scientific article published on 3 June 2016

Novel internally quenched substrate of the trypsin-like subunit of 20S eukaryotic proteasome

scientific article published on 24 August 2015

Peptide conjugates of lactoferricin analogues and antimicrobials-Design, chemical synthesis, and evaluation of antimicrobial activity and mammalian cytotoxicity

scientific article published on 05 April 2019

Peptide splicing in a double-sequence analogue of trypsin inhibitor SFTI-1 substituted in the P₁ positions by peptoid monomers.

scientific article published in May 2015

Peptomeric analogues of trypsin inhibitor SFTI-1 isolated from sunflower seeds

scientific article published in April 2008

Selection of peptomeric inhibitors of bovine alpha-chymotrypsin and cathepsin G based on trypsin inhibitor SFTI-1 using a combinatorial chemistry approach

scientific article

Spliced analogues of trypsin inhibitor SFTI-1 and their application for tracing proteolysis and delivery of cargos inside the cells

scientific article published on 14 September 2016

Truncation of Huia versabilis Bowman-Birk inhibitor increases its selectivity, matriptase-1 inhibitory activity and proteolytic stability

scientific article published on 10 March 2020

List of works by Dawid Debowski

Antimicrobial Activity of Chimera Peptides Composed of Human Neutrophil Peptide 1 (HNP-1) Truncated Analogues and Bovine Lactoferrampin

Atomic resolution crystal structure of HV-BBI protease inhibitor from amphibian skin in complex with bovine trypsin

Bladder cancer detection using a peptide substrate of the 20S proteasome.

Bowman-Birk Inhibitors: Insights into Family of Multifunctional Proteins and Peptides with Potential Therapeutical Applications

Conjugates of Ciprofloxacin and Levofloxacin with Cell-Penetrating Peptide Exhibit Antifungal Activity and Mammalian Cytotoxicity ⬇️

Convenient preparation of deuterium-labeled analogs of peptides containing N-substituted glycines for a stable isotope dilution LC-MS quantitative analysis.

Cyclic Peptidic Furin Inhibitors Developed by Combinatorial Chemistry

Design and chemical syntheses of potent matriptase-2 inhibitors based on trypsin inhibitor SFTI-1 isolated from sunflower seeds.

Fluorescent analogs of trypsin inhibitor SFTI-1 isolated from sunflower seeds--synthesis and applications.

Hybrid analogues of SFTI-1 modified in P1position by β- and γ-amino acids andN-substituted β-alanines

Implication of the disulfide bridge in trypsin inhibitor SFTI-1 in its interaction with serine proteinases.

Inhibition of human and yeast 20S proteasome by analogues of trypsin inhibitor SFTI-1

Inhibitors of Matriptase-2 Based on the Trypsin Inhibitor SFTI-1

Inhibitory and antimicrobial activities of OGTI and HV-BBI peptides, fragments and analogs derived from amphibian skin

Interactions between trypsin and its peptidic inhibitors studied by isothermal titration calorimetry (ITC)

Introduction of Pro and Its Analogues in the Conserved P1 Position of Trypsin Inhibitor SFTI-1 Retains Its Inhibitory Activity

Introduction of non-natural amino acid residues into the substrate-specific P1 position of trypsin inhibitor SFTI-1 yields potent chymotrypsin and cathepsin G inhibitors.

Investigation of Serine-Proteinase-Catalyzed Peptide Splicing in Analogues of Sunflower Trypsin Inhibitor 1 (SFTI-1)

Investigation of peptide splicing using two-peptide-chain analogs of trypsin inhibitor SFTI-1.

Matriptase-2: monitoring and inhibiting its proteolytic activity

Natural Proteinaceous Inhibitors of Serine Proteases

Noncovalent inhibitors of human 20S and 26S proteasome based on trypsin inhibitor SFTI-1.

Novel internally quenched substrate of the trypsin-like subunit of 20S eukaryotic proteasome

Peptide conjugates of lactoferricin analogues and antimicrobials-Design, chemical synthesis, and evaluation of antimicrobial activity and mammalian cytotoxicity

Peptide splicing in a double-sequence analogue of trypsin inhibitor SFTI-1 substituted in the P₁ positions by peptoid monomers.

Peptomeric analogues of trypsin inhibitor SFTI-1 isolated from sunflower seeds

Selection of peptomeric inhibitors of bovine alpha-chymotrypsin and cathepsin G based on trypsin inhibitor SFTI-1 using a combinatorial chemistry approach

Spliced analogues of trypsin inhibitor SFTI-1 and their application for tracing proteolysis and delivery of cargos inside the cells

Truncation of Huia versabilis Bowman-Birk inhibitor increases its selectivity, matriptase-1 inhibitory activity and proteolytic stability