Search filters

List of works by Dana Ferraris

6-Hydroxy-1,2,4-triazine-3,5(2H,4H)-dione Derivatives as Novel D-Amino Acid Oxidase Inhibitors

scientific article published on 26 August 2015

Accumulation of free ADP-ribose from mitochondria mediates oxidative stress-induced gating of TRPM2 cation channels

scientific article

Azetidine-based inhibitors of dipeptidyl peptidase IV (DPP IV).

scientific article published on January 2007

Catalytic, enantioselective alkylation of alpha-imino esters: the synthesis of nonnatural alpha-amino acid derivatives.

scientific article published in January 2002

D-Amino acid oxidase inhibitors based on the 5-hydroxy-1,2,4-triazin-6(1H)-one scaffold.

scientific article published on 23 February 2016

D-Amino-Acid Oxidase Inhibition Increases D-Serine Plasma Levels in Mouse But not in Monkey or Dog.

scientific article published on 16 October 2015

DPP IV inhibitor blocks mescaline-induced scratching and amphetamine-induced hyperactivity in mice.

scientific article published in June 2005

Design and synthesis of poly ADP-ribose polymerase-1 inhibitors. 2. Biological evaluation of aza-5[H]-phenanthridin-6-ones as potent, aqueous-soluble compounds for the treatment of ischemic injuries.

scientific article

Design and synthesis of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. Part 4: biological evaluation of imidazobenzodiazepines as potent PARP-1 inhibitors for treatment of ischemic injuries.

scientific article published in August 2003

Design and synthesis of poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors. Part 3: In vitro evaluation of 1,3,4,5-tetrahydro-benzo[c][1,6]- and [c][1,7]-naphthyridin-6-ones

scientific article published on 01 August 2003

Design and synthesis of potent inhibitors of the mono(ADP-ribosyl)transferase, PARP14.

scientific article published on 29 April 2017

Design, synthesis and evaluation of potent and selective inhibitors of mono-(ADP-ribosyl)transferases PARP10 and PARP14

scientific article published on 03 May 2018

Design, synthesis, and pharmacological evaluation of bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide 3 (BPTES) analogs as glutaminase inhibitors.

scientific article published on 30 November 2012

Design, synthesis, and pharmacological evaluation of fluorinated tetrahydrouridine derivatives as inhibitors of cytidine deaminase

scientific article published on 24 February 2014

Design, synthesis, and pharmacological evaluation of glutamate carboxypeptidase II (GCPII) inhibitors based on thioalkylbenzoic acid scaffolds

scientific article published on 12 June 2012

Development of a high-throughput method for the determination of pharmacological levels of plasma D-serine.

scientific article published on 16 August 2011

Diastereo- and Enantioselective Alkylation of alpha-Imino Esters with Enol Silanes Catalyzed by (R)-Tol-BINAP-CuClO(4).(MeCN)(2)

scientific article published on 01 September 1998

Discovery of 6-Diazo-5-oxo-l-norleucine (DON) Prodrugs with Enhanced CSF Delivery in Monkeys: A Potential Treatment for Glioblastoma

scientific article published on 25 August 2016

Dual leucine zipper kinase as a therapeutic target for neurodegenerative conditions.

scientific article published on October 2013

Evolution of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. From concept to clinic.

scientific article published on June 2010

Glutamate production by HIV-1 infected human macrophage is blocked by the inhibition of glutaminase

scientific article

Inhibition of xc- transporter-mediated cystine uptake by sulfasalazine analogs ⬇️

scientific article published on August 12, 2011

Ketopyrrolidines and ketoazetidines as potent dipeptidyl peptidase IV (DPP IV) inhibitors.

scientific article published in November 2004

Novel mechanism of inhibition of rat kidney-type glutaminase by bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide (BPTES)

scientific article

Nucleophilic metal complexes as acylation catalysts: solvent-dependent "switch" mechanisms leading to the first catalyzed Staudinger reaction

scientific article published on 01 December 1999

Peptidomimetics of Arg-Phe-NH2 as small molecule agonists of Mas-related gene C (MrgC) receptors.

scientific article

Recent Advances in the Discovery of D-Amino Acid Oxidase Inhibitors and Their Therapeutic Utility in Schizophrenia ⬇️

scientific article published on January 1, 2011

Structure-Activity Relationships of Glutamate Carboxypeptidase II (GCPII) Inhibitors ⬇️

scientific article published on January 1, 2012

Structure-function analysis of water-soluble inhibitors of the catalytic domain of exotoxin A from Pseudomonas aeruginosa

scientific article

Synthesis and SAR of 1-hydroxy-1H-benzo[d]imidazol-2(3H)-ones as Inhibitors of D-Amino Acid Oxidase.

scientific article

Synthesis and biological evaluation of D-amino acid oxidase inhibitors.

scientific article published on 29 May 2008

Synthesis of kojic acid derivatives as secondary binding site probes of D-amino acid oxidase

scientific article published on May 2013

Synthesis of substituted 5[H]phenanthridin-6-ones as potent poly(ADP-ribose)polymerase-1 (PARP1) inhibitors.

scientific article

Synthesis, characterization and antineoplastic activity of bis-aziridinyl dimeric naphthoquinone - A novel class of compounds with potent activity against acute myeloid leukemia cells

scientific article published on 17 November 2016

The discovery and structure-activity relationships of indole-based inhibitors of glutamate carboxypeptidase II.

scientific article published on 26 October 2010

The metabolic profile of tumors depends on both the responsible genetic lesion and tissue type.

scientific article published on February 2012

Unprecedented Binding Mode of Hydroxamate-Based Inhibitors of Glutamate Carboxypeptidase II: Structural Characterization and Biological Activity

scientific article

Paulina is supported by:

About Paulina

Help