List of works by Jef Rozenski

2'-O-hydroxyalkoxymethylribonucleosides and their incorporation into oligoribonucleotides

scientific article published on January 2007

2,5-Bis-(2-hydroxybenzoylamino)pentanoic Acid, a Salicylic Acid-Metabolite Isolated from Chicken: Characterization and Independent Synthesis

2,5-Bis-(2-hydroxybenzoylamino)pentanoic acid, a salicylic acid-metabolite isolated from chicken: characterization and independent synthesis.

scientific article

2-Hydroxyethoxyethylated Bases as Acyclic Analogues of 1,5-Anhydrohexitol Nucleoside Derivatives

2′-Deoxyuridines with a 5-Heteroaromatic Substituent: Synthesis and Biological Evaluation

3′-Deoxy-3′-hydroxymethyl-aldopentopyranosyl nucleoside synthesis. Part I

5'-Deoxy congeners of 9-(3-amido-3-deoxy-beta-D-xylofuranosyl)-N(6)-cyclopentyladenine: new adenosine A(1) receptor antagonists and inverse agonists

scientific article published in April 2002

5-Hydroxytryptophan as a building block in oligopeptides using Fmoc/tBu SPPS

5′-(N-aminoacyl)-sulfonamido-5′-deoxyadenosine: Attempts for a stable alternative for aminoacyl-sulfamoyl adenosines as aaRS inhibitors

scholarly article by Bharat Gadakh et al published March 2015 in European Journal of Medicinal Chemistry

A PKS/NRPS/FAS hybrid gene cluster from Serratia plymuthica RVH1 encoding the biosynthesis of three broad spectrum, zeamine-related antibiotics ⬇️

scientific article

A Single Amino Acid Substitution in Therminator DNA Polymerase Increases Incorporation Efficiency of Deoxyxylonucleotides

scientific article published on 26 October 2018

A novel, highly selective inhibitor of pestivirus replication that targets the viral RNA-dependent RNA polymerase

scientific article

A short path synthesis of [13C/15N] multilabeled pyrimidine nucleosides starting from glucopyranose nucleosides

scientific article published in March 2003

A standardized and biocompatible preparation of aggregate-free amyloid beta peptide for biophysical and biological studies of Alzheimer's disease

scientific article published on 11 May 2011

A synthetic substrate of DNA polymerase deviating from the bases, sugar, and leaving group of canonical deoxynucleoside triphosphates

scientific article

Abl1 inhibitory contaminants leach from plastic tubes.

scientific article

Achiral, acyclic nucleic acids: synthesis and biophysical studies of a possible prebiotic polymer

Alpha-homo-DNA and RNA form a parallel oriented non-A, non-B-type double helical structure.

scientific article published in December 2001

Amino acids derived from ornithine

Aminopurine and aminoquinazoline scaffolds for development of potential dengue virus inhibitors

scientific article published on 5 October 2016

An acyclic 5-nitroindazole nucleoside analogue as ambiguous nucleoside

scientific article

Analysis of nucleosides using the atmospheric-pressure solids analysis probe for ionization

article

Antibacterial 5'-O-(N-dipeptidyl)-sulfamoyladenosines.

scientific article

Application of the Mitsunobu-Type Condensation Reaction to the Synthesis of Phosphonate Derivatives of Cyclohexenyl and Cyclohexanyl Nucleosides

Aspartic acid based nucleoside phosphoramidate prodrugs as potent inhibitors of hepatitis C virus replication

scientific article published on May 2015

Astemizole analogues with reduced hERG inhibition as potent antimalarial compounds.

scientific article published on 7 October 2017

Base pairing involving artificial bases in vitro and in vivo.

scientific article

Base pairing properties of D- and L-cyclohexene nucleic acids (CeNA).

scientific article published in January 2003

Base substituted 5'-O-(N-isoleucyl)sulfamoyl nucleoside analogues as potential antibacterial agents.

scientific article

Biological effects of hexitol and altritol-modified siRNAs targeting B-Raf

scientific article published on 30 January 2009

Characterization and sequence confirmation of unnatural amino acid containing peptide libraries using electrospray ionization mass spectrometry

scientific article

Characterization and sequence verification of thiolated deoxyoligonucleotides used for microarray construction

scientific article published in 2006

Characterization of Oligonucleotide Sequence Isomers in Mixtures Using HPLC/MS

Characterization of insulin-degrading enzyme-mediated cleavage of Aβ in distinct aggregation states

scientific article published on 8 March 2016

Characterization of modification sites during peptide synthesis using liquid secondary ion/collision-induced dissociation mass spectrometry and a computer program

scholarly article by Jef Rozenski et al published November 1994 in Journal of Mass Spectrometry

Characterization of peptide chain length and constituency requirements for YejABEF-mediated uptake of microcin C analogues

scientific article published on 20 May 2011

Characterization of the posttranscriptional modifications in Legionella pneumophila small-subunit ribosomal RNA.

scientific article published in December 2008

ChemInform Abstract: Oligonucleotides Containing Disaccharide Nucleosides

ChemInform Abstract: Selection of New Sequence-Selective Unnatural Peptides Binding to Double-Stranded Deoxyribonucleic Acids (dsDNA) by Means of a Gel-Retardation Experiment for Library Analysis

ChemInform Abstract: Suzuki Reactions on Chloropyridazinones: An Easy Approach Towards Arylated 3(2H)-Pyridazinones

article by Bert U. W. Maes et al published 26 May 2010 in ChemInform

Chemical Etiology of Nucleic Acids: Aminopropyl Nucleic Acids (APNAs)

scientific article published on 01 April 2007

Chemical Morphing of DNA Containing Four Noncanonical Bases

article published in 2016

Chemical Morphing of DNA Containing Four Noncanonical Bases.

scientific article

Chemical incorporation of 1-methyladenosine into oligonucleotides

scientific article published on March 2002

Chemical incorporation of 1-methyladenosine, minor tRNA component, into oligonucleotides.

scientific article published in May 2003

Chemical incorporation of minor tRNA component O-β-D-ribofuranosyl-(1''-2')-adenosine-5''-phosphate into oligoribonucleotides

Cleavage of DNA without loss of genetic information by incorporation of a disaccharide nucleoside

scientific article

Conjugation of Oligonucleotides to 3′-Polar Moieties

article

Correction: Base pairing involving artificial bases and

Delivery of antisense oligonucleotides using cholesterol-modified sense dendrimers and cationic lipids

scientific article published on July 2005

Dendritic Nucleotides: Interaction with an Aliphatic Acid Monolayer

scientific article published on 01 September 2008

Design and synthesis of nucleolipids as possible activated precursors for oligomer formation via intramolecular catalysis: stability study and supramolecular organization

scientific article published on 9 December 2014

Detection of RNA hybridization by pyrene-labeled probes.

scientific article published in May 2009

Determination of Nearest Neighbors in Nucleic Acids by Mass Spectrometry

scientific article published on 01 April 1999

Development of Synthetic Strategies for the Construction of Pyrido[4,3-d]pyrimidine Libraries – the Discovery of a New Class of PDE-4 Inhibitors

article

Development of Synthetic Strategies for the Construction of Pyrido[4,3-d]pyrimidine Libraries — The Discovery of a New Class of PDE-4 Inhibitors

Development of a conjugate of (99m)Tc-EC with aminomethylenediphosphonate in the search for a bone tracer with fast clearance from soft tissue

scientific article published in January 2002

Discovery of 7-N-Piperazinylthiazolo[5,4-d]pyrimidine Analogues as a Novel Class of Immunosuppressive Agents with in Vivo Biological Activity

Discovery of an acyclic nucleoside phosphonate that inhibits Mycobacterium Tuberculosis ThyX based on the binding mode of a 5-alkynyl substrate analogue

scholarly article published 2014

Discovery of an acyclic nucleoside phosphonate that inhibits Mycobacterium tuberculosis ThyX based on the binding mode of a 5-alkynyl substrate analogue

scientific article

Discovery of bicyclic thymidine analogues as selective and high-affinity inhibitors of Mycobacterium tuberculosis thymidine monophosphate kinase

scientific article published in December 2004

Divergent strategy for the synthesis of alpha-aryl-substituted fosmidomycin analogues

scientific article published on 12 April 2007

Enantioselective Approach to the Synthesis of Cyclohexane Carbocyclic Nucleosides

Enzymatic Synthesis of Phosphonomethyl Oligonucleotides by Therminator Polymerase

scholarly article by Marleen Renders et al published 26 March 2007 in Angewandte Chemie International Edition

Enzymatic Synthesis of Phosphonomethyl Oligonucleotides by Therminator Polymerase

Enzymatic resolution and base pairing properties of D- and L-cyclohexenyl nucleic acids (CeNA).

scientific article

Evaluation of Capillary HPLC/Mass Spectrometry as an Alternative Analysis Method for Gel Electrophoresis of Oligonucleotides

Evaluation of Capillary HPLC/Mass Spectrometry as an Alternative Analysis Method for Gel Electrophoresis of Oligonucleotides

article published in 2004

Evidence for the isomerization and decarboxylation in the photoconversion of the red fluorescent protein DsRed

scientific article

Extended targeting potential and improved synthesis of Microcin C analogs as antibacterials.

scientific article

Gain of function of mutant p53 by coaggregation with multiple tumor suppressors

Genetic and functional characterization of cyclic lipopeptide white-line-inducing principle (WLIP) production by rice rhizosphere isolate Pseudomonas putida RW10S2.

scientific article published on 27 April 2012

Hybridisation potential of 1',3'-Di-O-methylaltropyranoside nucleic acids

scientific article published on 3 March 2015

Hybridization between “Six-Membered” Nucleic Acids:  RNA as a Universal Information System

scientific article published on 01 December 2001

Hybridization potential of oligonucleotides comprising 3'-O-methylated altritol nucleosides

scientific article published on 9 October 2012

Hybridization specificity, enzymatic activity and biological (Ha-ras) activity of oligonucleotides containing 2,4-dideoxy-beta-D-erythro-hexopyranosyl nucleosides

scientific article published in October 1993

Identification of a peptide inhibitor against glycosomal phosphoglycerate kinase of Trypanosoma brucei by a synthetic peptide library approach.

scientific article published on March 1995

Imidazopyridine- and purine-thioacetamide derivatives: potent inhibitors of nucleotide pyrophosphatase/phosphodiesterase 1 (NPP1).

scientific article

Improved hybridisation potential of oligonucleotides comprising O-methylated anhydrohexitol nucleoside congeners

scientific article published on October 2001

In search of Flavivirus inhibitors part 2: tritylated, diphenylmethylated and other alkylated nucleoside analogues

scientific article published on 10 February 2014

In search of flavivirus inhibitors: evaluation of different tritylated nucleoside analogues

scientific article published on 24 April 2013

Incorporation of 5-hydroxytryptophan in oligopeptides

Interpretation of oligonucleotide mass spectra for determination of sequence using electrospray ionization and tandem mass spectrometry.

scientific article published in July 1996

Isothiazolo[4,3-b]pyridines as inhibitors of cyclin G associated kinase : synthesis, structure-activity relationship studies and antiviral activity.

scientific article published on 07 August 2015

Mass spectrometric fragmentation of cyclic peptides belonging to the polymyxin and colistin antibiotics studied by ion trap and quadrupole/orthogonal-acceleration time-of-flight technology

scientific article

MccE provides resistance to protein synthesis inhibitor microcin C by acetylating the processed form of the antibiotic

scientific article

Methylated Hexitol Nucleic Acids, Towards Congeners with Improved Antisense Potential

scientific article published on 01 May 2003

Minimal interference from paricalcitol (Zemplar®) in underivatized 1,25-dihydroxyvitamin D LC-MS/MS assays.

scientific article published on 8 December 2013

Mixed oligonucleotide analogues with an acyclic carbohydrate moiety and a N-cyanoguanidine functionality

scientific article published in 1994

Modification of the universally unmodified uridine-33 in a mitochondria-imported edited tRNA and the role of the anticodon arm structure on editing efficiency

scientific article

Molecular plasticity regulates oligomerization and cytotoxicity of the multipeptide-length amyloid-β peptide pool

scientific article

N-alkylated aminoacyl sulfamoyladenosines as potential inhibitors of aminoacylation reactions and microcin C analogues containing D-amino acids

scientific article

Neurotoxicity of Alzheimer's disease Aβ peptides is induced by small changes in the Aβ42 to Aβ40 ratio

scientific article

New Techniques for the Rapid Characterization of Oligonucleotides by Mass Spectrometry

scientific article published on 01 June 1999

New dsDNA binding unnatural oligopeptides with pyrimidine selectivity

scientific article

New dsDNA-Binding Hybrid Molecules Combining an Unnatural Peptide and an Intercalating Moiety

scholarly article by Patrick Chaltin et al published March 2003 in Helvetica Chimica Acta

Oligonucleotide Analogues with 4-Hydroxy-N-Acetylprolinol as Sugar Substitute

article by Griet Ceulemans et al published December 1997 in Chemistry—A European Journal

Oligonucleotides Composed of 2‘-Deoxy-1‘,5‘-anhydro-d-mannitol Nucleosides with a Purine Base Moiety

article published in 1998

Oligonucleotides with 3-hydroxy-N-acetylprolinol as sugar substitute

article by Griet Ceulemans et al published November 1997 in Tetrahedron

Phenyltriazole-functionalized sulfamate inhibitors targeting tyrosyl- or isoleucyl-tRNA synthetase

scientific article published on 05 June 2020

Post-transcriptional modification mapping in the Clostridium acetobutylicum 16S rRNA by mass spectrometry and reverse transcriptase assays

scientific article published on 3 May 2007

Potential for Biocontrol of Hairy Root Disease by a Paenibacillus Clade

scientific article published on 22 March 2017

Pretargeting of necrotic tumors with biotinylated hypericin using 123I-labeled avidin: evaluation of a two-step strategy

scientific article

Problems and Prospects in the Characterization of Posttranscriptional Modifications in Large RNAs

Promysalin, a salicylate-containing Pseudomonas putida antibiotic, promotes surface colonization and selectively targets other Pseudomonas. ⬇️

scientific article published in October 2011

Proof of concept for the reduction of classical swine fever infection in pigs by a novel viral polymerase inhibitor

scientific article published on 4 March 2009

Protection of 1-methyladenosine and its chemical incorporation into oligonucleotides

Pseudouridine detection improvement by derivatization with methyl vinyl sulfone and capillary HPLC-mass spectrometry

scientific article published on 18 July 2005

Pyrrolo-C as a molecular probe for monitoring conformations of the tRNA 3' end.

scientific article published on 28 August 2008

Quantitative Structure-Activity Relationships for Antimicrobial Nitroheterocyclic Drugs

scholarly article by Jef Rozenski et al published 1995 in QSAR and Combinatorial Science

Recognition of HNA and 1,5-anhydrohexitol nucleotides by DNA metabolizing enzymes

scientific article

Recognition of threosyl nucleotides by DNA and RNA polymerases

scientific article published on November 2003

Ribavirin derivatives with a hexitol moiety: synthesis and antiviral evaluation

scientific article published on January 2003

SOS: a simple interactive program for ab initio oligonucleotide sequencing by mass spectrometry

scientific article published in March 2002

Screening of a synthetic pentapeptide library composed of d-amino acids against fructose-1,6-biphosphate aldolase

Stereocontrolled synthesis of phosphonate derivatives of tetrahydro- and dihydro-2H-pyranyl nucleosides: The selectivity of the Ferrier rearrangement

Stereospecific synthesis of a pentopyranosyl analogue of d4T monophosphate

scientific article published in 1994

Straightforward Synthesis of Labeled and Unlabeled Pyrimidine d4Ns via 2′,3′-Diyne seco Analogues through Olefin Metathesis Reactions

article published in 2003

Substituted 5-Benzyl-2-phenyl-5H-imidazo[4,5-c]pyridines: A New Class of Pestivirus Inhibitors

Substituted 5-benzyl-2-phenyl-5H-imidazo[4,5-c]pyridines: a new class of pestivirus inhibitors

scientific article published on 9 August 2006

Suzuki reactions on chloropyridazinones: an easy approach towards arylated 3(2 H )-pyridazinones

article by Bert U.W Maes et al published February 2001 in Tetrahedron

Synthesis and Antiviral Activity of the alpha-Analogues of 1,5-Anhydrohexitol Nucleosides (1,5-Anhydro-2,3-dideoxy-D-ribohexitol Nucleosides).

scientific article published in April 1997

Synthesis and Biological Evaluation of Lipophilic Nucleoside Analogues as Inhibitors of Aminoacyl-tRNA Synthetases

scientific article published on 09 October 2019

Synthesis and Biological Evaluation of a Series of New Cyclohexenyl Nucleosides

Synthesis and Conformational Analysis of 2?-Deoxy-2?-(3-methoxybenzamido)adenosine, a rational-designed inhibitor of trypanosomal glyceraldehyde phosphate dehydrogenase (GAPDH)

article

Synthesis and Conformational Properties of O-β-D-Ribofuranosyl-(1′′-2′)-guanosine and (Adenosine)-5′′-phosphate

Synthesis and Conformational Study of 3-Hydroxy-4-(Hydroxymethyl)-1-Cyclohexanyl Purines and Pyrimidines

article

Synthesis and Properties of O--D-ribofuranosyl-(1″→2′)-guanosine-5″- O-phosphate and Its Derivatives

scholarly article by Ekaterina V. Efimtseva et al published February 2003 in Helvetica Chimica Acta

Synthesis and Properties of O-β-D-Ribofuranosyl-(1″-2′)-Adenosine-5″-O-Phosphate and Its Derivatives

scholarly article by Andrei A. Rodionov et al published October 2000 in Nucleosides, Nucleotides & Nucleic Acids

Synthesis and Properties of Oligonucleotides Containing 2,4-Dihydroxycyclohexyl Nucleosides

scholarly article by Dorothée Bardiot et al published December 2005 in Helvetica Chimica Acta

Synthesis and Stability of Oligonucleotides Containing Acyclic Achiral Nucleoside Analogues with Two Base Moieties

Synthesis and Structure-Activity Relationship Studies of Benzo[b][1,4]oxazin-3(4H)-one Analogues as Inhibitors of Mycobacterial Thymidylate Synthase X

scientific article published on 20 February 2019

Synthesis and anti-BVDV activity of acridones as new potential antiviral agents

scientific article published in April 2006

Synthesis and antibacterial evaluation of a novel series of 2-(1,2-dihydro-3-oxo-3H-pyrazol-2-yl)benzothiazoles

scientific article

Synthesis and antiviral activity of a series of new cyclohexenyl nucleosides

scientific article published on January 2003

Synthesis and antiviral activity of acyclic analogues of 1,5-anhydrohexitol nucleosides using Mitsunobu reaction

Synthesis and antiviral activity of phosphonate derivatives of enantiomeric dihydro-2H-pyranyl nucleosides

scientific article published in 1995

Synthesis and base pairing properties of 1',5'-anhydro-L-hexitol nucleic acids (L-HNA).

scientific article

Synthesis and biological evaluation of a series of new cyclohexenyl nucleosides

scientific article published on May 2003

Synthesis and biological evaluation of novel PDMP analogues

scientific article published on 18 April 2006

Synthesis and cleavage experiments of oligonucleotide conjugates with a diimidazole-derived catalytic center

scientific article

Synthesis and conformational properties of O-beta-D-ribofuranosyl-(1''-2')-guanosine and (adenosine)-5''-phosphate

scientific article published in May 2003

Synthesis and evaluation of 5-substituted 2'-deoxyuridine monophosphate analogues as inhibitors of flavin-dependent thymidylate synthase in Mycobacterium tuberculosis

scientific article published on 9 June 2011

Synthesis and evaluation of 5-substituted-2'-deoxyuridine monophosphate analogues as inhibitors of flavin-dependent thymidylate synthase in Mycobacterium tuberculosis

scholarly article published 2011

Synthesis and evaluation of 6-aza-2'-deoxyuridine monophosphate analogs as inhibitors of thymidylate synthases, and as substrates or inhibitors of thymidine monophosphate kinase in Mycobacterium tuberculosis.

scientific article

Synthesis and evaluation of imidazole-4,5- and pyrazine-2,3-dicarboxamides targeting dengue and yellow fever virus

scientific article published on 22 September 2014

Synthesis and hybridization properties of inverse oligonucleotides.

scientific article published on August 1997

Synthesis and properties of aminopropyl nucleic acids

scientific article published in December 2005

Synthesis and properties of phosphorylated 3'-O-beta-D-ribofuranosyl-2'-deoxythymidine

scientific article published in April 2003

Synthesis and stability of oligonucleotides containing acyclic achiral nucleoside analogues with two base moieties

scientific article published on January 2004

Synthesis and structure-activity relationship studies of 2-(1,3,4-oxadiazole-2(3H)-thione)-3-amino-5-arylthieno[2,3-b]pyridines as inhibitors of DRAK2.

scientific article

Synthesis and structure-activity relationships of analogs of 2'-deoxy-2'-(3-methoxybenzamido)adenosine, a selective inhibitor of trypanosomal glycosomal glyceraldehyde-3-phosphate dehydrogenase.

scientific article

Synthesis of 1,5-Anhydrohexitol Nucleosides as Mimics of AZT, D4T and DDC

Synthesis of 2,4-dideoxy-.beta.-D-erythro-hexopyranosyl nucleosides

Synthesis of 3′-Fluoro-3′-deoxy-N6-cyclopentyladenosine

Synthesis of 3′-fluoromethylthio-, 3′-fluoromethylsulfinyl- and 3′-fluoromethylsulfonyl-substituted 3′-deoxythymidine

Synthesis of Oligoribonucleotides Containing Pyrimidine 2'-O-[(Hydroxyalkoxy)methyl]ribonucleosides

Synthesis of Peptidoglycan Units with UDP at the Anomeric Position

Synthesis of RNA ContainingO-β-D-Ribofuranosyl-(1″2′)-adenosine-5″-phosphate and 1-Methyladenosine, Minor Components of tRNA

scientific article published on 01 September 2005

Synthesis of Related Substances of Cefadroxil

Synthesis of a 2,4,6-trisubstituted 5-cyano-pyrimidine library and evaluation of its immunosuppressive activity in a Mixed Lymphocyte Reaction assay

scientific article

Synthesis of a new branched chain hexopyranosyl nucleoside: 1-[2′,3′-dideoxy-3′-C-(hydroxymethyl)-α-D-erythro-pentopyranosyl]-thymine

Synthesis of an Uncharged cAMP-Analogue

Synthesis of enantiomeric-pure cyclohexenyl nucleoside building blocks for oligonucleotide synthesis

Synthesis of homo-N-nucleosides, a series of C1' branched-chain nucleosides

Synthesis of homoceramides, novel ceramide analogues, and their lack of effect on the growth of hippocampal neurons

scientific article published in February 2002

Synthesis of protected D-altritol nucleosides as building blocks for oligonucleotide synthesis

Synthesis, Biological Evaluation, and Structure Analysis of a Series of New 1,5-Anhydrohexitol Nucleosides

article

Synthesis, cytotoxicity, and antiplasmodial and antitrypanosomal activity of new neocryptolepine derivatives

scientific article published on August 2002

Synthesis, enzymatic stability and physicochemical properties of oligonucleotides containing a N-cyanoguanidine linkage

Synthesis, in vitro cellular uptake and photo-induced antiproliferative effects of lipophilic hypericin acid derivatives.

scientific article published on 6 October 2005

Synthetic dsDNA-Binding Peptides Using Natural Compounds as Model

scholarly article by Filip Borgions et al published June 2006 in Helvetica Chimica Acta

Synthetic strategy and antiviral evaluation of diamide containing heterocycles targeting dengue and yellow fever virus

scientific article

The N1-(3'-Deoxythymidin-3'-yl)-N2-cyano-N3-(5'-deoxythymidin-5'-yl) Guanidine Dimeric Building Block in Automated DNA Synthesis and Mass Spectrometric Analysis of Its Integrity

article published in 1995

The RNA Modification Database, RNAMDB: 2011 update

scientific article

The RNA Modification Database: 1999 update

scientific article published on January 1999

The Small Subunit rRNA Modification Database

scientific article

The antimicrobial compound xantholysin defines a new group of Pseudomonas cyclic lipopeptides ⬇️

scientific article

The effect of addition of carbon powder to samples in liquid secondary ion mass spectrometry: Improved ionization of apolar compounds

article

Use of Cyclohexene Epoxides in the Preparation of Carbocyclic Nucleosides

Zebrafish bioassay-guided natural product discovery: isolation of angiogenesis inhibitors from East African medicinal plants

scientific article

α-Amino acids derived from ornithine as building blocks for peptide synthesis

article

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