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List of works by Jillian G Baker

A full pharmacological analysis of the three turkey β-adrenoceptors and comparison with the human β-adrenoceptors

scientific article

Agonist actions of "beta-blockers" provide evidence for two agonist activation sites or conformations of the human beta1-adrenoceptor

scientific article published in June 2003

Agonist and inverse agonist actions of beta-blockers at the human beta 2-adrenoceptor provide evidence for agonist-directed signaling

scientific article published on December 2003

Antagonist affinity measurements at the Gi-coupled human histamine H3 receptor expressed in CHO cells

scientific article published in 2008

Evidence for a secondary state of the human beta3-adrenoceptor.

scientific article published on 29 August 2005

Identification of key residues in transmembrane 4 responsible for the secondary, low-affinity conformation of the human β1-adrenoceptor

scientific article

Impact of polymorphic variants on the molecular pharmacology of the two-agonist conformations of the human β1-adrenoceptor

scientific article

Influence of agonist efficacy and receptor phosphorylation on antagonist affinity measurements: differences between second messenger and reporter gene responses

scientific article published in September 2003

Multiple GPCR conformations and signalling pathways: implications for antagonist affinity estimates.

scientific article published on 13 July 2007

Negative cooperativity across β1-adrenoceptor homodimers provides insights into the nature of the secondary low-affinity CGP 12177 β1-adrenoceptor binding conformation.

scientific article published on 2 April 2015

New fluorescent adenosine A1-receptor agonists that allow quantification of ligand-receptor interactions in microdomains of single living cells.

scientific article published on 24 January 2007

Novel selective β1-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease.

scientific article published on 11 April 2017

Pharmacological Analysis and Structure Determination of 7-Methylcyanopindolol-Bound β1-Adrenergic Receptor.

scientific article

Pharmacological characterization of CGP 12177 at the human beta(2)-adrenoceptor

scientific article published in October 2002

Pharmacology and direct visualisation of BODIPY-TMR-CGP: a long-acting fluorescent beta2-adrenoceptor agonist

scientific article published on May 2003

Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.

scientific article

Reporter-gene systems for the study of G-protein-coupled receptors.

scientific article

Role of key transmembrane residues in agonist and antagonist actions at the two conformations of the human beta1-adrenoceptor.

scientific article published on 7 August 2008

Salmeterol's extreme β2 selectivity is due to residues in both extracellular loops and transmembrane domains.

scientific article published on 16 October 2014

Similarity- and Substructure-Based Development of β2-Adrenergic Receptor Ligands Based on Unusual Scaffolds

scientific article published on 27 March 2017

Structure of a beta1-adrenergic G-protein-coupled receptor

scientific article

Structure-Based Discovery of Novel Ligands for the Orexin 2 Receptor

scientific article published on 25 September 2020

Synthesis and characterization of high-affinity 4,4-difluoro-4-bora-3a,4a-diaza-s-indacene-labeled fluorescent ligands for human β-adrenoceptors.

scientific article published on 16 September 2011

Synthesis and in vitro and in vivo characterization of highly β1-selective β-adrenoceptor partial agonists.

scientific article published on 10 May 2013

Temporal characteristics of cAMP response element-mediated gene transcription: requirement for sustained cAMP production

scientific article published in April 2004

The affinity and selectivity of α-adrenoceptor antagonists, antidepressants, and antipsychotics for the human α1A, α1B, and α1D-adrenoceptors

scientific article published on 01 August 2020

The pharmacological effects of the thermostabilising (m23) mutations and intra and extracellular (β36) deletions essential for crystallisation of the turkey β-adrenoceptor

scientific article published on 6 May 2011

The selectivity of beta-adrenoceptor agonists at human beta1-, beta2- and beta3-adrenoceptors

scientific article published on July 2010

The structural basis for agonist and partial agonist action on a β(1)-adrenergic receptor

scientific article

β-Blockers, heart disease and COPD: current controversies and uncertainties.

scientific article published on 7 December 2016

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