List of works - Alberto Leoni

2,5-Dimethyl-1H-pyrrole-3,4-dicarbaldehyde as a precolumn derivatization reagent for HPLC/UV detection of amino acids

scientific article published on 11 January 2010

2,7-dimethyl-3,8-dinitrodipyrazolo[1,5-a:1',5'-d]pyrazine-4,9-dione: a new labelling reagent for liquid chromatographic analysis of amino acids

article

4-Aminopyridine derivatives with antiamnesic activity

scientific article

Antitumor activity and COMPARE analysis of bis-indole derivatives

scientific article published on 28 March 2010

Antitumor activity of bis-indole derivatives

scientific article published on 04 July 2008

Antitumor activity of new substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones and 3-(5-imidazo[2,1-b]thiadiazolylmethylene)-2-indolinones: selectivity against colon tumor cells and effect on cell cycle-related events

article

Antitumor activity of new substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones and study of their effect on the cell cycle

scientific article

Antitumor activity of substituted E-3-(3,4,5-trimethoxybenzylidene)-1,3-dihydroindol-2-ones1.

scientific article published on November 2006

Ayurvedic preparation of Zingiber officinale Roscoe: effects on cardiac and on smooth muscle parameters.

scientific article

Bis-guanylhydrazone diimidazo[1,2-a:1,2-c]pyrimidine as a novel and specific G-quadruplex binding motif

scientific article published on 28 June 2010

Chemiluminescent high-throughput microassay applied to imidazo[2,1-b]thiazole derivatives as potential acetylcholinesterase and butyrylcholinesterase inhibitors

Chemopreventive and antioxidant activity of 6-substituted imidazo[2,1-b]thiazoles

scientific article published on 13 August 2013

Cystic fibrosis: a new target for 4-Imidazo[2,1-b]thiazole-1,4-dihydropyridines.

scientific article published on 13 May 2011

Design, synthesis and biological activity of a pyrrolo [2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid

scientific article published on 01 November 1998

Determination of Estragole in Fennel Herbal Teas by HS-SPME and GC–MS

article by Giulia Basaglia et al published 31 December 2013 in Analytical Letters

Determination of Phytomarkers in Pharmaceutical Preparations ofHemidesmus indicusRoots by Micellar Electrokinetic Chromatography and High-Performance Liquid Chromatography–Mass Spectrometry

Diethyl 4-(6-Chloroimidazo[2,1-b]thiazol-5-yl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate and Ethyl 4-(6-Chloroimidazo[2,1-b]thiazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxylate

Diphenidol-related diamines as novel muscarinic M4 receptor antagonists

scientific article

Effect of A-Ring Modifications on the DNA-Binding Behavior and Cytotoxicity of Pyrrolo[2,1-c][1,4]benzodiazepines†

scientific article published on 01 June 1999

Effects of new ubiquinone-imidazo[2,1-b]thiazoles on mitochondrial complex I (NADH-ubiquinone reductase) and on mitochondrial permeability transition pore

scientific article published in November 2004

Electronic nose and chiral-capillary electrophoresis in evaluation of the quality changes in commercial green tea leaves during a long-term storage

scientific article published on 9 May 2014

Imidazo[2,1-b]thiazole guanylhydrazones as RSK2 inhibitors

scientific article

Imidazo[2,1-b]thiazole system: a scaffold endowing dihydropyridines with selective cardiodepressant activity

scientific article

Inhibition of MDR1 activity and induction of apoptosis by analogues of nifedipine and diltiazem: an in vitro analysis.

scientific article

Ligand based approach to L-type calcium channel by imidazo[2,1-b]thiazole-1,4-dihydropyridines: from heart activity to brain affinity

scientific article published on 9 May 2013

N-Benzyl-2-chloroindole-3-carboxylic acids as potential anti-inflammatory agents. Synthesis and screening for the effects on human neutrophil functions and on COX1/COX2 activity

New antitumor imidazo[2,1-b]thiazole guanylhydrazones and analogues

scientific article published on 6 February 2008

New isatin derivatives with antioxidant activity

scientific article published on 28 December 2009

Novel thiazole derivatives: a patent review (2008 - 2012. Part 2).

scientific article published on 19 April 2014

Novel thiazole derivatives: a patent review (2008 - 2012; Part 1).

scientific article

Potential Antitumor Agents. 24.1Synthesis and Pharmacological Behavior of Imidazo[2,1-b]thiazole Guanylhydrazones Bearing at Least One Chlorine

scientific article published on 01 July 1996

Potential antitumor agents. 37. Synthesis and antitumor activity of guanylhydrazones from imidazo[2,1-b]thiazoles and from the new heterocyclic system thiazolo[2',3':2,3]imidazo[4,5-c]quinoline

scientific article

Substituted E-3-(2-Chloro-3-indolylmethylene)1,3-dihydroindol-2-ones with antitumor activity

scientific article published on March 2004

Substituted E-3-(2-chloro-3-indolylmethylene)1,3-dihydroindol-2-ones with antitumor activity. Effect on the cell cycle and apoptosis

scientific article published on 9 June 2007

Substituted E-3-(3-indolylmethylene)-1,3-dihydroindol-2-ones with antitumor activity. In depth study of the effect on growth of breast cancer cells

scientific article

Substituted E-3-(3-indolylmethylene)1,3-dihydroindol-2-ones with antiproliferative activity. Study of the effects on HL-60 leukemia cells

scientific article published on 3 April 2014

Synthesis and Screening for Antiacetylcholinesterase Activity of (1-Benzyl-4-oxopiperidin-3-ylidene)methylindoles and -pyrroles Related to Donepezil ⬇️

scientific article published on November 8, 2001

Synthesis and antiproliferative activity of imidazo[2,1-b][1,3,4]thiadiazole derivatives

scientific article published on 26 August 2014

Synthesis and antitubercular activity of imidazo[2,1-b]thiazoles.

scientific article published in September 2001

Synthesis and antitumor activity of 1,5,6-substituted E-3-(2-chloro-3-indolylmethylene)-1,3-dihydroindol-2-ones

scientific article published in June 2002

Synthesis and antitumor activity of a new class of pyrazolo[4,3-e]pyrrolo[1,2-a][1,4]diazepinone analogs of pyrrolo[1,4]benzodiazepines (PBDs)

scientific article published in 1993

Synthesis and antitumor activity of guanylhydrazones from 6-(2,4-dichloro-5-nitrophenyl)imidazo[2,1-b]thiazoles and 6-pyridylimidazo[2,1-b]thiazoles(1).

scientific article published in December 2006

Synthesis and chemiluminescent high throughput screening for inhibition of acetylcholinesterase activity by imidazo[2,1-b]thiazole derivatives

scientific article published on 29 August 2005

Synthesis and potential coanthracyclinic activity of pyridylmethylene and indolylmethylene lactams

article published in 1998

Synthesis of Sequence-Selective C8-Linked Pyrrolo[2,1-c][1,4]benzodiazepine DNA Interstrand Cross-Linking Agents

article

Synthesis of imidazo[2,1-b]thiazoles as herbicides

Thienylvinylindoles as inhibitors of mitochondrial NADH dehydrogenase

scientific article published on 01 July 1994

List of works by Alberto Leoni

2,5-Dimethyl-1H-pyrrole-3,4-dicarbaldehyde as a precolumn derivatization reagent for HPLC/UV detection of amino acids

2,7-dimethyl-3,8-dinitrodipyrazolo[1,5-a:1',5'-d]pyrazine-4,9-dione: a new labelling reagent for liquid chromatographic analysis of amino acids

4-Aminopyridine derivatives with antiamnesic activity

Antitumor activity and COMPARE analysis of bis-indole derivatives

Antitumor activity of bis-indole derivatives

Antitumor activity of new substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones and 3-(5-imidazo[2,1-b]thiadiazolylmethylene)-2-indolinones: selectivity against colon tumor cells and effect on cell cycle-related events

Antitumor activity of new substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones and study of their effect on the cell cycle

Antitumor activity of substituted E-3-(3,4,5-trimethoxybenzylidene)-1,3-dihydroindol-2-ones1.

Ayurvedic preparation of Zingiber officinale Roscoe: effects on cardiac and on smooth muscle parameters.

Bis-guanylhydrazone diimidazo[1,2-a:1,2-c]pyrimidine as a novel and specific G-quadruplex binding motif

Chemiluminescent high-throughput microassay applied to imidazo[2,1-b]thiazole derivatives as potential acetylcholinesterase and butyrylcholinesterase inhibitors

Chemopreventive and antioxidant activity of 6-substituted imidazo[2,1-b]thiazoles

Cystic fibrosis: a new target for 4-Imidazo[2,1-b]thiazole-1,4-dihydropyridines.

Design, synthesis and biological activity of a pyrrolo [2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid

Determination of Estragole in Fennel Herbal Teas by HS-SPME and GC–MS

Determination of Phytomarkers in Pharmaceutical Preparations ofHemidesmus indicusRoots by Micellar Electrokinetic Chromatography and High-Performance Liquid Chromatography–Mass Spectrometry

Diethyl 4-(6-Chloroimidazo[2,1-b]thiazol-5-yl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate and Ethyl 4-(6-Chloroimidazo[2,1-b]thiazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxylate

Diphenidol-related diamines as novel muscarinic M4 receptor antagonists

Effect of A-Ring Modifications on the DNA-Binding Behavior and Cytotoxicity of Pyrrolo[2,1-c][1,4]benzodiazepines†

Effects of new ubiquinone-imidazo[2,1-b]thiazoles on mitochondrial complex I (NADH-ubiquinone reductase) and on mitochondrial permeability transition pore

Electronic nose and chiral-capillary electrophoresis in evaluation of the quality changes in commercial green tea leaves during a long-term storage

Imidazo[2,1-b]thiazole guanylhydrazones as RSK2 inhibitors

Imidazo[2,1-b]thiazole system: a scaffold endowing dihydropyridines with selective cardiodepressant activity

Inhibition of MDR1 activity and induction of apoptosis by analogues of nifedipine and diltiazem: an in vitro analysis.

Ligand based approach to L-type calcium channel by imidazo[2,1-b]thiazole-1,4-dihydropyridines: from heart activity to brain affinity

N-Benzyl-2-chloroindole-3-carboxylic acids as potential anti-inflammatory agents. Synthesis and screening for the effects on human neutrophil functions and on COX1/COX2 activity

New antitumor imidazo[2,1-b]thiazole guanylhydrazones and analogues

New isatin derivatives with antioxidant activity

Novel thiazole derivatives: a patent review (2008 - 2012. Part 2).

Novel thiazole derivatives: a patent review (2008 - 2012; Part 1).

Potential Antitumor Agents. 24.1Synthesis and Pharmacological Behavior of Imidazo[2,1-b]thiazole Guanylhydrazones Bearing at Least One Chlorine

Potential antitumor agents. 37. Synthesis and antitumor activity of guanylhydrazones from imidazo[2,1-b]thiazoles and from the new heterocyclic system thiazolo[2',3':2,3]imidazo[4,5-c]quinoline

Substituted E-3-(2-Chloro-3-indolylmethylene)1,3-dihydroindol-2-ones with antitumor activity

Substituted E-3-(2-chloro-3-indolylmethylene)1,3-dihydroindol-2-ones with antitumor activity. Effect on the cell cycle and apoptosis

Substituted E-3-(3-indolylmethylene)-1,3-dihydroindol-2-ones with antitumor activity. In depth study of the effect on growth of breast cancer cells

Substituted E-3-(3-indolylmethylene)1,3-dihydroindol-2-ones with antiproliferative activity. Study of the effects on HL-60 leukemia cells

Synthesis and Screening for Antiacetylcholinesterase Activity of (1-Benzyl-4-oxopiperidin-3-ylidene)methylindoles and -pyrroles Related to Donepezil ⬇️

Synthesis and antiproliferative activity of imidazo[2,1-b][1,3,4]thiadiazole derivatives

Synthesis and antitubercular activity of imidazo[2,1-b]thiazoles.

Synthesis and antitumor activity of 1,5,6-substituted E-3-(2-chloro-3-indolylmethylene)-1,3-dihydroindol-2-ones

Synthesis and antitumor activity of a new class of pyrazolo[4,3-e]pyrrolo[1,2-a][1,4]diazepinone analogs of pyrrolo[1,4]benzodiazepines (PBDs)

Synthesis and antitumor activity of guanylhydrazones from 6-(2,4-dichloro-5-nitrophenyl)imidazo[2,1-b]thiazoles and 6-pyridylimidazo[2,1-b]thiazoles(1).

Synthesis and chemiluminescent high throughput screening for inhibition of acetylcholinesterase activity by imidazo[2,1-b]thiazole derivatives

Synthesis and potential coanthracyclinic activity of pyridylmethylene and indolylmethylene lactams

Synthesis of Sequence-Selective C8-Linked Pyrrolo[2,1-c][1,4]benzodiazepine DNA Interstrand Cross-Linking Agents

Synthesis of imidazo[2,1-b]thiazoles as herbicides

Thienylvinylindoles as inhibitors of mitochondrial NADH dehydrogenase