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List of works by George Karageorgis

A novel evolutionary approach for the discovery of small bioactive molecules ⬇️

doctoral thesis

Activity-Directed Synthesis with Intermolecular Reactions: Development of a Fragment into a Range of Androgen Receptor Agonists ⬇️

scientific article published on 11 September 2015

Activity-Directed Synthesis with Intermolecular Reactions: Development of a Fragment into a Range of Androgen Receptor Agonists

article

Chromopynones are pseudo natural product glucose uptake inhibitors targeting glucose transporters GLUT-1 and -3 ⬇️

Efficient discovery of bioactive scaffolds by activity-directed synthesis ⬇️

scientific article published on 24 August 2014

Frontispiece: Activity-Directed Synthesis with Intermolecular Reactions: Development of a Fragment into a Range of Androgen Receptor Agonists

article

Frontispiz: Activity-Directed Synthesis with Intermolecular Reactions: Development of a Fragment into a Range of Androgen Receptor Agonists

article

Guided by Evolution: Biology-Oriented Synthesis of Bioactive Compound Classes

scholarly article by Herbert Waldmann & George Karageorgis published 11 October 2018 in Synthesis

Inhibition of Glucose Transporters and Glutaminase Synergistically Impairs Tumor Cell Growth

scientific article published on 11 July 2019

Principle and design of pseudo-natural products

scientific article published on 03 February 2020

Realisation of small molecule libraries based on frameworks distantly related to natural products ⬇️

scientific article published on 12 April 2018

Synthesis of Indomorphan Pseudo-Natural Product Inhibitors of Glucose Transporters GLUT-1 and -3

scientific article published on 07 October 2019

The Pseudo Natural Product Myokinasib Is a Myosin Light Chain Kinase 1 Inhibitor with Unprecedented Chemotype

scientific article published on 24 January 2019

Translation of innovative chemistry into screening libraries: an exemplar partnership from the European Lead Factory ⬇️

scientific article published on 09 May 2018

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