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List of works by Frédéric Bihel

A Yeast/Drosophila Screen to Identify New Compounds Overcoming Frataxin Deficiency

scientific article published on 11 October 2015

Access to 4-alkylaminopyridazine derivatives via nitrogen-assisted regioselective Pd-catalyzed reactions

scientific article published on 27 October 2014

Aminoguanidine hydrazone derivatives as non-peptide NPFF1 receptor antagonists reverse opioid induced hyperalgesia

scientific article published on 4 May 2018

CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors

scientific article published on 7 May 2015

CamKII inhibitors reduce mitotic instability, connexon anomalies and progression of the in vivo behavioral phenotype in transgenic animals expressing a mutated Gjb1 gene

scientific article

Design and validation of a homogeneous time-resolved fluorescence cell-based assay targeting the ligand-gated ion channel 5-HT3A.

scientific article published on 18 May 2015

Development of Dipeptidic hGPR54 Agonists.

scientific article published on 26 August 2016

Development of a peptidomimetic antagonist of neuropeptide FF receptors for the prevention of opioid-induced hyperalgesia

scientific article published on 7 February 2015

Development of sub-nanomolar dipeptidic ligands of neuropeptide FF receptors

scientific article published on 17 October 2012

Diastereoselective Synthesis of Nonplanar 3-Amino-1,2,4-oxadiazine Scaffold: Structure Revision of Alchornedine

scientific article published on 16 November 2020

Direct guanidinylation of aryl and heteroaryl halides via copper-catalyzed cross-coupling reaction

scientific article published on 13 December 2011

Discovery of a Subnanomolar helical D-tridecapeptide inhibitor of gamma-secretase

scientific article published on 01 July 2004

Effects of systematic N-terminus deletions and benzoylations of endogenous RF-amide peptides on NPFF1R, NPFF2R, GPR10, GPR54 and GPR103

scientific article published on 23 July 2015

Erratum to: CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors

scientific article published on 25 January 2016

Fukuyama Cross-Coupling Approach to Isoprekinamycin: Discovery of the Highly Active and Bench-Stable Palladium Precatalyst POxAP

scientific article published on 18 January 2019

Heteroarylguanidines as Allosteric Modulators of ASIC1a and ASIC3 Channels

scientific article published on 22 March 2018

Induction of ATP Release, PPIX Transport, and Cholesterol Uptake by Human Red Blood Cells Using a New Family of TSPO Ligands

scholarly article by Irene Marginedas-Freixa published in October 2018

Involvement of neuropeptide FF receptors in neuroadaptive responses to acute and chronic opiate treatments.

scientific article published on January 2012

Microwave-assisted cyclic amidine synthesis using TiCl4

scientific article published on 12 July 2006

Mitochondria modulatory effects of new TSPO ligands in a cellular model of tauopathies

scientific article published on 13 October 2019

Neuropeptide FF receptors as novel targets for limbic seizure attenuation

scientific article published on 9 May 2015

New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.

scientific article published on March 2001

New PDE4 inhibitors based on pharmacophoric similarity between papaverine and tofisopam

scientific article published on 12 August 2011

Nucleophilic substitution of azide acting as a pseudo leaving group: one-step synthesis of various aza heterocycles

scientific article published on 24 October 2013

Opioid adjuvant strategy: improving opioid effectiveness

scientific article published on 22 February 2016

Pharmacological characterization of the mouse NPFF2 receptor.

scientific article published on 26 November 2009

Structure-activity relationship study around guanabenz identifies two derivatives retaining antiprion activity but having lost α2-adrenergic receptor agonistic activity

scientific article published on 22 September 2014

Substituted thiazolamide coupled to a redox delivery system: a new gamma-secretase inhibitor with enhanced pharmacokinetic profile.

scientific article published on 10 January 2005

Synthesis and antiproliferative effects of 5,6-disubstituted Pyridazin-3(2H)-ones designed as conformationally constrained combretastatin A-4 Analogues

scientific article published on September 2013

Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new beta-amyloid peptide production inhibitors and their activities on various classes of protease

scientific article

The effect of neuropeptide FF in the amygdala kindling model.

scientific article

The long-lasting love affair between the budding yeast Saccharomyces cerevisiae and the Epstein-Barr virus

scientific article published on 27 August 2015

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds.

scientific article published on 4 October 2017

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