Search filters

List of works by Gang Cheng

A base-promoted tandem reaction of 3-(1-alkynyl)chromones with 1,3-dicarbonyl compounds: an efficient approach to functional xanthones

scientific article published on 01 January 2009

Covalent docking modelling-based discovery of tripeptidyl epoxyketone proteasome inhibitors composed of aliphatic-heterocycles

scientific article published on 26 December 2018

Design, synthesis, and biological activity of diaryl ether inhibitors of Toxoplasma gondii enoyl reductase

scientific article

Design, synthesis, and molecular docking study of 3H-imidazole[4,5-c]pyridine derivatives as CDK2 inhibitors

scientific article published on 30 April 2018

Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as Orally Active, Low hERG Blocking Akt Inhibitors via Conformational Restriction and Structure-Based Design

scientific article published on 24 July 2019

Discovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors

scientific article published on 07 July 2019

Discrimination of potent inhibitors of Toxoplasma gondii enoyl-acyl carrier protein reductase by a thermal shift assay

scientific article published on 13 December 2013

Identification of new NIK inhibitors by discriminatory analysis-based molecular docking and biological evaluation

scientific article published on 22 May 2019

Inhibition of 1-Deoxy- d -Xylulose-5-Phosphate Reductoisomerase by Lipophilic Phosphonates: SAR, QSAR, and Crystallographic Studies

scientific article

Novel N-benzoyl-2-hydroxybenzamide disrupts unique parasite secretory pathway

scientific article

One-pot Synthesis of 6-Aza-chromone Derivatives Through Cascade Carbonylation-Sonogashira-Cyclization.

scientific article

One-pot synthesis of furocoumarins through cascade addition-cyclization-oxidation

scientific article published on 07 June 2007

Rehmannia glutinosa Libosch Extracts Prevent Bone Loss and Architectural Deterioration and Enhance Osteoblastic Bone Formation by Regulating the IGF-1/PI3K/mTOR Pathway in Streptozotocin-Induced Diabetic Rats

scientific article published on 15 August 2019

Resveratrol-maltol hybrids as multi-target-directed agents for Alzheimer's disease

scientific article published on 09 August 2018

Selective Inhibitors of Histone Methyltransferase DOT1L: Design, Synthesis, and Crystallographic Studies

scientific article

Storable N-phenylcarbamate palladacycles for rapid functionalization of an alkyne-encoded protein

scientific article

Storable palladacycles for selective functionalization of alkyne-containing proteins

scientific article published on August 2013

Structures of 1-Deoxy-D-Xylulose-5-Phosphate Reductoisomerase/Lipophilic Phosphonate Complexes

scientific article

Synthesis and Site-Specific Incorporation of Red-Shifted Azobenzene Amino Acids into Proteins

scientific article

Synthesis and structure-activity relationship investigation of adenosine-containing inhibitors of histone methyltransferase DOT1L

scientific article

Three-component, one-pot reaction for the combinatorial synthesis of 1,3,4-substituted pyrazoles

scientific article published on 01 May 2006

Three-component, one-pot synthesis of novel 2,4-substituted 5-azolylthiopyrimidine library for screening against anti-influenza virus A.

scientific article

Two efficient cascade reactions to synthesize substituted furocoumarins

scientific article published on 28 May 2008