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List of works by Achim Schlapbach

A novel Pd-catalyzed cyclization reaction of ureas for the synthesis of dihydroquinazolinone p38 kinase inhibitors.

scientific article published in January 2004

An allosteric MALT1 inhibitor is a molecular corrector rescuing function in an immunodeficient patient

scientific article published on 28 January 2019

Design and preparation of 2-benzamido-pyrimidines as inhibitors of IKK

scientific article published on 19 October 2005

Discovery of a novel class of highly potent inhibitors of the p53-MDM2 interaction by structure-based design starting from a conformational argument

scientific article

Identification of human kinases involved in hepatitis C virus replication by small interference RNA library screening.

scientific article

In vitro and in vivo characterization of a novel, highly potent p53-MDM2 inhibitor

scientific article published on 26 August 2018

In vivo and in vitro SAR of tetracyclic MAPKAP-K2 (MK2) inhibitors. Part II

scientific article

Low-molecular-weight MK2 inhibitors: a tough nut to crack!

scientific article published on October 2009

Modulating ADME Properties by Fluorination: MK2 Inhibitors with Improved Oral Exposure.

scientific article published on 20 March 2018

N -aryl-piperidine-4-carboxamides as a novel class of potent inhibitors of MALT1 proteolytic activity

scientific article published on 09 May 2018

Novel 3-aminopyrazole inhibitors of MK-2 discovered by scaffold hopping strategy

scientific article

Novel CCR1 antagonists with oral activity in the mouse collagen induced arthritis

scientific article published on 28 September 2005

Pyrrolo-pyrimidones: a novel class of MK2 inhibitors with potent cellular activity.

scientific article

The T-cell fingerprint of MALT1 paracaspase revealed by selective inhibition.

scientific article published on 21 December 2017

The role of interstitial macrophages in nephropathy of type 2 diabetic db/db mice.

scientific article published on April 2007

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