List of works by Juraj Velcicky

An efficient organometallic approach to new carbocyclic nucleoside analogues

scientific article published on 01 February 2002

Design and synthesis of potent and orally active GPR4 antagonists with modulatory effects on nociception, inflammation, and angiogenesis

scientific article published on 29 June 2017

Development of Selective, Orally Active GPR4 Antagonists with Modulatory Effects on Nociception, Inflammation, and Angiogenesis.

scientific article published on 26 April 2017

Discovery and Optimization of Novel SUCNR1 Inhibitors: Design of Zwitterionic Derivatives with a Salt Bridge for the Improvement of Oral Exposure

scientific article published on 28 August 2020

Discovery of the First Potent, Selective, and Orally Bioavailable Signal Peptide Peptidase-Like 2a (SPPL2a) Inhibitor Displaying Pronounced Immunomodulatory Effects In Vivo.

scientific article

In vivo and in vitro SAR of tetracyclic MAPKAP-K2 (MK2) inhibitors. Part II

scientific article

Iron-containing nucleoside analogues with pronounced apoptosis-inducing activity.

scientific article published on March 2004

Modulating ADME Properties by Fluorination: MK2 Inhibitors with Improved Oral Exposure.

scientific article published on 20 March 2018

Novel 3-aminopyrazole inhibitors of MK-2 discovered by scaffold hopping strategy

scientific article

Nucleoside analogues with a 1,3-diene-Fe(CO)3 substructure: stereoselective synthesis, configurational assignment, and apoptosis-inducing activity.

scientific article published on 9 August 2013

Palladium-catalyzed cyanomethylation of aryl halides through domino Suzuki coupling-isoxazole fragmentation

scientific article published on 19 April 2011

Pyrrolo-pyrimidones: a novel class of MK2 inhibitors with potent cellular activity.

scientific article

Total synthesis of (-)- and ent-(+)-vindorosine: tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition of 1,3,4-oxadiazoles

scientific article published on 01 January 2006

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