List of works - Pedro Merino

(+)-Methyl (1R,2S)-2-{[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-1-phenylcyclopropanecarboxylate [(+)-MR200] Derivatives as Potent and Selective Sigma Receptor Ligands: Stereochemistry and Pharmacological Properties

scientific article published on 8 December 2017

1,3-dipolar cycloaddition of furfuryl nitrones with acrylates. A convenient approach to protected 4-hydroxypyroglutamic acids

scientific article published on 01 March 2000

A new entry to glycosylamines

scientific article published on 01 June 1997

An investigation of the Lewis acid mediated 1,3-dipolar cycloaddition between N-benzyl-C-(2-pyridyl)nitrone and allylic alcohol. Direct entry to isoxazolidinyl C-nucleosides.

scientific article published in July 2003

Azomethine Ylides from Nitrones: Using Catalytic nBuLi for the Totally Stereoselective Synthesis of trans-2-Alkyl-3-oxazolines

scientific article published on 3 June 2016

Catalytic Enantioselective Hydrophosphonylation of Aldehydes and Imines

Chemical synthesis of heterocyclic-sugar nucleoside analogues

scientific article published on June 2010

Correction to "Self-Regeneration of Chirality with l-Cysteine through 1,3-Dipolar Cycloadditions between Diazoalkanes and Enantiomerically Pure Thiazolines: Experimental and Computational Studies"

scientific article published on 18 May 2018

Current developments in the synthesis and biological activity of aza-C-nucleosides: immucillins and related compounds.

scientific article published on January 2008

Dissecting the Structural and Chemical Determinants of the "Open-to-Closed" Motion in the Mannosyltransferase PimA from Mycobacteria

scientific article published on 04 August 2020

Enantiodivergent synthesis of D- and L-erythro-sphingosines through Mannich-type reactions of N-benzyl-2,3-O-isopropylidene-D-glyceraldehyde nitrone

scientific article published on 01 June 2006

Enantioselective 1,3-dipolar cycloaddition of nitrones to methacrolein catalyzed by (eta5-C5Me5)M{(R)-prophos} containing complexes (M = Rh, Ir; (R)-prophos = 1,2-bis(diphenylphosphino)propane): on the origin of the enantioselectivity

scientific article published in September 2005

Enantioselective Synthesis of Tropanes: Brønsted Acid Catalyzed Pseudotransannular Desymmetrization

scientific article published on 10 February 2020

Enantioselective Synthesis, DFT Calculations, and Preliminary Antineoplastic Activity of Dibenzo 1-Azaspiro[4.5]decanes on Drug-Resistant Leukemias

scientific article published on 01 February 2019

Expanding the limits of organoboron chemistry: synthesis of functionalized arylboronates

scientific article published on 01 September 2010

Glycomimetics Targeting Glycosyltransferases: Synthetic, Computational and Structural Studies of Less-Polar Conjugates

scientific article

Heterocyclic nucleosides: chemical synthesis and biological properties.

scientific article

Inhibitors against Fungal Cell Wall Remodeling Enzymes.

scientific article

Iterative organometallic addition to chiral hydroxylated cyclic nitrones: highly stereoselective syntheses of alpha,alpha'- and alpha,alpha-substituted hydroxypyrrolidines

scientific article published on 01 October 2003

Mechanistic Insights into the Mode of Action of Bifunctional Pyrrolidine-Squaramide-Derived Organocatalysts

scientific article

New concise total synthesis of (+)-lentiginosine and some structural analogues

scientific article published on 01 August 2005

Organocatalyzed asymmetric alpha-aminoxylation of aldehydes and ketones--an efficient access to enantiomerically pure alpha-hydroxycarbonyl compounds, diols, and even amino alcohols

scientific article published on 01 June 2004

Recent progress on fucosyltransferase inhibitors.

scientific article published on December 2012

Self-Regeneration of Chirality with l-Cysteine through 1,3-Dipolar Cycloadditions between Diazoalkanes and Enantiomerically Pure Thiazolines: Experimental and Computational Studies

scientific article published on 14 March 2018

Sequential Metal-Free Thermal 1,3-Dipolar Cycloaddition of Unactivated Azomethine Ylides

scientific article published on 06 June 2018

Sequential nucleophilic addition/intramolecular cycloaddition to chiral nonracemic cyclic nitrones: a highly stereoselective approach to polyhydroxynortropane alkaloids

scientific article published on 29 April 2011

Stereodivergent approaches to the synthesis of isoxazolidine analogues of alpha-amino acid nucleosides. Total synthesis of isoxazolidinyl deoxypolyoxin C and uracil polyoxin C

scientific article published on 01 September 2000

Stereoselective hydride transfer by aryl-alcohol oxidase, a member of the GMC superfamily

scientific article published on 23 January 2012

Stereoselective synthesis and biological evaluations of novel 3'-deoxy-4'-azaribonucleosides as inhibitors of hepatitis C virus RNA replication

scientific article published on July 2009

Structural Insights into the Mechanism of Protein O-Fucosylation

scientific article published in 2011

Synthesis of Enantiopure Constrained α,β-Cycloaliphatic Cystines via Diels-Alder Reaction with Homochiral Thiazolines

scientific article published on 27 September 2018

Synthesis of O- and C-glycosides derived from β-(1,3)-D-glucans.

scientific article published on 30 July 2013

Synthesis, Biological and In Silico Evaluation of Pure Nucleobase-Containing Spiro (Indane-Isoxazolidine) Derivatives as Potential Inhibitors of MDM2-p53 Interaction

scientific article published on 10 August 2019

The complete characterization of a rhodium Lewis acid-dipolarophile complex as an intermediate for the enantioselective catalytic 1,3-dipolar cycloaddition of C,N-diphenylnitrone to methacrolein

scientific article published in March 2004

Thiourea catalyzed organocatalytic enantioselective Michael addition of diphenyl phosphite to nitroalkenes

scientific article published on 25 February 2011

Transient and intermediate carbocations in ruthenium tetroxide oxidation of saturated rings

scientific article published on 11 July 2019

Truncated reverse isoxazolidinyl nucleosides: a new class of allosteric HIV-1 reverse transcriptase inhibitors

scientific article

Tunable diastereoselection of biased rigid systems by Lewis acid induced conformational effects: a rationalization of the vinylation of cyclic nitrones en route to polyhydroxylated pyrrolidines.

scientific article published on August 2010

UDP-GlcNAc Analogues as Inhibitors of O -GlcNAc Transferase (OGT): Spectroscopic, Computational, and Biological Studies

scientific article published on 30 April 2018

[2n2π + 2n2π] cycloadditions: an alternative to forbidden [4π + 4π] processes. The case of nitrone dimerization.

scientific article

List of works by Pedro Merino

(+)-Methyl (1R,2S)-2-{[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-1-phenylcyclopropanecarboxylate [(+)-MR200] Derivatives as Potent and Selective Sigma Receptor Ligands: Stereochemistry and Pharmacological Properties

1,3-dipolar cycloaddition of furfuryl nitrones with acrylates. A convenient approach to protected 4-hydroxypyroglutamic acids

A new entry to glycosylamines

An investigation of the Lewis acid mediated 1,3-dipolar cycloaddition between N-benzyl-C-(2-pyridyl)nitrone and allylic alcohol. Direct entry to isoxazolidinyl C-nucleosides.

Azomethine Ylides from Nitrones: Using Catalytic nBuLi for the Totally Stereoselective Synthesis of trans-2-Alkyl-3-oxazolines

Catalytic Enantioselective Hydrophosphonylation of Aldehydes and Imines

Chemical synthesis of heterocyclic-sugar nucleoside analogues

Correction to "Self-Regeneration of Chirality with l-Cysteine through 1,3-Dipolar Cycloadditions between Diazoalkanes and Enantiomerically Pure Thiazolines: Experimental and Computational Studies"

Current developments in the synthesis and biological activity of aza-C-nucleosides: immucillins and related compounds.

Dissecting the Structural and Chemical Determinants of the "Open-to-Closed" Motion in the Mannosyltransferase PimA from Mycobacteria

Enantiodivergent synthesis of D- and L-erythro-sphingosines through Mannich-type reactions of N-benzyl-2,3-O-isopropylidene-D-glyceraldehyde nitrone

Enantioselective 1,3-dipolar cycloaddition of nitrones to methacrolein catalyzed by (eta5-C5Me5)M{(R)-prophos} containing complexes (M = Rh, Ir; (R)-prophos = 1,2-bis(diphenylphosphino)propane): on the origin of the enantioselectivity

Enantioselective Synthesis of Tropanes: Brønsted Acid Catalyzed Pseudotransannular Desymmetrization

Enantioselective Synthesis, DFT Calculations, and Preliminary Antineoplastic Activity of Dibenzo 1-Azaspiro[4.5]decanes on Drug-Resistant Leukemias

Expanding the limits of organoboron chemistry: synthesis of functionalized arylboronates

Glycomimetics Targeting Glycosyltransferases: Synthetic, Computational and Structural Studies of Less-Polar Conjugates

Heterocyclic nucleosides: chemical synthesis and biological properties.

Inhibitors against Fungal Cell Wall Remodeling Enzymes.

Iterative organometallic addition to chiral hydroxylated cyclic nitrones: highly stereoselective syntheses of alpha,alpha'- and alpha,alpha-substituted hydroxypyrrolidines

Mechanistic Insights into the Mode of Action of Bifunctional Pyrrolidine-Squaramide-Derived Organocatalysts

New concise total synthesis of (+)-lentiginosine and some structural analogues

Organocatalyzed asymmetric alpha-aminoxylation of aldehydes and ketones--an efficient access to enantiomerically pure alpha-hydroxycarbonyl compounds, diols, and even amino alcohols

Recent progress on fucosyltransferase inhibitors.

Self-Regeneration of Chirality with l-Cysteine through 1,3-Dipolar Cycloadditions between Diazoalkanes and Enantiomerically Pure Thiazolines: Experimental and Computational Studies

Sequential Metal-Free Thermal 1,3-Dipolar Cycloaddition of Unactivated Azomethine Ylides

Sequential nucleophilic addition/intramolecular cycloaddition to chiral nonracemic cyclic nitrones: a highly stereoselective approach to polyhydroxynortropane alkaloids

Stereodivergent approaches to the synthesis of isoxazolidine analogues of alpha-amino acid nucleosides. Total synthesis of isoxazolidinyl deoxypolyoxin C and uracil polyoxin C

Stereoselective hydride transfer by aryl-alcohol oxidase, a member of the GMC superfamily

Stereoselective synthesis and biological evaluations of novel 3'-deoxy-4'-azaribonucleosides as inhibitors of hepatitis C virus RNA replication

Structural Insights into the Mechanism of Protein O-Fucosylation

Synthesis of Enantiopure Constrained α,β-Cycloaliphatic Cystines via Diels-Alder Reaction with Homochiral Thiazolines

Synthesis of O- and C-glycosides derived from β-(1,3)-D-glucans.

Synthesis, Biological and In Silico Evaluation of Pure Nucleobase-Containing Spiro (Indane-Isoxazolidine) Derivatives as Potential Inhibitors of MDM2-p53 Interaction

The complete characterization of a rhodium Lewis acid-dipolarophile complex as an intermediate for the enantioselective catalytic 1,3-dipolar cycloaddition of C,N-diphenylnitrone to methacrolein

Thiourea catalyzed organocatalytic enantioselective Michael addition of diphenyl phosphite to nitroalkenes

Transient and intermediate carbocations in ruthenium tetroxide oxidation of saturated rings

Truncated reverse isoxazolidinyl nucleosides: a new class of allosteric HIV-1 reverse transcriptase inhibitors

Tunable diastereoselection of biased rigid systems by Lewis acid induced conformational effects: a rationalization of the vinylation of cyclic nitrones en route to polyhydroxylated pyrrolidines.

UDP-GlcNAc Analogues as Inhibitors of O -GlcNAc Transferase (OGT): Spectroscopic, Computational, and Biological Studies

[2n2π + 2n2π] cycloadditions: an alternative to forbidden [4π + 4π] processes. The case of nitrone dimerization.