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List of works by Matthias Schmidt

Application of docking and QM/MM-GBSA rescoring to screen for novel Myt1 kinase inhibitors

scientific article

Augmented reversible photoswitching of drug-target interaction through "surface borrowing".

scientific article

Computer-aided design, synthesis and biological characterization of novel inhibitors for PKMYT1

scientific article published on 24 October 2018

Evaluation of potential Myt1 kinase inhibitors by TR-FRET based binding assay

scientific article

Identification of PKMYT1 inhibitors by screening the GSK published protein kinase inhibitor set I and II

scientific article published on 20 June 2018

Identification of peptidic substrates for the human kinase Myt1 using peptide microarrays

scientific article published on 19 May 2015

In vitro and in silico studies on substrate recognition and acceptance of human PKMYT1, a Cdk1 inhibitory kinase

scientific article published on 23 November 2011

New 1,3-dioxolane and 1,3-dioxane derivatives as effective modulators to overcome multidrug resistance

scientific article published on 19 January 2007

New modified single chained glycolipids. Part 1: synthesis of deoxy and partially O-methylated glycolipids with or without a sulfur containing spacer.

scientific article

Regulation of G2/M Transition by Inhibition of WEE1 and PKMYT1 Kinases.

scientific article published on 23 November 2017

Structural basis for the inhibition of histone deacetylase 8 (HDAC8), a key epigenetic player in the blood fluke Schistosoma mansoni

scientific article

Structure-Based Design and Biological Characterization of Selective Histone Deacetylase 8 (HDAC8) Inhibitors with Anti-Neuroblastoma Activity

scientific article published on 30 November 2017

Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as Sm HDAC8 Inhibitors for the Treatment of Schistosomiasis

scientific article published on 4 July 2018

Synthesis, biological characterisation and structure activity relationships of aromatic bisamidines active against Plasmodium falciparum

scientific article published on 23 December 2016

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