Search filters

List of works by Peter Goekjian

6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury

scientific article published on 10 October 2017

Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition

scientific article published on December 2006

Expeditive synthesis of trithiotriazine-cored glycoclusters and inhibition of Pseudomonas aeruginosa biofilm formation

scientific article

Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors

scientific article

Glycosylated asterisks are among the most potent low valency inducers of Concanavalin A aggregation

scientific article

Identification of potential cellular targets of aloisine A by affinity chromatography

scientific article published on 18 June 2009

NMR screening applied to the fragment-based generation of inhibitors of creatine kinase exploiting a new interaction proximate to the ATP binding site.

scientific article

RET kinase inhibitors: a review of recent patents (2012-2015).

scientific article published on 20 September 2016

Sibiriline, a new small chemical inhibitor of receptor-interacting protein kinase 1, prevents immune-dependent hepatitis

scientific article published on 17 July 2017

Synthesis and biological evaluation of benzo[4,5]imidazo[1,2-c]pyrimidine and benzo[4,5]imidazo[1,2-a]pyrazine derivatives as anaplastic lymphoma kinase inhibitors

scientific article published on 10 January 2014

Synthesis of substituted exo-glucals via a modified Julia olefination and identification as selective β-glucosidase inhibitors

scientific article published on 01 January 2014

Targeting RNA structure in SMN2 reverses spinal muscular atrophy molecular phenotypes.

scientific article

Thienoquinolines as novel disruptors of the PKCε/RACK2 protein-protein interaction

scientific article published on 08 April 2014

Total synthesis of bistramide A and its 36(Z) isomers: differential effect on cell division, differentiation, and apoptosis.

scientific article published on 26 April 2012