List of works - Ross McGeary

3-mercapto-1,2,4-triazoles and N-acylated thiosemicarbazides as metallo-β-lactamase inhibitors

scientific article

A Backbone Linker for BOC-Based Peptide Synthesis and On-Resin Cyclization: Synthesis of Stylostatin 1†,§

scientific article published on 01 April 1999

Binuclear metallohydrolases: complex mechanistic strategies for a simple chemical reaction.

scientific article published on 14 June 2012

Captopril analogues as metallo-β-lactamase inhibitors.

scientific article published on 4 February 2016

Crystal structure of Mycobacterium tuberculosis ketol-acid reductoisomerase at 1.0 Å resolution - a potential target for anti-tuberculosis drug discovery

scientific article

Cyclodextrin-crosslinked poly(acrylic acid): Synthesis, physicochemical characterization and controlled release of diflunisal and fluconazole from hydrogels.

scientific article published on 14 January 2013

Cyclodextrin-crosslinked poly(acrylic acid): adhesion and controlled release of diflunisal and fluconazole from solid dosage forms.

scientific article published on 11 January 2013

Design, synthesis, and in vitro and biological evaluation of potent amino acid-derived thiol inhibitors of the metallo-β-lactamase IMP-1.

scientific article published on 9 March 2016

Development of a liposaccharide-based delivery system and its application to the design of group A streptococcal vaccines.

scientific article

Fibroblast growth factor 1: a key regulator of human adipogenesis.

scientific article published on December 2004

Identification and characterization of an unusual metallo-β-lactamase from Serratia proteamaculans.

scientific article

Identification of novel target sites and an inhibitor of the dengue virus E protein

scientific article published on 25 February 2009

Identification of purple acid phosphatase inhibitors by fragment-based screening: promising new leads for osteoporosis therapeutics

scientific article

Inhibition of purple acid phosphatase with alpha-alkoxynaphthylmethylphosphonic acids

scientific article published on 05 November 2008

Metal chelation, radical scavenging and inhibition of Aβ₄₂ fibrillation by food constituents in relation to Alzheimer's disease.

scientific article published on 26 November 2015

Molecular packing of functionalized fluorinated lipids in Langmuir monolayers

scientific article

Multifunctional Analogs of Kynurenic Acid for the Treatment of Alzheimer's Disease: Synthesis, Pharmacology, and Molecular Modeling Studies

scientific article published on 21 August 2017

Penicillin inhibitors of purple acid phosphatase

scientific article published on 04 February 2012

Pharmacokinetics of doxorubicinol in dogs

scientific article published on 01 October 2006

Saponins from Quillaja saponaria Molina: Isolation, Characterization and Ability to Form Immuno Stimulatory Complexes (ISCOMs)

scientific article published in October 2006

Simultaneous determination of thymine and its sequential catabolites dihydrothymine and β-ureidoisobutyrate in human plasma and urine using liquid chromatography-tandem mass spectrometry with pharmacokinetic application

scientific article

Simultaneous liquid chromatographic determination of doxorubicin and its major metabolite doxorubicinol in parrot plasma.

scientific article published on 15 September 2005

Small Peptides Do Not Inhibit Human Non-Pancreatic Secretory Phospholipase-A2 (Type IIA)

scientific article published on 01 August 2000

Suramin: clinical uses and structure-activity relationships.

scientific article

Synthesis and evaluation of novel purple acid phosphatase inhibitors

scientific article published on 13 November 2018

Synthesis and kinetic testing of new inhibitors for a metallo-β-lactamase from Klebsiella pneumonia and Pseudomonas aeruginosa.

scientific article published on 21 October 2011

Synthesis and kinetic testing of tetrahydropyrimidine-2-thione and pyrrole derivatives as inhibitors of the metallo-β-lactamase from Klebsiella pneumonia and Pseudomonas aeruginosa

scientific article published on 23 July 2012

Synthesis and polymerization studies of organic-soluble eumelanins.

scientific article

Synthesis of Nickel-Chelating Fluorinated Lipids for Protein Monolayer Crystallizations

scientific article published on 01 February 2009

Synthesis of a series of carbon-14 labeled tetrahydropyrido[4,3-d]pyrimidin-4(3H)-ones

scientific article published on 29 August 2013

Synthesis of cationic derivatives of Quil A and the preparation of cationic immune-stimulating complexes (ISCOMs).

scientific article published on 16 April 2009

Synthesis, modelling and kinetic assays of potent inhibitors of purple acid phosphatase

scientific article published on 13 March 2011

The applications of binuclear metallohydrolases in medicine: recent advances in the design and development of novel drug leads for purple acid phosphatases, metallo-β-lactamases and arginases.

scientific article published on 08 February 2014

The development and application of a novel safety-catch linker for BOC-based assembly of libraries of cyclic peptides.

scientific article

The identification of new metallo-β-lactamase inhibitor leads from fragment-based screening.

scientific article

The role of Zn-OR and Zn-OH nucleophiles and the influence of para-substituents in the reactions of binuclear phosphatase mimetics

scientific article

Toxicokinetics of the active doxorubicin metabolite, doxorubicinol, in sulphur-crested cockatoos (Cacatua galerita)

scientific article published on 02 January 2007

‘Click’ assembly of glycoclusters and discovery of a trehalose analogue that retards Aβ40 aggregation and inhibits Aβ40-induced neurotoxicity

scientific article published in September 2014

List of works by Ross McGeary

3-mercapto-1,2,4-triazoles and N-acylated thiosemicarbazides as metallo-β-lactamase inhibitors

A Backbone Linker for BOC-Based Peptide Synthesis and On-Resin Cyclization: Synthesis of Stylostatin 1†,§

Binuclear metallohydrolases: complex mechanistic strategies for a simple chemical reaction.

Captopril analogues as metallo-β-lactamase inhibitors.

Crystal structure of Mycobacterium tuberculosis ketol-acid reductoisomerase at 1.0 Å resolution - a potential target for anti-tuberculosis drug discovery

Cyclodextrin-crosslinked poly(acrylic acid): Synthesis, physicochemical characterization and controlled release of diflunisal and fluconazole from hydrogels.

Cyclodextrin-crosslinked poly(acrylic acid): adhesion and controlled release of diflunisal and fluconazole from solid dosage forms.

Design, synthesis, and in vitro and biological evaluation of potent amino acid-derived thiol inhibitors of the metallo-β-lactamase IMP-1.

Development of a liposaccharide-based delivery system and its application to the design of group A streptococcal vaccines.

Fibroblast growth factor 1: a key regulator of human adipogenesis.

Identification and characterization of an unusual metallo-β-lactamase from Serratia proteamaculans.

Identification of novel target sites and an inhibitor of the dengue virus E protein

Identification of purple acid phosphatase inhibitors by fragment-based screening: promising new leads for osteoporosis therapeutics

Inhibition of purple acid phosphatase with alpha-alkoxynaphthylmethylphosphonic acids

Metal chelation, radical scavenging and inhibition of Aβ₄₂ fibrillation by food constituents in relation to Alzheimer's disease.

Molecular packing of functionalized fluorinated lipids in Langmuir monolayers

Multifunctional Analogs of Kynurenic Acid for the Treatment of Alzheimer's Disease: Synthesis, Pharmacology, and Molecular Modeling Studies

Penicillin inhibitors of purple acid phosphatase

Pharmacokinetics of doxorubicinol in dogs

Saponins from Quillaja saponaria Molina: Isolation, Characterization and Ability to Form Immuno Stimulatory Complexes (ISCOMs)

Simultaneous determination of thymine and its sequential catabolites dihydrothymine and β-ureidoisobutyrate in human plasma and urine using liquid chromatography-tandem mass spectrometry with pharmacokinetic application

Simultaneous liquid chromatographic determination of doxorubicin and its major metabolite doxorubicinol in parrot plasma.

Small Peptides Do Not Inhibit Human Non-Pancreatic Secretory Phospholipase-A2 (Type IIA)

Suramin: clinical uses and structure-activity relationships.

Synthesis and evaluation of novel purple acid phosphatase inhibitors

Synthesis and kinetic testing of new inhibitors for a metallo-β-lactamase from Klebsiella pneumonia and Pseudomonas aeruginosa.

Synthesis and kinetic testing of tetrahydropyrimidine-2-thione and pyrrole derivatives as inhibitors of the metallo-β-lactamase from Klebsiella pneumonia and Pseudomonas aeruginosa

Synthesis and polymerization studies of organic-soluble eumelanins.

Synthesis of Nickel-Chelating Fluorinated Lipids for Protein Monolayer Crystallizations

Synthesis of a series of carbon-14 labeled tetrahydropyrido[4,3-d]pyrimidin-4(3H)-ones

Synthesis of cationic derivatives of Quil A and the preparation of cationic immune-stimulating complexes (ISCOMs).

Synthesis, modelling and kinetic assays of potent inhibitors of purple acid phosphatase

The applications of binuclear metallohydrolases in medicine: recent advances in the design and development of novel drug leads for purple acid phosphatases, metallo-β-lactamases and arginases.

The development and application of a novel safety-catch linker for BOC-based assembly of libraries of cyclic peptides.

The identification of new metallo-β-lactamase inhibitor leads from fragment-based screening.

The role of Zn-OR and Zn-OH nucleophiles and the influence of para-substituents in the reactions of binuclear phosphatase mimetics

Toxicokinetics of the active doxorubicin metabolite, doxorubicinol, in sulphur-crested cockatoos (Cacatua galerita)

‘Click’ assembly of glycoclusters and discovery of a trehalose analogue that retards Aβ40 aggregation and inhibits Aβ40-induced neurotoxicity