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List of works by Jennette A Sakoff

(Z)-2-(3,4-Dichlorophenyl)-3-(1H-Pyrrol-2-yl)Acrylonitrile Exhibits Selective Antitumor Activity in Breast Cancer Cell Lines via the Aryl Hydrocarbon Receptor Pathway.

scientific article published on 21 December 2017

A facile hybrid 'flow and batch' access to substituted 3,4-dihydro-2H-benzo[b][1,4]oxazinones

scientific article

A simple HPLC method for plasma level monitoring of mitotane and its two main metabolites in adrenocortical cancer patients

scientific article published on 13 June 2011

Alterations in uterine calcium ions during induction of the decidual cell reaction in pseudopregnant mice.

scientific article published in May 1994

Amino Alcohol Acrylonitriles as Activators of the Aryl Hydrocarbon Receptor Pathway: An Unexpected MTT Phenotypic Screening Outcome

scientific article published on 28 February 2020

Anhydride modified cantharidin analogues: synthesis, inhibition of protein phosphatases 1 and 2A and anticancer activity.

scientific article published on August 2000

Anticancer activity and protein phosphatase 1 and 2A inhibition of a new generation of cantharidin analogues

scientific article

Association of thymidylate synthase enhancer region polymorphisms with thymidylate synthase activity in vivo

scientific article published on 08 June 2010

Building a better dynasore: the dyngo compounds potently inhibit dynamin and endocytosis

scientific article published on 9 October 2013

Cantharidin analogues: synthesis and evaluation of growth inhibition in a panel of selected tumour cell lines

scientific article published on February 2003

Combining the platinum(ii) drug candidate kiteplatin with 1,10-phenanthroline analogues

scientific article published in December 2017

Cytotoxic 2-phenyacrylnitriles, the importance of the cyanide moiety and discovery of potent broad spectrum cytotoxic agents

scientific article

Cytotoxic compounds from Laurencia pacifica

scientific article published on 20 September 2014

Cytotoxicity of a Series of Norcantharidin-Inspired Tetrahydroepoxyisoindole Carboxamides.

scientific article published on 06 December 2016

Dichlorophenylacrylonitriles as AhR Ligands That Display Selective Breast Cancer Cytotoxicity in vitro

scientific article published on 02 July 2018

Focused library development of 2-phenylacrylamides as broad spectrum cytotoxic agents

scientific article

Heterocyclic substituted cantharidin and norcantharidin analogues—synthesis, protein phosphatase (1 and 2A) inhibition, and anti-cancer activity

scientific article published on 02 April 2007

In vitro antibacterial and anticancer properties of Helicteres hirsuta Lour. leaf and stem extracts and their fractions

scientific article published on 12 September 2018

In vitro anticancer properties of selected Eucalyptus species.

scientific article

Inhibition of dynamin by dynole 34-2 induces cell death following cytokinesis failure in cancer cells

scientific article published on 12 July 2011

Inhibition of dynamin mediated endocytosis by the dynoles--synthesis and functional activity of a family of indoles

scientific article

Investigating the cytotoxicity of platinum(II) complexes incorporating bidentate pyridyl-1,2,3-triazole "click" ligands

scientific article published on 15 June 2016

Modified norcantharidins; synthesis, protein phosphatases 1 and 2A inhibition, and anticancer activity

scientific article published on April 2004

Multifaceted Studies of the DNA Interactions and In Vitro Cytotoxicity of Anticancer Polyaromatic Platinum(II) Complexes.

scientific article published on 24 May 2016

Norcantharidin analogues with nematocidal activity in Haemonchus contortus

scientific article published on 13 April 2011

Norcantharidin analogues: synthesis, anticancer activity and protein phosphatase 1 and 2A inhibition

scientific article

Norcantharimide analogues possessing terminal phosphate esters and their anti-cancer activity

scientific article

Norcantharimides, synthesis and anticancer activity: Synthesis of new norcantharidin analogues and their anticancer evaluation

scientific article published on 20 June 2007

Physicochemical Properties, Antioxidant and Anti-proliferative Capacities of Dried Leaf and Its Extract from Xao tam phan (Paramignya trimera).

scientific article published on 25 January 2017

Physicochemical Properties, Antioxidant and Cytotoxic Activities of Crude Extracts and Fractions from Phyllanthus amarus

scientific article published on 18 June 2017

Physicochemical, Antioxidant, and Cytotoxic Properties of Xao Tam Phan (Paramignya trimera) Root Extract and Its Fractions

scientific article published on 28 December 2016

Phytochemical, antioxidant, anti-proliferative and antimicrobial properties of Catharanthus roseus root extract, saponin-enriched and aqueous fractions

scientific article published on 03 April 2019

Protein phosphatase inhibition: structure based design. Towards new therapeutic agents

scientific article published on January 2004

Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain.

scientific article

Pyrimidyn compounds: dual-action small molecule pyrimidine-based dynamin inhibitors.

scientific article

Quantification of hTERT splice variants in melanoma by SYBR green real-time polymerase chain reaction indicates a negative regulatory role for the beta deletion variant.

scientific article published on October 2008

Quinolone-1-(2H)-ones as hedgehog signalling pathway inhibitors

scientific article published on 7 June 2016

Role of the clathrin terminal domain in regulating coated pit dynamics revealed by small molecule inhibition

scientific article

Serine-threonine protein phosphatase inhibitors: development of potential therapeutic strategies

scientific article

Serine/threonine protein phosphatase inhibition enhances the effect of thymidylate synthase inhibition

scientific article published on 25 November 2003

Simple liquid chromatographic method for the determination of uracil and dihydrouracil plasma levels: a potential pretreatment predictor of 5-fluorouracil toxicity.

scientific article

Small molecule inhibitors of serine/threonine protein phosphatases.

scientific article

Small-Molecule Inhibitors of the NusB-NusE Protein-Protein Interaction with Antibiotic Activity

scientific article published on 25 July 2017

Steroids from an Australian sponge Psammoclema sp.

scientific article published in January 2009

Synthesis and Analysis of the Structure, Diffusion and Cytotoxicity of Heterocyclic Platinum(IV) Complexes

scientific article published on 6 October 2015

Synthesis and Cytotoxicity of Octahydroepoxyisoindole-7-carboxylic Acids and Norcantharidin-Amide Hybrids as Norcantharidin Analogues

scientific article published on 14 May 2019

Synthesis and anticancer activity of a series of norcantharidin analogues

scientific article

Synthesis and anticancer activity of focused compound libraries from the natural product lead, oroidin

scientific article

Synthesis and biological activity of Delta-5,6-norcantharimides: importance of the 5,6-bridge

scientific article

Synthesis and biological evaluation of norcantharidin analogues: Towards PP1 selectivity

scientific article published on 24 August 2007

Synthesis and evaluation of novel ellipticines as potential anti-cancer agents

scientific article published on February 2013

Synthesis, characterisation and influence of lipophilicity on cellular accumulation and cytotoxicity of unconventional platinum(iv) prodrugs as potent anticancer agents

scientific article published on 01 November 2019

Synthesis, characterisation and potent cytotoxicity of unconventional platinum(iv) complexes with modified lipophilicity

scientific article published on 01 November 2019

Telomere length in haemopoietic stem cells can be determined from that of mononuclear blood cells or whole blood

scientific article published on October 2002

Telomere length predicts neutrophil recovery in the absence of G-CSF after autologous peripheral blood stem cell transplantation

scientific article published on 01 September 2004

The Role of Calcium in the Artificially Induced Decidual Cell Reaction in Pseudopregnant Mice

scientific article published on 01 April 1996

The aryl hydrocarbon receptor (AhR) as a breast cancer drug target

scientific article published on 12 November 2019

The dynamin inhibitors MiTMAB and OcTMAB induce cytokinesis failure and inhibit cell proliferation in human cancer cells

scientific article published on 22 June 2010

The first two cantharidin analogues displaying PP1 selectivity

scientific article published in February 2002

The synthesis and biological activity of novel anthracenone-pyranones and anthracenone-furans

scientific article published on 22 April 2015

Uterine lipid alterations during early pseudopregnancy and following the artificial induction of decidualization by Concanavalin A in QS mice

scientific article published on 01 May 1996

Uterine receptivity to the artificial deciduogenic agent, concanavalin A, in pseudopregnant QS mice.

scientific article

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