List of works - Marcella Bassetto

A new antiviral scaffold for human norovirus identified with computer-aided approaches on the viral polymerase

scientific article published on 05 December 2019

A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer

scientific article published on 03 July 2019

Antivirals in medical biodefense

scientific article published on 19 February 2020

Computational Studies towards the Identification of Novel Rhodopsin-Binding Compounds as Chemical Chaperones for Misfolded Opsins

scientific article published on 23 October 2020

Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus

scientific article

Computer-aided identification, synthesis and evaluation of substituted thienopyrimidines as novel inhibitors of HCV replication

scientific article

Concise synthesis and biological evaluation of 2-Aroyl-5-amino benzo[b]thiophene derivatives as a novel class of potent antimitotic agents

scientific article

Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer

scientific article published on 22 April 2016

Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents

scientific article

Design, synthesis and evaluation against Chikungunya virus of novel small-molecule antiviral agents

scientific article published on 6 January 2018

In silico identification, design and synthesis of novel piperazine-based antiviral agents targeting the hepatitis C virus helicase

scientific article published on 23 October 2016

In silico structure-based design and synthesis of novel anti-RSV compounds

scientific article published on 8 August 2015

Novel Nucleoside Analogues as Effective Antiviral Agents for Zika Virus Infections

scientific article published on 20 October 2020

Novel symmetrical phenylenediamines as potential anti-hepatitis C virus agents.

scientific article published on 4 November 2016

Polyfluorinated groups in medicinal chemistry.

scientific article published on January 2015

Potent, long-acting cyclopentane-1,3-Dione thromboxane (A2)-receptor antagonists

scientific article published on 24 July 2014

Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety

scientific article published on 2 June 2016

Rational design and synthesis of novel phenylsulfonyl-benzamides as anti-prostate cancer agents.

scientific article published on 26 May 2017

Rational design of highly potent broad-spectrum enterovirus inhibitors targeting the nonstructural protein 2C

scientific article published on 06 November 2020

Rational modifications on a benzylidene-acrylohydrazide antiviral scaffold, synthesis and evaluation of bioactivity against Chikungunya virus

scientific article published on 23 February 2018

Shape-based virtual screening, synthesis and evaluation of novel pyrrolone derivatives as antiviral agents against HCV.

scientific article

Synthesis and biological evaluation of 2-(alkoxycarbonyl)-3-anilinobenzo[b]thiophenes and thieno[2,3-b]pyridines as new potent anticancer agents

scientific article published on 18 March 2013

Synthesis and biological evaluation of 2-substituted-4-(3',4',5'-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents

scientific article published on 12 October 2012

List of works by Marcella Bassetto

A new antiviral scaffold for human norovirus identified with computer-aided approaches on the viral polymerase

A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer

Antivirals in medical biodefense

Computational Studies towards the Identification of Novel Rhodopsin-Binding Compounds as Chemical Chaperones for Misfolded Opsins

Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus

Computer-aided identification, synthesis and evaluation of substituted thienopyrimidines as novel inhibitors of HCV replication

Concise synthesis and biological evaluation of 2-Aroyl-5-amino benzo[b]thiophene derivatives as a novel class of potent antimitotic agents

Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer

Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents

Design, synthesis and evaluation against Chikungunya virus of novel small-molecule antiviral agents

In silico identification, design and synthesis of novel piperazine-based antiviral agents targeting the hepatitis C virus helicase

In silico structure-based design and synthesis of novel anti-RSV compounds

Novel Nucleoside Analogues as Effective Antiviral Agents for Zika Virus Infections

Novel symmetrical phenylenediamines as potential anti-hepatitis C virus agents.

Polyfluorinated groups in medicinal chemistry.

Potent, long-acting cyclopentane-1,3-Dione thromboxane (A2)-receptor antagonists

Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety

Rational design and synthesis of novel phenylsulfonyl-benzamides as anti-prostate cancer agents.

Rational design of highly potent broad-spectrum enterovirus inhibitors targeting the nonstructural protein 2C

Rational modifications on a benzylidene-acrylohydrazide antiviral scaffold, synthesis and evaluation of bioactivity against Chikungunya virus

Shape-based virtual screening, synthesis and evaluation of novel pyrrolone derivatives as antiviral agents against HCV.

Synthesis and biological evaluation of 2-(alkoxycarbonyl)-3-anilinobenzo[b]thiophenes and thieno[2,3-b]pyridines as new potent anticancer agents

Synthesis and biological evaluation of 2-substituted-4-(3',4',5'-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents