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List of works by Robert L Summers

1H-NMR metabolite profiles of different strains of Plasmodium falciparum

scientific article

A series of structurally simple chloroquine chemosensitizing dibemethin derivatives that inhibit chloroquine transport by PfCRT.

scientific article published on 22 February 2011

Chlorpheniramine Analogues Reverse Chloroquine Resistance in Plasmodium falciparum by Inhibiting PfCRT.

scientific article

Diverse mutational pathways converge on saturable chloroquine transport via the malaria parasite's chloroquine resistance transporter

scientific article

Functional characteristics of the malaria parasite's "chloroquine resistance transporter": implications for chemotherapy

scientific article published on July 2010

Inferring a complete genotype-phenotype map from a small number of measured phenotypes

scientific article published on 29 September 2020

Know your enemy: understanding the role of PfCRT in drug resistance could lead to new antimalarial tactics

scientific article published on June 2012

Mimicking the intramolecular hydrogen bond: synthesis, biological evaluation, and molecular modeling of benzoxazines and quinazolines as potential antimalarial agents.

scientific article

Multiple drugs compete for transport via the Plasmodium falciparum chloroquine resistance transporter at distinct but interdependent sites

scientific article (publication date: 26 December 2014)

Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: further structure-activity relationships, in vivo studies, and preliminary toxicity profiling

scientific article

Quinine dimers are potent inhibitors of the Plasmodium falciparum chloroquine resistance transporter and are active against quinoline-resistant P. falciparum

scientific article

Quinoline antimalarials containing a dibemethin group are active against chloroquinone-resistant Plasmodium falciparum and inhibit chloroquine transport via the P. falciparum chloroquine-resistance transporter (PfCRT).

scientific article

Verapamil-Sensitive Transport of Quinacrine and Methylene Blue via the Plasmodium falciparum Chloroquine Resistance Transporter Reduces the Parasite's Susceptibility to these Tricyclic Drugs

scientific article published on 26 October 2015