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List of works by Serge Mignani

4,10-Dihydro-4-oxo-4H-imidazo[1,2-a]indeno[1,2-e]pyrazin-2-carboxylic acid derivatives: highly potent and selective AMPA receptors antagonists with in vivo activity

scientific article published on 01 May 2000

9-Carboxymethyl-5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazin-4-one-2-carbocylic acid (RPR117824): selective anticonvulsive and neuroprotective AMPA antagonist.

scientific article published in May 2002

A novel class of ethacrynic acid derivatives as promising drug-like potent generation of anticancer agents with established mechanism of action

scientific article published on 11 June 2016

Advances in combination therapies based on nanoparticles for efficacious cancer treatment: an analytical report

scientific article

Anti-Inflammatory Effect of Anti-TNF-α SiRNA Cationic Phosphorus Dendrimer Nanocomplexes Administered Intranasally in a Murine Acute Lung Injury Model

scientific article

Anticancer copper(II) phosphorus dendrimers are potent proapoptotic Bax activators

scientific article

Anticancer siRNA cocktails as a novel tool to treat cancer cells. Part (B). Efficiency of pharmacological action

scientific article published on 18 March 2015

Bioisosteres of 9-carboxymethyl-4-oxo-imidazo[1,2-a]indeno-[1,2-e]pyrazin-2-carboxylic acid derivatives. Progress towards selective, potent in vivo AMPA antagonists with longer durations of action.

scientific article

Can dendrimer based nanoparticles fight neurodegenerative diseases? Current situation versus other established approaches

Carboxylative trimethylenemethane cycloadditions catalyzed by palladium

scientific article published on 01 September 1986

Cationic Phosphorus Dendrimer Enhances Photodynamic Activity of Rose Bengal against Basal Cell Carcinoma Cell Lines

scientific article

Comparative EPR studies of Cu(ii)-conjugated phosphorous-dendrimers in the absence and presence of normal and cancer cells

scholarly article in RSC Advances, vol. 4 no. 69, 2014

Complexing Methylene Blue with Phosphorus Dendrimers to Increase Photodynamic Activity

scientific article published on 23 February 2017

Compound high-quality criteria: a new vision to guide the development of drugs, current situation

scientific article

Cyclotriphosphazene core-based dendrimers for biomedical applications: an update on recent advances

scientific article published on 29 January 2018

Dendrimer space concept for innovative nanomedicine: A futuristic vision for medicinal chemistry

scientific article from 2013

Dendrimer-Enabled Therapeutic Antisense Delivery Systems as Innovation in Medicine

scientific article published on 27 June 2019

Dendrimer-protein interactions versus dendrimer-based nanomedicine

scientific article

Dendrimers in combination with natural products and analogues as anti-cancer agents

scientific article published on 20 November 2017

Doxorubicin-Conjugated PAMAM Dendrimers for pH-Responsive Drug Release and Folic Acid-Targeted Cancer Therapy

Enhanced Delivery of Therapeutic siRNA into Glioblastoma Cells Using Dendrimer-Entrapped Gold Nanoparticles Conjugated with β-Cyclodextrin

scientific article published on 27 February 2018

Expand classical drug administration ways by emerging routes using dendrimer drug delivery systems: A concise overview ⬇️

scientific article published on February 13, 2013

Fluorescent Phosphorus Dendrimer as a Spectral Nanosensor for Macrophage Polarization and Fate Tracking in Spinal Cord Injury

scientific article published on 14 July 2015

Fluorescent Phosphorus Dendrimers: Towards Material and Biological Applications

scientific article published on 01 August 2019

Fourier transform infrared spectroscopy (FTIR) characterization of the interaction of anti-cancer photosensitizers with dendrimers

scientific article published on 27 October 2015

From PtCl(2)- and acid-catalyzed to uncatalyzed cycloisomerization of 2-propargyl anilines: access to functionalized indoles

scientific article published on 01 January 2007

From metallodrugs to metallodendrimers for nanotherapy in oncology: a concise overview.

scientific article published on January 2012

Hydrogels of Polycationic Acetohydrazone-Modified Phosphorus Dendrimers for Biomedical Applications: Gelation Studies and Nucleic Acid Loading

In vitro PAMAM, phosphorus and viologen-phosphorus dendrimers prevent rotenone-induced cell damage

scientific article published on 7 August 2014

Indeno[1,2-b]pyrazin-2,3-diones: a new class of antagonists at the glycine site of the NMDA receptor with potent in vivo activity

scientific article published on 01 June 2000

Interactions gold/phosphorus dendrimers. Versatile ways to hybrid organic–metallic macromolecules

scholarly article by Jean Pierre Majoral et al published March 2018 in Coordination Chemistry Reviews

Interference of cationic polymeric nanoparticles with clinical chemistry tests--clinical relevance.

scientific article published in August 2014

Investigations on dendrimer space reveal solid and liquid tumor growth-inhibition by original phosphorus-based dendrimers and the corresponding monomers and dendrons with ethacrynic acid motifs

scientific article published on March 2015

Mechanism of cationic phosphorus dendrimer toxicity against murine neural cell lines

scientific article published on 30 July 2013

Metal-based phosphorus dendrimers as novel nanotherapeutic strategies to tackle cancers: A concise overview

scientific article published on 07 August 2019

Multivalent Copper(II)-Conjugated Phosphorus Dendrimers with Noteworthy In Vitro and In Vivo Antitumor Activities: A Concise Overview

scientific article published on 25 November 2020

Neuroprotective effects of RPR 104632, a novel antagonist at the glycine site of the NMDA receptor, in vitro.

scientific article published on April 1996

Neutral high-generation phosphorus dendrimers inhibit macrophage-mediated inflammatory response in vitro and in vivo.

scientific article published on 28 August 2017

New Ways to Treat Tuberculosis Using Dendrimers as Nanocarriers

Original Multivalent Gold(III) and Dual Gold(III)-Copper(II) Conjugated Phosphorus Dendrimers as Potent Antitumoral and Antimicrobial Agents

scientific article published on 29 September 2017

Original multivalent copper(II)-conjugated phosphorus dendrimers and corresponding mononuclear copper(II) complexes with antitumoral activities

scientific article published on 7 March 2013

Phosphorus dendrimers and photodynamic therapy. Spectroscopic studies on two dendrimer-photosensitizer complexes: Cationic phosphorus dendrimer with rose bengal and anionic phosphorus dendrimer with methylene blue

scientific article published on 24 June 2015

Phosphorus-containing nanoparticles: biomedical patents review

scientific article

Potent anticancer efficacy of first-in-class Cu(II) and Au(III) metaled phosphorus dendrons with distinct cell death pathways

scientific article published on 06 March 2020

Promising low-toxicity of viologen-phosphorus dendrimers against embryonic mouse hippocampal cells.

scientific article published on 30 September 2013

Rearrangement of Homoallylic Alcohols Induced by DAST

scientific article published on 01 May 2006

Revisiting Cationic Phosphorus Dendrimers as a Nonviral Vector for Optimized Gene Delivery Towards Cancer Therapy Applications

scientific article published on 29 April 2020

Riluzole series. Synthesis and in vivo "antiglutamate" activity of 6-substituted-2-benzothiazolamines and 3-substituted-2-imino-benzothiazolines

scientific article published on 01 July 1999

Spiro-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one derivatives are mixed AMPA and NMDA glycine-site antagonists active in vivo

scientific article published on 01 October 1999

Stable functionalized PEGylated quantum dots micelles with a controlled stoichiometry

scientific article published on 22 November 2010

Symmetrical and unsymmetrical incorporation of active biological monomers on the surface of phosphorus dendrimers

Synthesis and potent anticonvulsant activities of 4-oxo-imidazo[1,2-a]inden.

scientific article published in December 2000

Synthesis and structure-activity relationships of 4,10-dihydro-4-oxo-4H-imidazo[1,2-a]indeno[1,2-e]pyrazine derivatives: highly potent and selective AMPA receptor antagonists with in vivo activity.

scientific article published on February 2004

Synthesis of Onion-Peel Nanodendritic Structures with Sequential Functional Phosphorus Diversity

scientific article published on 05 March 2015

Synthesis of dissymmetric phosphorus dendrimers using an unusual protecting group

Thiazoyl phosphines. Design, reactivity, and complexation

scientific article published on 26 May 2016

Total Synthesis of Herbimycin A

scientific article published on 01 January 2007

Why and how have drug discovery strategies in pharma changed? What are the new mindsets?

scientific article published on 13 September 2015

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