List of works - Frederik Diness

Azotides as Modular Peptide-Based Ligands for Asymmetric Lewis Acid Catalysis

scientific article published on 13 May 2019

Biophysical characterization of the proton-coupled oligopeptide transporter YjdL.

scientific article published on 23 August 2012

C-Terminal lactamization of peptides

scientific article published on 24 December 2020

C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles.

scientific article published on 29 February 2016

Catalyst-Free N-Arylation Using Unactivated Fluorobenzenes

scientific article published on 02 July 2012

Click-Chemistry-Mediated Synthesis of Selective Melanocortin Receptor 4 Agonists.

scientific article

Comparative studies of adhesion peptides based on l- or d-amino acids.

scientific article published in September 2016

Comparative α-helicity of cyclic pentapeptides in water

scientific article

Computational Evolution of Threonine-Rich β-Hairpin Peptides Mimicking Specificity and Affinity of Antibodies

scientific article published on 28 January 2019

Constraining cyclic peptides to mimic protein structure motifs.

scientific article

Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12

scientific article published on 23 February 2020

Diversity-Oriented Syntheses by Combining CuAAC and Stereoselective INCIC Reactions with Peptides

scientific article

Mechanism and Scope of Base-Controlled Catalyst-Free N-Arylation of Amines with Unactivated Fluorobenzenes

scientific article

Metabolically stable cellular adhesion to inert surfaces.

scientific article published on 16 September 2011

Metallo-Organozymes with Specific Proteolytic Activity

scientific article published on 30 October 2018

Probing the aglycon binding site of a beta-glucosidase: a collection of C-1-modified 2,5-dideoxy-2,5-imino-D-mannitol derivatives and their structure-activity relationships as competitive inhibitors.

scientific article

Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity.

scientific article published on January 2010

Rational Tuning of Fluorobenzene Probes for Cysteine-Selective Protein Modification

scientific article published on 14 April 2018

Sequential direct SNAr reactions of pentafluorobenzenes with azole or indole derivatives

scientific article published on 28 May 2014

Solid-phase synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines by stereoselective intramolecular N-carbamyliminium Pictet-Spengler reactions

scientific article published on 01 October 2006

Sustainable Flow Synthesis of Encoded Beads for Combinatorial Chemistry and Chemical Biology

scientific article published on 18 July 2018

Synthesis and stability of strongly acidic benzamide derivatives

scientific article published on 27 February 2018

Synthesis of the Thiazole–Thiazoline Fragment of Largazole Analogues

scientific article published on 08 November 2011

The Pictet-Spengler reaction in solid-phase combinatorial chemistry.

scientific article

Total Synthesis, Structure, and Oral Absorption of a Thiazole Cyclic Peptide, Sanguinamide A

scientific article published on 06 November 2012

Twists or turns: stabilising alpha vs. beta turns in tetrapeptides

scientific article published on 03 October 2019

X-ray diffraction data as a source of the vibrational free-energy contribution in polymorphic systems

scientific article published on 08 May 2019

List of works by Frederik Diness

Azotides as Modular Peptide-Based Ligands for Asymmetric Lewis Acid Catalysis

Biophysical characterization of the proton-coupled oligopeptide transporter YjdL.

C-Terminal lactamization of peptides

C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles.

Catalyst-Free N-Arylation Using Unactivated Fluorobenzenes

Click-Chemistry-Mediated Synthesis of Selective Melanocortin Receptor 4 Agonists.

Comparative studies of adhesion peptides based on l- or d-amino acids.

Comparative α-helicity of cyclic pentapeptides in water

Computational Evolution of Threonine-Rich β-Hairpin Peptides Mimicking Specificity and Affinity of Antibodies

Constraining cyclic peptides to mimic protein structure motifs.

Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12

Diversity-Oriented Syntheses by Combining CuAAC and Stereoselective INCIC Reactions with Peptides

Mechanism and Scope of Base-Controlled Catalyst-Free N-Arylation of Amines with Unactivated Fluorobenzenes

Metabolically stable cellular adhesion to inert surfaces.

Metallo-Organozymes with Specific Proteolytic Activity

Probing the aglycon binding site of a beta-glucosidase: a collection of C-1-modified 2,5-dideoxy-2,5-imino-D-mannitol derivatives and their structure-activity relationships as competitive inhibitors.

Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity.

Rational Tuning of Fluorobenzene Probes for Cysteine-Selective Protein Modification

Sequential direct SNAr reactions of pentafluorobenzenes with azole or indole derivatives

Solid-phase synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines by stereoselective intramolecular N-carbamyliminium Pictet-Spengler reactions

Sustainable Flow Synthesis of Encoded Beads for Combinatorial Chemistry and Chemical Biology

Synthesis and stability of strongly acidic benzamide derivatives

Synthesis of the Thiazole–Thiazoline Fragment of Largazole Analogues

The Pictet-Spengler reaction in solid-phase combinatorial chemistry.

Total Synthesis, Structure, and Oral Absorption of a Thiazole Cyclic Peptide, Sanguinamide A

Twists or turns: stabilising alpha vs. beta turns in tetrapeptides

X-ray diffraction data as a source of the vibrational free-energy contribution in polymorphic systems