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List of works by Werner Sieghart

6,3'-Dinitroflavone is a low efficacy modulator of GABA(A) receptors.

scientific article

8-Substituted Triazolobenzodiazepines: <i>In Vitro</i> and <i>In Vivo</i> Pharmacology in Relation to Structural Docking at the α1 Subunit-Containing GABA<sub>A</sub> Receptor

scientific article published on 20 April 2021

A novel positive allosteric modulator of the GABA(A) receptor: the action of (+)-ROD188

scientific article

A novel serine kinase with specificity for beta3-subunits is tightly associated with GABA(A) receptors

scientific article published on 01 July 1999

A novel site on gamma 3 subunits important for assembly of GABA(A) receptors

scientific article (publication date: 23 August 2002)

A polymorphism (5-HTTLPR) in the serotonin transporter promoter gene is associated with DSM-IV depression subtypes in seasonal affective disorder.

scientific article published in November 2003

A propofol binding site on mammalian GABAA receptors identified by photolabeling

scientific article

A rapid and simple method for efficient coating of microtiter plates using low amounts of antigen in the presence of detergent

scientific article published on 01 December 1986

AMPA and kainate receptors mediate mutually exclusive effects on GABA(A) receptor expression in cultured mouse cerebellar granule neurones

scientific article

Abolition of zolpidem sensitivity in mice with a point mutation in the GABAA receptor gamma2 subunit.

scientific article

Additional support for linkage of schizophrenia and bipolar disorder to chromosome 3q29

scientific article published on 06 March 2007

Affinity of various ligands for benzodiazepine receptors in rat cerebellum and hippocampus.

scientific article published in December 1984

Allosteric modulation of GABAA receptors via multiple drug-binding sites.

scientific article

Alterations in GABAA Receptor Subunit Expression in the Amygdala and Entorhinal Cortex in Human Temporal Lobe Epilepsy

scientific article published on 01 November 2019

Alterations in the expression of GABAA receptor subunits in cerebellar granule cells after the disruption of the alpha6 subunit gene.

scientific article published in May 1999

Altered receptor subtypes in the forebrain of GABA(A) receptor delta subunit-deficient mice: recruitment of gamma 2 subunits.

scientific article

Alternate use of distinct intersubunit contacts controls GABAA receptor assembly and stoichiometry.

scientific article

An updated unified pharmacophore model of the benzodiazepine binding site on gamma-aminobutyric acid(a) receptors: correlation with comparative models

scientific article

Antiallergic drug cromolyn may inhibit histamine secretion by regulating phosphorylation of a mast cell protein

scientific article published on 01 January 1980

Antibodies specific for GABAA receptor alpha subunits reveal that chronic alcohol treatment down-regulates alpha-subunit expression in rat brain regions

scientific article published on 01 November 1993

Antiseizure activity of novel gamma-aminobutyric acid (A) receptor subtype-selective benzodiazepine analogues in mice and rat models

scientific article published on April 2009

Anxiolytic-like effects of 8-acetylene imidazobenzodiazepines in a rhesus monkey conflict procedure

scientific article published on August 18, 2010

Anxioselective anxiolytics: additional perspective.

scientific article published on 5 February 2013

Apparent identity of alpha-subunit of pyruvate dehydrogenase and the protein phosphorylated in the presence of glutamate in P2-fractions of rat cerebral cortex

scientific article published on 01 January 1984

Are GABAA receptors containing alpha5 subunits contributing to the sedative properties of benzodiazepine site agonists?

scientific article

Assembly of GABA(A) receptors (Review).

scientific article published on May 2008

Association Studies of Candidate Genes in Bipolar Disorders

article

Association of proteins irreversibly labeled by 3H-flunitrazepam with different benzodiazepine

scientific article published on January 1, 1983

Association study of schizophrenia spectrum disorders and dopamine D3 receptor gene: is schizoaffective disorder special?

article

Attenuated sensitivity to neuroactive steroids in gamma-aminobutyrate type A receptor delta subunit knockout mice.

scientific article published on October 1999

Azemiopsin from Azemiops feae viper venom, a novel polypeptide ligand of nicotinic acetylcholine receptor.

scientific article

Behavioural correlates of an altered balance between synaptic and extrasynaptic GABAAergic inhibition in a mouse model.

scientific article published in October 2004

Benzodiazepine receptors: multiple receptors or multiple conformations?

scientific article published on 01 January 1985

Benzodiazepine-induced spatial learning deficits in rats are regulated by the degree of modulation of α1 GABA(A) receptors

scientific article

Benzodiazepine-mediated regulation of alpha1, alpha2, beta1-3 and gamma2 GABA(A) receptor subunit proteins in the rat brain hippocampus and cortex.

scientific article

Benzodiazepines modulate GABAreceptors by reducing a gamma-subunit-mediated inhibition of GABA sensitivity

scientific article published on 12 November 2009

Bidirectional alterations of GABA(A) receptor subunit peptide levels in rat cortex during chronic ethanol consumption and withdrawal.

scientific article published in July 1997

Binding of gamma-aminobutyric acidA receptors to tubulin

scientific article published on 01 September 1994

Binge alcohol drinking is associated with GABAAα2-regulated Toll-like receptor 4 (TLR4) expression in the central amygdala

scientific article published on February 28, 2011

Biochemical, immunological, and pharmacological characterization of GABAA-benzodiazepine receptor subtypes

scientific article published on January 1, 1992

Biological evaluation of 2'-[18F]fluoroflumazenil ([18F]FFMZ), a potential GABA receptor ligand for PET.

scientific article published in February 2004

Biperiden and Haloperidol Plasma Levels and Extrapyramidal Side Effects in Schizophrenic Patients

scientific article published on 01 January 1997

CYP2D6 genotype and phenotyping by determination of dextromethorphan and metabolites in serum of healthy controls and of patients under psychotropic medication.

scientific article published on December 1997

Ca2+ and cyclic AMP regulate phosphorylation of same two membrane-associated proteins specific to nerve tissue

scientific article published on May 1, 1979

Calcium-dependent protein phosphorylation during secretion by exocytosis in the mast cell

scientific article published on September 28, 1978

Cellular localization and differential distribution of GABAA receptor subunit proteins and messenger RNAs within hypothalamic magnocellular neurons

scientific article published on 01 February 1995

Cerebellar α6 subunit-containing GABAA receptors: A novel therapeutic target for disrupted prepulse inhibition in neuropsychiatric disorders.

scientific article published on 8 March 2018

Clinical-pharmacological study with the two isomers (d-, l-) of fenfluramine and its comparison with chlorpromazine and d-amphetamine: blood levels, EEG mapping and safety evaluation.

scientific article published in June 1993

Clusters of GABAA receptors on cultured hippocampal cells correlate only partially with functional synapses.

scientific article published in April 1999

Colocalization of GABA, glycine, and their receptors at synapses in the rat spinal cord

scientific article published on 01 February 1996

Comparative bioavailability studies with a new mixed-micelles solution of diazepam utilizing radioreceptor assay, psychometry and EEG brain mapping.

scientific article published in October 1988

Comparative modeling of GABA(A) receptors: limits, insights, future developments.

scientific article

Comparative models of GABAA receptor extracellular and transmembrane domains: important insights in pharmacology and function.

scientific article

Comparison of benzodiazepine receptor binding in membranes from human or rat brain.

scientific article published in August 1985

Comparison of benzodiazepine receptors in cerebellum and inferior colliculus.

scientific article

Comparison of tryptic peptides of benzodiazepine binding proteins photolabeled with [3H]flunitrazepam or [3H]Ro 15-4513

scientific article published on 01 April 1987

Comparison of two different benzodiazepine binding proteins by peptide mapping after limited proteolysis

scientific article published on 01 May 1988

Composition of the GABA(A) receptors of retinal dopaminergic neurons

scientific article published on 01 September 1999

Cultured Hippocampal Pyramidal Neurons Express Two Kinds of GABAA Receptors

scientific article

Deep amino acid sequencing of native brain GABAA receptors using high-resolution mass spectrometry

scientific article published on January 2012

Deficits in phosphorylation of GABA(A) receptors by intimately associated protein kinase C activity underlie compromised synaptic inhibition during status epilepticus

scientific article

Deficits in spatial memory correlate with modified {gamma}-aminobutyric acid type A receptor tyrosine phosphorylation in the hippocampus.

scientific article

Design and Synthesis of Novel Deuterated Ligands Functionally Selective for the γ-Aminobutyric Acid Type A Receptor (GABAAR) α6 Subtype with Improved Metabolic Stability and Enhanced Bioavailability.

scientific article published on 26 February 2018

Detection and binding properties of GABA(A) receptor assembly intermediates.

scientific article published on 23 February 2001

Development of gamma-aminobutyric acidergic synapses in cultured hippocampal neurons

scientific article

Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands

scientific article

Differential degradation of different benzodiazepine binding proteins by incubation of membranes from cerebellum or hippocampus with trypsin.

scientific article published in July 1985

Differential localization of GABA(A) receptor subunits in relation to rat striatopallidal and pallidopallidal synapses.

scientific article published on 11 January 2011

Differential regulation of GABA(A) receptor gene expression by ethanol in the rat hippocampus versus cerebral cortex.

scientific article

Differential regulation of synaptic GABAA receptors by cAMP-dependent protein kinase in mouse cerebellar and olfactory bulb neurones.

scientific article published in December 1999

Distribution of GABAA receptor alpha 1 subunit-like immunoreactivity in comparison with that of enkephalin and substance P in the rat forebrain

scientific article published on 01 June 1995

Distribution of alpha1, alpha4, gamma2, and delta subunits of GABAA receptors in hippocampal granule cells

scientific article

Dopamine D3 receptor gene polymorphism and response to clozapine in schizophrenic Pakistani patients

article

Drug interactions with cyclic nucleotide and protein phosphorylation systems

scientific article published on January 1, 1979

Dual mode of stimulation by the beta-carboline ZK 91085 of recombinant GABA(A) receptor currents: molecular determinants affecting its action

scientific article

EDPC: a novel high affinity ligand for the benzodiazepine site on rat GABA(A) receptors.

scientific article

Early postnatal switch in GABAA receptor α-subunits in the reticular thalamic nucleus

scientific article published on 2 December 2015

Engineered Flumazenil Recognition Site Provides Mechanistic Insight Governing Benzodiazepine Modulation in GABA Receptors

scientific article published on 23 July 2018

Establishing a new mouse model for investigating the function of amygdala neurons in anxiety.

scientific article published on 5 November 2008

European multicentre association study of schizophrenia: a study of the DRD2 Ser311Cys and DRD3 Ser9Gly polymorphisms

scientific article published on 01 February 1998

European multicentre evaluation of the analytical performance of the Abbott AxSYM Abused Drugs Assays

scientific article published on 01 February 1997

Evidence That Sedative Effects of Benzodiazepines Involve Unexpected GABAA Receptor Subtypes: Quantitative Observation Studies in Rhesus Monkeys

scientific article published on 02 May 2018

Evidence for association of a high affinity avermectin binding site with the benzodiazepine receptor.

scientific article published in June 1984

Evidence for the existence of differential O-glycosylated alpha 5-subunits of the gamma-aminobutyric acidA receptor in the rat brain.

scientific article published in January 1993

Evidence for the existence of several different alpha- and beta-subunits of the GABA/benzodiazepine receptor complex from rat brain.

scientific article published in February 1989

Extensive heterogeneity of recombinant gamma-aminobutyric acidA receptors expressed in alpha 4 beta 3 gamma 2-transfected human embryonic kidney 293 cells.

scientific article

Fear learning induces structural and functional plasticity at GABAergic synapses in the basolateral amygdala.

scientific article published on 5 September 2011

Fear learning triggers structural changes at GABAergic synapses in the basal amygdala.

scientific article published on 16 November 2010

First In Vivo Testing of Compounds Targeting Group 3 Medulloblastomas Using an Implantable Microdevice as a New Paradigm for Drug Development.

scientific article

Formation of GABAA receptor complexes containing α1 and α5 subunits is paralleling a multiple T-maze learning task in mice

scientific article published on 7 May 2016

From synapse to behavior: rapid modulation of defined neuronal types with engineered GABAA receptors.

scientific article

Functional correlation of GABA(A) receptor alpha subunits expression with the properties of IPSCs in the developing thalamus.

scientific article published in March 2000

GABA A receptors: subtypes provide diversity of function and pharmacology

scientific article

GABA expression dominates neuronal lineage progression in the embryonic rat neocortex and facilitates neurite outgrowth via GABA(A) autoreceptor/Cl- channels.

scientific article

GABA influences the development of the ventromedial nucleus of the hypothalamus.

scientific article published in December 2001

GABA receptor associated drug receptors.

scientific article published on January 1981

GABA(A) Receptors: Post-Synaptic Co-Localization and Cross-Talk with Other Receptors.

scientific article

GABA(A) benzodiazepine receptors and epilepsy

scientific article published on 01 March 1990

GABA(A) receptor assembly. Identification and structure of gamma(2) sequences forming the intersubunit contacts with alpha(1) and beta(3) subunits

scientific article published on 01 March 2000

GABA(A) receptor subtype-selectivity of novel bicuculline derivatives

scientific article published in January 2015

GABA(A) receptor subunits in the rat hippocampus I: immunocytochemical distribution of 13 subunits.

scientific article published in October 1997

GABA(A) receptor subunits in the rat hippocampus II: altered distribution in kainic acid-induced temporal lobe epilepsy.

scientific article published in October 1997

GABA(A) receptor subunits in the rat hippocampus III: altered messenger RNA expression in kainic acid-induced epilepsy.

scientific article published in October 1997

GABA(A) receptors: immunocytochemical distribution of 13 subunits in the adult rat brain.

scientific article

GABAA alpha6-containing receptors are selectively compromised in cerebellar granule cells of the ataxic mouse, stargazer.

scientific article

GABAA receptor phosphorylation and functional modulation in cortical neurons by a protein kinase C-dependent pathway.

scientific article published on December 2000

GABAA receptor subunit composition and functional properties of Cl- channels with differential sensitivity to zolpidem in embryonic rat hippocampal cells.

scientific article

GABAA receptor subunits in the human amygdala and hippocampus: Immunohistochemical distribution of 7 subunits.

scientific article published on 12 October 2017

GABAA, Receptor α1, α4, and β3 Subunit mRNA and Protein Expression in the Frontal Cortex of Human Alcoholics

scientific article published on June 1, 1998

Gel-based mass spectrometric analysis of a strongly hydrophobic GABAA-receptor subunit containing four transmembrane domains

scientific article published on 2 July 2009

Gel-based mass spectrometric analysis of recombinant GABA(A) receptor subunits representing strongly hydrophobic transmembrane proteins

scientific article

Genetic polymorphisms for drug metabolism (CYP2D6) and tardive dyskinesia in schizophrenia

scientific article published on 01 July 1998

Genome scan for susceptibility loci for schizophrenia

scientific article published in January 2000

Genome scan for susceptibility loci for schizophrenia and bipolar disorder

scientific article published on July 2002

Gephyrin, the enigmatic organizer at GABAergic synapses

scientific article published on 15 May 2012

Glutamate-Stimulated Phosphorylation of a Specific Protein in P2Fractions of Rat Cerebral Cortex

scientific article published on November 1, 1981

Heterogeneity of GABAA receptors

scientific article published on January 1, 1992

Heterogeneity of GABAA-benzodiazepine receptors

scientific article published on February 1, 1991

Histaminergic pharmacology of homo-oligomeric β3 γ-aminobutyric acid type A receptors characterized by surface plasmon resonance biosensor technology.

scientific article published on 15 April 2012

Homologous sites of GABA(A) receptor alpha(1), beta(3) and gamma(2) subunits are important for assembly.

scientific article

Identification of amino acid residues important for assembly of GABA receptor alpha1 and gamma2 subunits.

scientific article published on 12 January 2006

Identification of amino acid residues of GABA(A) receptor subunits contributing to the formation and affinity of the tert-butylbicyclophosphorothionate binding site.

scientific article

Identification of an amino acid sequence within GABA(A) receptor beta3 subunits that is important for receptor assembly.

scientific article published on January 2003

Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface

scientific article published on May 2013

Identification of the cyclic AMP-dependent protein kinase responsible for endogenous phosphorylation of substrate proteins in synaptic membrane fraction from rat brain

scientific article published on December 10, 1979

Immunoaffinity purification of gamma-aminobutyric acidA (GABAA) receptors containing gamma 1-subunits. Evidence for the presence of a single type of gamma-subunit in GABAA receptors

scientific article published on 01 October 1994

Immunocytochemical localization of the alpha 1 and beta 2/3 subunits of the GABAA receptor in relation to specific GABAergic synapses in the dentate gyrus

scientific article published on 01 April 1995

Immunohistochemical and neurochemical evidence for GABAA receptor heterogeneity between the hypothalamus and cortex.

scientific article published on October 1994

Improved radioimmunoassay of melatonin in serum

scientific article published on 01 April 1987

In vivo and in vitro evaluation of [18F]FETO with respect to the adrenocortical and GABAergic system in rats.

scientific article published on 3 July 2003

Increased Expression of GABAAReceptor β-Subunits in the Hippocampus of Patients with Temporal Lobe Epilepsy

scientific article (publication date: August 2003)

Initially expressed early rat embryonic GABA(A) receptor Cl- ion channels exhibit heterogeneous channel properties.

scientific article

Insights into functional pharmacology of α₁ GABA(A) receptors: how much does partial activation at the benzodiazepine site matter?

scientific article published on 18 May 2013

Interaction between serotonin 5-HT2A receptor gene and dopamine transporter (DAT1) gene polymorphisms influences personality trait of persistence in Austrian Caucasians

scientific article published in March 2010

Interaction of allosteric ligands with GABAA receptors containing one, two, or three different subunits

scientific article

Interaction of benzodiazepine agonists and antagonists with different benzodiazepine receptors

scientific article published on January 1, 1983

International Union of Pharmacology. XV. Subtypes of gamma-aminobutyric acidA receptors: classification on the basis of subunit structure and receptor function

scientific article published on June 1, 1998

Investigation of the abundance and subunit composition of GABAA receptor subtypes in the cerebellum of alpha1-subunit-deficient mice.

scientific article published on 8 November 2005

Irreversible Binding of [3H]Flunitrazepam to Different Proteins in Various Brain Regions

scientific article published on July 1, 1983

Ligand-gated ion channel subunit partnerships: GABAA receptor alpha6 subunit gene inactivation inhibits delta subunit expression.

scientific article published in February 1997

Localization of GABA‐A receptor alpha subunits on neurochemically distinct cell types in the rat locus coeruleus

scientific article published on June 21, 2011

Long-range interactions in neuronal gene expression: evidence from gene targeting in the GABA(A) receptor beta2-alpha6-alpha1-gamma2 subunit gene cluster

scientific article published on 01 July 2000

Molecular basis of pharmacological heterogeneity of GABAA receptors

scientific article published on May 1, 1992

Molecular basis of the γ-aminobutyric acid A receptor α3 subunit interaction with the clustering protein gephyrin

scientific journal article

Molecular heterogeneity of benzodiazepine receptors

scientific article published on 01 July 1980

Multiplicity of GABAA--benzodiazepine receptors.

scientific article

Mutagenesis and computational docking studies support the existence of a histamine binding site at the extracellular β3+β3- interface of homooligomeric β3 GABAA receptors

scientific article published on 29 April 2016

N-Deglycosylation and immunological identification indicates the existence of β-subunit isoforms of the rat GABAAreceptor

scientific article published on August 5, 1991

Neuronal localization of Ca2+-dependent protein phosphorylation in brain

scientific article published on 01 March 1980

Neuronal localization of specific brain phosphoproteins

scientific article published on November 10, 1978

Neurosteroid Analog Photolabeling of a Site in the Third Transmembrane Domain of the β3 Subunit of the GABAA Receptor

scientific article published on May 30, 2012

Neurotoxins from snake venoms and α-conotoxin ImI inhibit functionally active ionotropic γ-aminobutyric acid (GABA) receptors

scientific article published on 28 July 2015

No association of clock gene T3111C polymorphism and affective disorders

article

No association of the neuropeptide Y (Leu7Pro) and ghrelin gene (Arg51Gln, Leu72Met, Gln90Leu) single nucleotide polymorphisms with eating disorders

article

Non-association of dopamine D4 and D2 receptor genes with personality in healthy individuals

scientific article published in September 2000

Patterns of mRNA and protein expression for 12 GABAA receptor subunits in the mouse brain.

scientific article published on 18 January 2013

Pentameric ligand-gated ion channel ELIC is activated by GABA and modulated by benzodiazepines

scientific article

Pharmacological properties of GABAA receptors containing gamma1 subunits.

scientific article

Phosphorylation of a single mast cell protein in response to drugs that inhibit secretion

scientific article published on 01 October 1981

Photoaffinity labeling of benzodiazepine receptors with a partial inverse agonist

scientific article published on June 15, 1984

Photoaffinity labeling of different benzodiazepine receptors at physiological temperature.

scientific article published on December 1984

Plasticity of GABAA receptors after ethanol pre-exposure in cultured hippocampal neurons.

scientific article

Possible association between childhood absence epilepsy and the gene encoding GABRB3

article

Possible linkage of schizophrenia and bipolar affective disorder to chromosome 3q29

scientific article published on 01 May 2004

Postnatal development of proteins associated with different benzodiazepine receptors.

scientific article published on January 1986

Postnatal development of proteins irreversibly labeled by [3H]flunitrazepam.

scientific article published in July 1982

Potassium-evoked release of taurine from synaptosomal fractions of rat cerebral cortex.

scientific article published in November 1976

Potency of several type I-benzodiazepine receptor ligands for inhibition of [3H]flunitrazepam binding in different rat brain tissues

scientific article published on May 2, 1991

Properties of [3H]flunitrazepam binding to different benzodiazepine binding proteins

scientific article published on 01 April 1983

Properties of [3H]taurine release from crude synaptosomal fractions of rat cerebral cortex

scientific article published on December 1, 1979

Properties of a high affinity binding site for [3H]avermectin B1a.

scientific article published in April 1984

Protein kinase C phosphorylation regulates membrane insertion of GABAA receptor subtypes that mediate tonic inhibition.

scientific article

Quantitative localisation of synaptic and extrasynaptic GABAA receptor subunits on hippocampal pyramidal cells by freeze-fracture replica immunolabelling.

scientific article published on 14 November 2010

Rat beta 3 subunits expressed in human embryonic kidney 293 cells form high affinity [35S]t-butylbicyclophosphorothionate binding sites modulated by several allosteric ligands of gamma-aminobutyric acid type A receptors

scientific article published on 01 September 1995

Regulation of GABA(A) receptor dynamics by interaction with purinergic P2X(2) receptors.

scientific article published on 22 February 2011

Removal of GABA(A) receptor γ2 subunits from parvalbumin neurons causes wide-ranging behavioral alterations

scientific article

Response of thyrotropin to thyrotropin-releasing hormone as predictor of treatment outcome. Prediction of recovery and relapse in treatment with antidepressants and neuroleptics

scientific article published on 01 September 1986

Role of the GABAAreceptor γ2 subunit in the development of gonadotropin-releasing hormone neurons in vivo

article

Schizophrenia and the dopamine-beta-hydroxylase gene: results of a linkage and association study

article

Schizophrenia and the dopamine-β-hydroxylase gene

article

Search for α3β₂/₃γ2 subtype selective ligands that are stable on human liver microsomes

scientific article

Sedimentation and release properties of P2 fractions derived from rat cerebral cortex slices incubated with radiolabeled GABA for a short or long time period.

scientific article published in November 1981

Sedimentation and release properties of glial particles present in P2-fractions isolated from rat cerebral cortex

scientific article published on July 6, 1979

Sedimentation characteristics of subcellular vesicles derived from three glial systems

scientific article published on June 1, 1978

Segregation of different GABAA receptors to synaptic and extrasynaptic membranes of cerebellar granule cells

scientific article

Several new benzodiazepines selectively interact with a benzodiazepine receptor subtype

scientific article

Sh-I-048A, an in vitro non-selective super-agonist at the benzodiazepine site of GABAA receptors: the approximated activation of receptor subtypes may explain behavioral effects

scientific article published on 25 January 2014

Somatostatin-induced phosphorylation of mast cell proteins

scientific article published on 01 October 1981

Spatio-temporal expression analysis of the calcium-binding protein calumenin in the rodent brain

scientific article

Spontaneous cross-link of mutated alpha1 subunits during GABA(A) receptor assembly.

scientific article published on 4 December 2006

Stoichiometry and assembly of a recombinant GABAA receptor subtype.

scientific article published on April 1997

Striatal efferents preferentially innervate neurons in the ventral pallidum containing GABAA receptor alpha 1 subunit-like immunoreactivity

scientific article published on 01 June 1996

Structure and pharmacology of gamma-aminobutyric acidA receptor subtypes.

scientific article

Structure and subunit composition of GABA(A) receptors.

scientific article

Structure, pharmacology, and function of GABAA receptor subtypes.

scientific article published on January 2006

Subcellular distribution of dopamine-sensitive adenylate cyclase.

scientific article published in June 1976

Subtype selectivity of α+β- site ligands of GABAA receptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors.

scientific article published on May 2013

Subunit Compensation and Plasticity of Synaptic GABAA Receptors Induced by Ethanol in ?4 Subunit Knockout Mice

scientific article published on September 23, 2011

Subunit composition and pharmacological characterization of gamma-aminobutyric acid type A receptors in frog pituitary melanotrophs

scientific article published on 01 March 2000

Subunit composition and quantitative importance of hetero-oligomeric receptors: GABAA receptors containing alpha6 subunits.

scientific article published in April 1998

Synthesis and GABA(A) receptor activity of 6-oxa-analogs of neurosteroids

scientific article published on 01 June 2000

Synthesis, in vitro affinity, and efficacy of a bis 8-ethynyl-4H-imidazo[1,5a]- [1,4]benzodiazepine analogue, the first bivalent alpha5 subtype selective BzR/GABA(A) antagonist.

scientific article published on December 2003

Targeted disruption of the GABA(A) receptor delta subunit gene leads to an up-regulation of gamma 2 subunit-containing receptors in cerebellar granule cells

scientific journal article

The Cell Adhesion Molecule Neuroplastin-65 Is a Novel Interaction Partner of γ-Aminobutyric Acid Type A Receptors

scientific article published on March 2, 2012

The GABAA receptor alpha+beta- interface: a novel target for subtype selective drugs

scientific article

The alpha 6 subunit of the GABAA receptor is concentrated in both inhibitory and excitatory synapses on cerebellar granule cells

scientific journal article

The citalopram challenge test in patients with major depression and in healthy controls

scientific article published on 01 November 1999

The gamma 2 subunit of the GABAA receptor is concentrated in synaptic junctions containing the alpha 1 and beta 2/3 subunits in hippocampus, cerebellum and globus pallidus

scientific article published on 01 January 1996

The influence of phenotype on the outcome of linkage analysis of schizophrenia

scientific article published on 01 October 1996

The parvalbumin-positive interneurons in the mouse dentate gyrus express GABAA receptor subunits α1, β2, and δ along their extrasynaptic cell membrane

scientific article

The α1, α2, α3, and γ2 subunits of GABAA receptors show characteristic spatial and temporal expression patterns in rhombencephalic structures during normal human brain development

scientific article published on 31 October 2015

The α6 subunit-containing GABA receptor: A novel drug target for inhibition of trigeminal activation

scholarly article by Pi-Chuan Fan et al published 15 September 2018 in Neuropharmacology

Transient transfection coupled to baculovirus infection for rapid protein expression screening in insect cells

scientific article

Two novel residues in M2 of the gamma-aminobutyric acid type A receptor affecting gating by GABA and picrotoxin affinity.

scientific article published on 12 December 2000

Understanding subtype-selective allosteric modulation of GABAA receptors.

scientific article published on 17 September 2012

Unexpected Properties of δ-Containing GABAA Receptors in Response to Ligands Interacting with the α+ β- Site.

scientific article published on 26 September 2013

Unraveling the function of GABA(A) receptor subtypes.

scientific article

Unravelling the role of GABAA receptor subtypes in distinct neurons and behaviour

scientific article published on May 15, 2012

Uptake of taurine into subcellular fractions of C-6 glioma cells

scientific article published on May 1, 1976

Various proteins from rat brain, specifically and irreversibly labeled by [3H]flunitrazepam, are distinct alpha-subunits of the GABA-benzodiazepine receptor complex

scientific article published on 01 August 1988

[35S]tert.-butylbicyclophosphorothionate and avermectin bind to different sites associated with the gamma- aminobutyric acid-benzodiazepine receptor complex.

scientific article published in September 1984

[3H]propyl-6-azido-beta-carboline-3-carboxylate: a new photoaffinity label for the GABAA-benzodiazepine receptor.

scientific article published in July 1995

[Comparison of the bioavailability of two diazepam preparations. Clinical comparison between a new commercial preparation and a standard preparation after oral and intramuscular administration]

scientific article published on 01 April 1986

[Orally-administered taurine in therapy-resistant epilepsy (author's transl)]

scientific article published on 01 February 1977

gamma-Aminobutyric acid, acting through gamma -aminobutyric acid type A receptors, inhibits the biosynthesis of neurosteroids in the frog hypothalamus.

scientific article published on December 2000

gamma-Aminobutyric acidA receptors displaying association of gamma 3-subunits with beta 2/3 and different alpha-subunits exhibit unique pharmacological properties

scientific article