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List of works by Eiji Kawanishi

C-Glucosides with heteroaryl thiophene as novel sodium-dependent glucose cotransporter 2 inhibitors

scientific article published on June 4, 2013

Discovery of 2-[(E)-2-(7-Fluoro-3-methylquinoxalin-2-yl)vinyl]-6-pyrrolidin-1-yl-N-(tetrahydro-2H-pyran-4-yl)pyrimidin-4-amine Hydrochloride as a Highly Selective PDE10A Inhibitor

scientific article published on 01 January 2018

Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety

scientific article published on 19 June 2019

Discovery of canagliflozin, a novel C-glucoside with thiophene ring, as sodium-dependent glucose cotransporter 2 inhibitor for the treatment of type 2 diabetes mellitus.

scientific article published on September 2010

N-Glucosides as human sodium-dependent glucose cotransporter 2 (hSGLT2) inhibitors

scientific article published on 17 August 2013

Phosphodiesterase 10A PET Radioligand Development Program: From Pig to Human

article

Synthesis and biological evaluation of thiophene-C-glucosides as sodium-dependent glucose cotransporter 2 inhibitors.

scientific article published in January 2013

Synthesis and properties of GuNA purine/pyrimidine nucleosides and oligonucleotides

scientific article published on 12 November 2020

Synthetic Method for 2'-Amino-LNA Bearing Any of the Four Nucleobases via a Transglycosylation Reaction.

scientific article published on 12 March 2018

Tandem base-promoted ring opening/brook rearrangement/allylic alkylation of O-silyl cyanohydrins of beta-silyl-alpha,beta-epoxyaldehydes

scientific article published in May 2002

Tandem base-promoted ring-opening/Brook rearrangement/allylic alkylation of O-silyl cyanohydrins of beta-silyl-alpha,beta-epoxyaldehyde: scope and mechanism

scientific article published in November 2003