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List of works by Marco Lanza

Analgesic efficacy of CR4056, a novel imidazoline-2 receptor ligand, in rat models of inflammatory and neuropathic pain

scientific article

Biological profile and bioavailability of imidazoline compounds on morphine tolerance modulation.

scientific article published on 16 November 2015

CGP 52432: a novel potent and selective GABAB autoreceptor antagonist in rat cerebral cortex.

scientific article published in June 1993

CR4056, a new analgesic I2 ligand, is highly effective against bortezomib-induced painful neuropathy in rats.

scientific article

CR4056, a powerful analgesic imidazoline-2 receptor ligand, inhibits the inflammation-induced PKCε phosphorylation and membrane translocation in sensory neurons

scientific article published on 07 November 2019

Characterization of a novel putative cognition enhancer mediating facilitation of glycine effect on strychnine-resistant sites coupled to NMDA receptor complex ⬇️

scientific article published on August 1, 1997

Cholecystokinin (CCK) increases GABA release in the rat anterior nucleus accumbens via CCK(B) receptors located on glutamatergic interneurons

scientific article (publication date: 2000)

Cognition Enhancing Profile of CR 2249, a New NMDA-Glycine Site Modulator

Dendrimeric tetravalent ligands for the serotonin-gated ion channel

scientific article published on 23 June 2014

Development of subnanomolar-affinity serotonin 5-HT receptor ligands based on quinoline structures

scientific article published on 03 July 2018

Efficacy of CR4056, a first-in-class imidazoline-2 analgesic drug, in comparison with naproxen in two rat models of osteoarthritis.

scientific article

Experimental pharmacology of glucosamine sulfate.

scientific article published on 09 October 2011

Exploring multitarget interactions to reduce opiate withdrawal syndrome and psychiatric comorbidity

scientific article

Functional in vitro characterization of CR 3394: a novel voltage dependent N-methyl-D-aspartate (NMDA) receptor antagonist.

scientific article published on 19 October 2005

Improved efficacy, tolerance, safety and abuse liability profile of the combination CR4056-morphine over morphine alone in rodent models

scientific article published on 10 March 2020

Modulation of imidazoline I2 binding sites by CR4056 relieves postoperative hyperalgesia in male and female rats

scientific article

Multivalent ligands for the serotonin 5-HT receptor

scientific article published on 09 February 2017

Pharmacological characterisation of CR6086, a potent prostaglandin E2 receptor 4 antagonist, as a new potential disease-modifying anti-rheumatic drug.

scientific article published in March 2018

Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds

scientific article published on 8 February 2013

Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold.

scientific article

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