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List of works by Micha Fridman

6''-Thioether tobramycin analogues: towards selective targeting of bacterial membranes

scientific article published on 12 April 2012

A new class of branched aminoglycosides: pseudo-pentasaccharide derivatives of neomycin B

scientific article published on 01 October 2003

A synthetic pentasaccharide with GTPase activity

scientific article published on 01 December 2001

Antifungal Imidazole-Decorated Cationic Amphiphiles with Markedly Low Hemolytic Activity.

scientific article published on 3 June 2016

Antifungal activity, mode of action variability, and subcellular distribution of coumarin-based antifungal azoles

scientific article published on 02 July 2019

Antimycobacterial activity of DNA intercalator inhibitors of Mycobacterium tuberculosis primase DnaG.

scientific article published on 24 September 2014

Assessment of 6'- and 6'''-N-acylation of aminoglycosides as a strategy to overcome bacterial resistance

scientific article published in March 2011

Cationic Amphiphiles Induce Macromolecule Denaturation and Organelle Decomposition in Pathogenic Yeast

scientific article published on 11 November 2018

Cationic Pillararenes Potently Inhibit Biofilm Formation without Affecting Bacterial Growth and Viability

scientific article published on 8 January 2016

Characterization of non-dialyzable constituents from cranberry juice that inhibit adhesion, co-aggregation and biofilm formation by oral bacteria.

scientific article

Characterization of rhodosaminyl transfer by the AknS/AknT glycosylation complex and its use in reconstituting the biosynthetic pathway of aclacinomycin A.

scientific article published on 8 August 2007

Chemical Modifications Reduce Auditory Cell Damage Induced by Aminoglycoside Antibiotics

scientific article published on 29 January 2020

Chemoenzymatic Formation of Novel Aminocoumarin Antibiotics by the Enzymes CouN1 and CouN7†

scientific article published in 2007

Combining Colistin and Fluconazole Synergistically Increases Fungal Membrane Permeability and Antifungal Cidality

scientific article published on 20 January 2021

Derivatives of Ribosome-Inhibiting Antibiotic Chloramphenicol Inhibit the Biosynthesis of Bacterial Cell Wall.

scientific article published in May 2018

Design of membrane targeting tobramycin-based cationic amphiphiles with reduced hemolytic activity

article

Di-N-Methylation of Anti-Gram-Positive Aminoglycoside-Derived Membrane Disruptors Improves Antimicrobial Potency and Broadens Spectrum to Gram-Negative Bacteria.

scientific article published on 29 September 2015

Effects of 5-O-Ribosylation of Aminoglycosides on Antimicrobial Activity and Selective Perturbation of Bacterial Translation

scientific article published on 10 August 2016

Exploring the Effects of Glycosylation and Etherification of the Side Chains of the Anticancer Drug Mitoxantrone.

scientific article published on 31 July 2015

Fluorescent Tracking of the Endoplasmic Reticulum in Live Pathogenic Fungal Cells

scientific article published on 26 November 2018

Guiding Drugs to Target-Harboring Organelles: Stretching Drug-Delivery to a Higher Level of Resolution

scientific article published on 12 August 2019

Increased Degree of Unsaturation in the Lipid of Antifungal Cationic Amphiphiles Facilitates Selective Fungal Cell Disruption.

scientific article

Inhibition of glioma progression by a newly discovered CD38 inhibitor.

scientific article

Localizing Antifungal Drugs to the Correct Organelle Can Markedly Enhance their Efficacy

scientific article published on 25 March 2018

One-Pot Chemoenzymatic Cascade for Labeling of the Epigenetic Marker 5-Hydroxymethylcytosine

scientific article published on 27 July 2015

One-pot synthesis of glucosamine oligosaccharides

scientific article published on 01 January 2002

Phosphonium pillar[5]arenes as a new class of efficient biofilm inhibitors: importance of charge cooperativity and the pillar platform.

scientific article published on 9 August 2016

Real-Time Imaging of the Azole Class of Antifungal Drugs in Live Candida Cells.

scientific article

Serum Prevents Interactions between Antimicrobial Amphiphilic Aminoglycosides and Plasma Membranes

scientific article published on 11 November 2020

Structural insights of lincosamides targeting the ribosome of Staphylococcus aureus

scientific article published on September 2017

Synthesis and evaluation of hetero- and homodimers of ribosome-targeting antibiotics: antimicrobial activity, in vitro inhibition of translation, and drug resistance

scientific article published on July 2013

Synthesis and evaluation of membrane permeabilizing properties of cationic amphiphiles derived from the disaccharide trehalose.

scientific article published on 2 February 2016

Targeting anthracycline-resistant tumor cells with synthetic aloe-emodin glycosides

scientific article published on 12 May 2011

The relationship between the structure and toxicity of aminoglycoside antibiotics

scientific article published on 25 April 2020

The structure of anthracycline derivatives determines their subcellular localization and cytotoxic activity.

scientific article published on 4 February 2013

Tobramycin and nebramine as pseudo-oligosaccharide scaffolds for the development of antimicrobial cationic amphiphiles

scientific article published on 04 February 2015

Tuning the Effects of Bacterial Membrane Permeability through Photo-Isomerization of Antimicrobial Cationic Amphiphiles.

scientific article

Using biological performance similarity to inform disaccharide library design

scientific article

hChAT: a tool for the chemoenzymatic generation of potential acetyl/butyrylcholinesterase inhibitors.

scientific article published in September 2009

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