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List of works by Salvatore Bongarzone

Assessing the feasibility of intranasal radiotracer administration for in brain PET imaging

scientific article published on 30 August 2018

BACE1: Now We Can See You.

scientific article published on 4 April 2018

Carbon-11 Carboxylation of Trialkoxysilane and Trimethylsilane Derivatives Using [¹¹C]CO2

Carbon-11 carboxylation of trialkoxysilane and trimethylsilane derivatives using [11C]CO2

scientific article published on 25 March 2020

Complementary medicinal chemistry-driven strategies toward new antitrypanosomal and antileishmanial lead drug candidates

scientific article

Computational studies on the prion protein

scientific article

Development of [18F]FAMTO: A novel fluorine-18 labelled positron emission tomography (PET) radiotracer for imaging CYP11B1 and CYP11B2 enzymes in adrenal glands

scientific article published on 09 November 2018

Discovery of a class of diketopiperazines as antiprion compounds.

scientific article

Docking Ligands on Protein Surfaces: The Case Study of Prion Protein

Dominant-negative effects in prion diseases: insights from molecular dynamics simulations on mouse prion protein chimeras

scientific article published on 30 August 2012

Electrochemical [11C]CO2 to [11C]CO conversion for PET imaging

scientific article published on 24 February 2017

From [11C]CO2 to [11C]amides: a rapid one-pot synthesis via the Mitsunobu reaction.

scientific article published on 27 April 2017

Hybrid lipoic acid derivatives to attack prion disease on multiple fronts

scientific article published on 15 March 2011

Imaging biotin trafficking in vivo with positron emission tomography

scientific article published on 13 July 2020

Imaging niacin trafficking with positron emission tomography reveals in vivo monocarboxylate transporter distribution

scientific article published on 06 July 2020

Impact of [64Cu][Cu(ATSM)] PET/CT in the evaluation of hypoxia in a patient with Glioblastoma: a case report

scientific article published on 06 December 2019

In-loop flow [11 C]CO2 fixation and radiosynthesis of N,N'-[11 C]dibenzylurea

scientific article

Instantaneous Conversion of [11 C]CO2 to [11 C]CO via Fluoride-Activated Disilane Species.

scientific article

Molecular motions in drug design: the coming age of the metadynamics method

scientific article published on 17 February 2011

Multitarget ligands and theranostics: sharpening the medicinal chemistry sword against prion diseases.

scientific article

PET Imaging as a Tool for Assessing COVID-19 Brain Changes

Parallel synthesis, evaluation, and preliminary structure-activity relationship of 2,5-diamino-1,4-benzoquinones as a novel class of bivalent anti-prion compound

scientific article

Privileged structure-guided synthesis of quinazoline derivatives as inhibitors of trypanothione reductase

scientific article published on 20 April 2009

Quantification of [(11)C]PIB PET for imaging myelin in the human brain: a test-retest reproducibility study in high-resolution research tomography

scientific article

Radiolabeling of [11C]FPS-ZM1, a receptor for advanced glycation end products-targeting positron emission tomography radiotracer, using a [11C]CO2-to-[11C]CO chemical conversion

scientific article published on 26 February 2020

Rapid one-pot radiosynthesis of [carbonyl-11C]formamides from primary amines and [11C]CO2

scientific article published on 01 September 2020

Rational approach to an antiprion compound with a multiple mechanism of action

scientific article published on 29 October 2015

Structure-Driven Discovery of α,γ-Diketoacid Inhibitors Against UL89 Herpesvirus Terminase

scientific article published on 01 August 2018

Synthesis and evaluation of a library of 2,5-bisdiamino-benzoquinone derivatives as probes to modulate protein-protein interactions in prions

scientific article

Targeting the Receptor for Advanced Glycation Endproducts (RAGE): A Medicinal Chemistry Perspective.

scientific article published on 08 May 2017

The concept of privileged structures in rational drug design: focus on acridine and quinoline scaffolds in neurodegenerative and protozoan diseases

scientific article published on January 18, 2011

[(11)C]CO2 to [(11)C]CO conversion mediated by [(11)C]silanes: a novel route for [(11)C]carbonylation reactions.

scientific article published in July 2015