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List of works by Reik Löser

2-(diethylamino)thieno1,3ŏxazin-4-ones as stable inhibitors of human leukocyte elastase

scientific article published on 01 December 1999

A fluorescence anisotropy-based assay for determining the activity of tissue transglutaminase.

scientific article published on 17 February 2016

Active Site Mapping of Human Cathepsin F with Dipeptide Nitrile Inhibitors

scientific article published on 26 June 2015

Antimalarial activity of azadipeptide nitriles

scientific article

Cathepsin B: Active site mapping with peptidic substrates and inhibitors

scientific article published on 19 October 2018

Cathepsin S inhibitors: WO2010070615 ⬇️

scientific article published on January 20, 2011

Characterization of Tissue Transglutaminase as a Potential Biomarker for Tissue Response toward Biomaterials

scientific article published on 18 October 2019

Corrigendum: Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminase 2

scientific article published on 16 August 2016

Cyclopeptides containing the DEKS motif as conformationally restricted collagen telopeptide analogues: synthesis and conformational analysis.

scientific article

Cysteine cathepsins: their role in tumor progression and recent trends in the development of imaging probes

scientific article

Dipeptide-derived nitriles containing additional electrophilic sites: potentially irreversible inhibitors of cysteine proteases.

scientific article published in December 2009

Evaluation of Fluorine-18-Labeled α1(I)-N-Telopeptide Analogs as Substrate-Based Radiotracers for PET Imaging of Melanoma-Associated Lysyl Oxidase.

scientific article published on 26 April 2018

Microplate assay for quantitative determination of cathepsin activities in viable cells using derivatives of 4-methoxy-beta-naphthylamide.

scientific article published on October 2006

Nε-Acryloyllysine Piperazides as Irreversible Inhibitors of Transglutaminase 2: Synthesis, Structure-Activity Relationships, and Pharmacokinetic Profiling

scientific article published on 10 May 2018

Rational Structure-Based Rescaffolding Approach to De Novo Design of Interleukin 10 (IL-10) Receptor-1 Mimetics

scientific article

Site-selective radiolabeling of peptides by (18)F-fluorobenzoylation with [(18F)]SFB in solution and on solid phase: a comparative study

scientific article published on 01 October 2012

Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminase 2.

scientific article

Synthesis and preliminary radiopharmacological characterisation of an 11 C-labelled azadipeptide nitrile as potential PET tracer for imaging of cysteine cathepsins

scientific article published on 15 May 2019

Synthesis, 18F-labelling and radiopharmacological characterisation of the C-terminal 30mer of Clostridium perfringens enterotoxin as a potential claudin-targeting peptide

scientific article published on 27 September 2018

Targeting lysyl oxidase for molecular imaging in breast cancer

scientific article

The Pyrazolo[3,4-d]pyrimidine-Based Kinase Inhibitor NVP-BHG712: Effects of Regioisomers on Tumor Growth, Perfusion, and Hypoxia in EphB4-Positive A375 Melanoma Xenografts

scientific article published on 03 November 2020

Tissue transglutaminase: an emerging target for therapy and imaging.

scientific article published on December 2013

Tos-Nos-Mos: Synthesis of different aryl sulfonate precursors for the radiosynthesis of the alpha7 nicotinic acetylcholine receptor radioligand [(18)F]NS14490.

scientific article published on 28 April 2016

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