List of works - Daniel Conole

3,5-Dialkoxypyridine analogues of bedaquiline are potent antituberculosis agents with minimal inhibition of the hERG channel

scientific article published on 15 February 2019

6-Cyano Analogues of Bedaquiline as Less Lipophilic and Potentially Safer Diarylquinolines for Tuberculosis

scientific article

Biophysical screening methods for extracellular domain peptide receptors, application to natriuretic peptide receptor C ligands

scientific article published on 10 October 2018

Chemical Instability and Promiscuity of Arylmethylidenepyrazolinone-Based MDMX Inhibitors

scientific article published on 19 September 2018

Discovery of a novel fluorescent chemical probe suitable for evaluation of neuropilin-1 binding of small molecules

scientific article published on 20 January 2020

Fatty Acid-Derived Pro-Toxicants of the Rat Selective Toxicant Norbormide

scientific article published on 4 May 2016

Prodrugs of N-dicarboximide derivatives of the rat selective toxicant norbormide

scientific article published in September 2013

Recent Developments in Cell Permeable Deubiquitinating Enzyme Activity-Based Probes

scientific article published on 18 December 2019

Structure-activity relationships for analogs of the tuberculosis drug bedaquiline with the naphthalene unit replaced by bicyclic heterocycles

scientific article published on 20 February 2018

Structure-activity relationships for unit C pyridyl analogues of the tuberculosis drug bedaquiline

scientific article published on 15 February 2019

Synthesis and methemoglobinemia-inducing properties of analogues of para-aminopropiophenone designed as humane rodenticides

scientific article published on 31 October 2013

Synthesis and methemoglobinemia-inducing properties of benzocaine isosteres designed as humane rodenticides

scientific article published on 20 February 2014

Synthesis and structure-activity relationships for tetrahydroisoquinoline-based inhibitors of Mycobacterium tuberculosis

scientific article published on 24 September 2020

Synthetic Studies to Help Elucidate the Metabolism of the Preclinical Candidate TBAJ-876-A Less Toxic and More Potent Analogue of Bedaquiline

scientific article published on 20 March 2020

Targeting STAT3 signaling using stabilised sulforaphane (SFX-01) inhibits endocrine resistant stem-like cells in ER-positive breast cancer

scientific article published on 30 May 2020

The maturation of DNA encoded libraries: opportunities for new users

scientific article published on 04 December 2020

List of works by Daniel Conole