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List of works by Nicolas Inguimbert

Access to α,α-Disubstituted Disilylated Amino Acids and Their Use in Solid-Phase Peptide Synthesis

scientific article published on 08 September 2015

Asp218 participates with Asp213 to bind a Ca2+ atom into the S1 subsite of aminopeptidase A: a key element for substrate specificity.

scientific article published in November 2008

Biochemical and structural analysis of the binding determinants of a vascular endothelial growth factor receptor peptidic antagonist

scientific article published on June 2010

Biological Activities of Cyclic and Acyclic B-Type Laxaphycins in SH-SY5Y Human Neuroblastoma Cells

scientific article published on 15 July 2020

Biophysical Studies of the Induced Dimerization of Human VEGF Receptor 1 Binding Domain by Divalent Metals Competing with VEGF-A.

scientific article

Characterization of a new anticancer agent, EAPB0203, and its main metabolites: nuclear magnetic resonance and liquid chromatography-mass spectrometry studies

scientific article published on 31 October 2012

Chemiluminescence immunoassays for estradiol and ethinylestradiol based on new biotinylated estrogen derivatives.

scientific article published in September 2017

Cooperation and cheating orchestrate Vibrio assemblages and polymicrobial synergy in oysters infected with OsHV-1 virus

scientific article published in 2023

Development and validation of LC-MS methods for peptaibol quantification in fungal extracts according to their lengths.

scientific article published on 4 December 2015

Development of a chemiluminescent screening assay for detection of vascular endothelial growth factor receptor 1 ligands

scientific article published on 30 March 2007

Disulfide and amide-bridged cyclic peptide analogues of the VEGF81–91 fragment: Synthesis, conformational analysis and biological evaluation

article

Efficient microwave-assisted one shot synthesis of peptaibols using inexpensive coupling reagents

scientific article published on 12 March 2014

Enhancing the Antimicrobial Activity of Alamethicin F50/5 by Incorporating N-terminal Hydrophobic Triazole Substituents.

scientific article published on 18 September 2017

Exploration of the S(')(1) subsite of neprilysin: a joined molecular modeling and site-directed mutagenesis study

scientific article published on 01 June 2000

First total synthesis and stereochemical revision of laxaphycin B and its extension to lyngbyacyclamide A

scientific article published on 15 July 2013

Helical peptides from VEGF and Vammin hotspots for modulating the VEGF-VEGFR interaction.

scientific article published on 4 February 2013

How are 1,2,3-triazoles accommodated in helical secondary structures?

scientific article published on 25 April 2018

Immunosensors for estradiol and ethinylestradiol based on new synthetic estrogen derivatives: application to wastewater analysis.

scientific article published on 30 January 2013

Isolation and Synthesis of Laxaphycin B-Type Peptides: A Case Study and Clues to Their Biosynthesis.

scientific article published on 5 December 2015

NI956/QGC006, a Potent Orally Active, Brain-Penetrating Aminopeptidase A Inhibitor for Treating Hypertension

scientific article published on 01 June 2019

On-resin cyclization of peptide ligands of the Vascular Endothelial Growth Factor Receptor 1 by copper(I)-catalyzed 1,3-dipolar azide-alkyne cycloaddition

scientific article published on 22 August 2007

Oxovanadium-salen and -salan complexes as effective labels for electrochemical immunosensing: a case study for estradiol detection

scientific article published on 01 February 2014

Parallel solid-phase synthesis of a small library of linear and hydrocarbon-bridged analogues of VEGF(81-91): potential biological tools for studying the VEGF/VEGFR-1 interaction.

scientific article

Peptaibols as a model for the insertions of chemical modifications

scientific article published on 20 September 2018

Photodegradation of Myrigalone A, an Allelochemical from Myrica gale: Photoproducts and Effect of Terpenes

scientific article published on 25 June 2019

Rational design, structure, and biological evaluation of cyclic peptides mimicking the vascular endothelial growth factor.

scientific article

Salen/salan metallic complexes as redox labels for electrochemical aptasensors

scientific article published on 09 October 2019

Soluble fms-like tyrosine kinase-1 antibody for diagnosis purposes (WO2010075475)

scientific article published on 21 April 2011

Straightforward strategy to substitute amide bonds by 1,2,3-triazoles in peptaibols analogs using Aibψ[Tz]-Xaa dipeptides

scientific article published on 18 March 2015

Structure and biological evaluation of new cyclic and acyclic laxaphycin-A type peptides

scientific article published on 26 March 2019

Structure-based design of a bicyclic peptide antagonist of the vascular endothelial growth factor receptors.

scientific article published on June 2008

Synthesis and in vitro activities of new non-peptidic APA inhibitors.

scientific article published in February 2005

Targeting VEGFR1 on endothelial progenitors modulates their differentiation potential.

scientific article published on 14 January 2014

Towards the total synthesis of trichormamide A, a cyclic undecapeptide

scientific article published in 2018

Trichormamide C Structural Confirmation through Total Synthesis and Extension to Analogs

scientific article published on 19 December 2019