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List of works by Kurt Vermeire

135 Safety Concerns for Cyanovirin as a Microbicidal Anti-HIV Agent

article

A Proteomic Study on the Membrane Protein Fraction of T Cells Confirms High Substrate Selectivity for the ER Translocation Inhibitor Cyclotriazadisulfonamide

scientific article published on 02 September 2021

A Proteomic Survey Indicates Sortilin as a Secondary Substrate of the ER Translocation Inhibitor Cyclotriazadisulfonamide (CADA).

scientific article published on 20 December 2016

Anti-HIV agents targeting the interaction of gp120 with the cellular CD4 receptor

scientific article published in October 2005

CADA inhibits human immunodeficiency virus and human herpesvirus 7 replication by down-modulation of the cellular CD4 receptor

scientific article published on October 2002

CADA, a Potential Anti-HIV Microbicide that Specifically Targets the Cellular CD4 Receptor

article

CADA, a novel CD4-targeted HIV inhibitor, is synergistic with various anti-HIV drugs in vitro

scientific article

CADA, a potential anti-HIV microbicide that specifically targets the cellular CD4 receptor

scientific article published in May 2008

CD4 down-modulating compounds with potent anti-HIV activity

scientific article published on January 2004

Carbohydrate-binding agents efficiently prevent dendritic cell-specific intercellular adhesion molecule-3-grabbing nonintegrin (DC-SIGN)-directed HIV-1 transmission to T lymphocytes

scientific article published on 20 October 2006

Chlorogenic Compounds from Coffee Beans Exert Activity against Respiratory Viruses.

scientific article published on 2 November 2016

Cyclotriazadisulfonamides: promising new CD4-targeted anti-HIV drugs

scientific article

Design and cellular kinetics of dansyl-labeled CADA derivatives with anti-HIV and CD4 receptor down-modulating activity

scientific article

Development and in vitro evaluation of chloroquine gels as microbicides against HIV-1 infection

scientific article

Early identification of availability issues for poorly water-soluble microbicide candidates in biorelevant media: a case study with saquinavir

scientific article published on 6 June 2011

Endothelial dysfunction in dengue virus pathology

scientific article

Establishment of a novel CCR5 and CXCR4 expressing CD4+ cell line which is highly sensitive to HIV and suitable for high-throughput evaluation of CCR5 and CXCR4 antagonists

scientific article

Evaluation of SDF-1/CXCR4-induced Ca2+ signaling by fluorometric imaging plate reader (FLIPR) and flow cytometry

scientific article published on January 2003

Fluorescent CXCL12AF647 as a novel probe for nonradioactive CXCL12/CXCR4 cellular interaction studies

scientific article published on October 2004

Human immunodeficiency virus type 1 escape from cyclotriazadisulfonamide-induced CD4-targeted entry inhibition is associated with increased neutralizing antibody susceptibility

scientific article

Immunomodulatory properties of interferon-gamma. An update

scientific article published on 01 September 1998

Improving potencies and properties of CD4 down-modulating CADA analogs

scientific article published on 06 December 2011

Inhibition of human immunodeficiency virus replication by a dual CCR5/CXCR4 antagonist

scientific article published on December 2004

Inhibitors of HIV infection via the cellular CD4 receptor

scientific article

Inhibitors of protein translocation across membranes of the secretory pathway: novel antimicrobial and anticancer agents.

scientific article published on 5 January 2018

Mac-1(+) myelopoiesis induced by CFA: a clue to the paradoxical effects of IFN-gamma in autoimmune disease models.

scientific article

Mannose-specific plant lectins from the Amaryllidaceae family qualify as efficient microbicides for prevention of human immunodeficiency virus infection

scientific article published on October 2004

Mechanistic Studies on a Novel Hydrophobic Derivative of Aglycoristocetin with Potent and Broad Activity Against Influenza Viruses

article published in 2011

Metal complexes of pyridine-fused macrocyclic polyamines targeting the chemokine receptor CXCR4.

scientific article published on 4 September 2015

Microvirin, a novel alpha(1,2)-mannose-specific lectin isolated from Microcystis aeruginosa, has anti-HIV-1 activity comparable with that of cyanovirin-N but a much higher safety profile

scientific article

Modest human immunodeficiency virus coreceptor function of CXCR3 is strongly enhanced by mimicking the CXCR4 ligand binding pocket in the CXCR3 receptor

scientific article published on 24 January 2007

Mutations at the CXCR4 interaction sites for AMD3100 influence anti-CXCR4 antibody binding and HIV-1 entry

scientific article published in July 2003

Preprotein signature for full susceptibility to the co-translational translocation inhibitor cyclotriazadisulfonamide

scientific article published on 25 November 2019

Pro-inflammatory properties of stromal cell-derived factor-1 (CXCL12) in collagen-induced arthritis

scientific article

Profile of Resistance of Human Immunodeficiency Virus to Mannose-Specific Plant Lectins

article

Profile of resistance of human immunodeficiency virus to mannose-specific plant lectins

scientific article published on October 2004

Resistance mutations in human immunodeficiency virus type 1 integrase selected with elvitegravir confer reduced susceptibility to a wide range of integrase inhibitors

scientific article published on 20 August 2008

Resistance of HIV-1 to the broadly HIV-1-neutralizing, anti-carbohydrate antibody 2G12.

scientific article published on 21 November 2006

Ribonuclease-neutralized pancreatic microsomal membranes from livestock for in vitro co-translational protein translocation.

scientific article published on 4 June 2015

Safety concerns for the potential use of cyanovirin-N as a microbicidal anti-HIV agent

article

Signal peptide-binding drug as a selective inhibitor of co-translational protein translocation

scientific article (publication date: December 2014)

Specific CD4 down-modulating compounds with potent anti-HIV activity

scientific article

Sugar-binding proteins potently inhibit dendritic cell human immunodeficiency virus type 1 (HIV-1) infection and dendritic-cell-directed HIV-1 transfer

scientific article

Synergistic in vitro anti-HIV type 1 activity of tenofovir with carbohydrate-binding agents (CBAs).

scientific article published on 8 April 2011

Synthesis and structure-activity relationship studies of CD4 down-modulating cyclotriazadisulfonamide (CADA) analogues

scientific article published on February 2006

Synthesis of CADA Analog Prodrugs Designed as Novel Down-modulators of the CD4 Receptor

scientific article published in 2009

Synthesis of Novel CADA Analog Prodrugs Designed as Down-Modulators of the CD4 Receptor

scientific article published in 2011

The Anti-HIV potency of cyclotriazadisulfonamide analogs is directly correlated with their ability to down-modulate the CD4 receptor

scientific article

The antiviral activity of the CXCR4 antagonist AMD3100 is independent of the cytokine-induced CXCR4/HIV coreceptor expression level

scientific article

The candidate sulfonated microbicide, PRO 2000, has potential multiple mechanisms of action against HIV-1

article

Toward Unsymmetrical CADA Analogs as Novel Down-modulators of the CD4 Receptor

scientific article published in 2009

Tuning Side Arm Electronics in Unsymmetrical Cyclotriazadisulfonamide (CADA) Endoplasmic Reticulum (ER) Translocation Inhibitors to Improve their Human Cluster of Differentiation 4 (CD4) Receptor Down-Modulating Potencies.

scientific article published on 14 March 2016

Unsymmetrical cyclotriazadisulfonamide (CADA) compounds as human CD4 receptor down-modulating agents

scientific article published on 29 July 2011

Use of a sequential high throughput screening assay to identify novel inhibitors of the eukaryotic SRP-Sec61 targeting/translocation pathway

scientific article published in PLoS ONE

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