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List of works by Henriëtte M.G. Willems

2,3-Substituted 2-azanorbornanes as polar β-turn mimetics

scientific article published in 1997

De novo ligand design to partially flexible active sites: application of the ReFlex algorithm to carboxypeptidase A, acetylcholinesterase, and the estrogen receptor

scientific article published on 31 January 2008

Generation and selection of novel estrogen receptor ligands using the de novo structure-based design tool, SkelGen.

scientific article

Identification and Investigation of Novel Binding Fragments in the Fatty Acid Binding Protein 6 (FABP6)

scientific article

Isoindolinone-based inhibitors of the MDM2-p53 protein-protein interaction.

scientific article published on March 2005

Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery

scientific article

Receptor flexibility in the in silico screening of reagents in the S1' pocket of human collagenase

scientific article published in May 2004

Small-molecule inhibitors of the MDM2-p53 protein-protein interaction based on an isoindolinone scaffold

scientific article

Structural Biology and Anticancer Drug Design

Structure-Activity and Structure-Conformation Relationships of Aryl Propionic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1/Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1/NRF2) Protein-Protein Interaction

scientific article published on 25 April 2019

The design of dipeptide helical mimetics, Part I: the synthesis of 1,6-disubstituted indanes

article

The design of dipeptide helical mimetics: The synthesis, tachykinin receptor affinity and conformational analysis of 1,1,6-trisubstituted indanes

article

The design of dipeptide helical mimetics: the synthesis and biological activity of trisubstituted indanes

article

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