List of works - Dale L. Boger

C1-CBP-vancomycin: Impact of a Vancomycin C-Terminus Trimethylammonium Cation on Pharmacological Properties and Insights into Its Newly Introduced Mechanism of Action

scientific article published on 31 October 2019

Design of Benzoxathiazin-3-one 1,1-Dioxides as a New Class of Irreversible Serine Hydrolase Inhibitors: Discovery of a Uniquely Selective PNPLA4 Inhibitor.

scientific article published on 12 May 2017

Diprovocims: A New and Exceptionally Potent Class of Toll-like Receptor Agonists

scientific article published on 16 October 2018

Direct Synthesis of β-Aminoenals through Reaction of 1,2,3-Triazine with Secondary Amines

scientific article published on 28 June 2017

Discovery of small-molecule enzyme activators by activity-based protein profiling

scientific article published on 08 June 2020

Divergent Total Syntheses of (-)-Pseudocopsinine and (-)-Minovincinine

scientific article published on 18 November 2020

Inverse Electron Demand Diels-Alder Reactions of Heterocyclic Azadienes, 1-Aza-1,3-Butadienes, Cyclopropenone Ketals, and Related Systems. A Retrospective

scientific article published on 23 May 2019

Maxamycins: Durable Antibiotics Derived by Rational Redesign of Vancomycin

scientific article published on 02 November 2020

N-Terminus Alkylation of Vancomycin: Ligand Binding Affinity, Antimicrobial Activity, and Site-Specific Nature of Quaternary Trimethylammonium Salt Modification

scientific article published on 08 August 2018

Next-Generation Total Synthesis of Vancomycin

scientific article published on 04 September 2020

Selective N1/N4 1,4-Cycloaddition of 1,2,4,5-Tetrazines Enabled by Solvent Hydrogen Bonding

scientific article published on 30 November 2020

Small Molecular Weapons against Multi-Drug Resistance

scientific article published in 2021

Structural Basis of TLR2/TLR1 Activation by the Synthetic Agonist Diprovocim

scientific article published on 13 March 2019

Structural evolution of a DNA repair self-resistance mechanism targeting genotoxic secondary metabolites

scientific article published on 26 November 2021

Synthesis, Characterization, and Cycloaddition Reactivity of a Monocyclic Aromatic 1,2,3,5-Tetrazine

scientific article published on 02 October 2019

Synthesis, Characterization, and Rapid Cycloadditions of 5-Nitro-1,2,3-triazine

scientific article published on 16 April 2018

The Difference a Single Atom Can Make: Synthesis and Design at the Chemistry-Biology Interface.

scientific article published on 25 September 2017

The quest for supernatural products: the impact of total synthesis in complex natural products medicinal chemistry

scientific article published on 10 November 2020

Total Syntheses of Vancomycin-Related Glycopeptide Antibiotics and Key Analogues

scientific article

Total Synthesis and Stereochemical Assignment of Streptide

scientific article published on 17 October 2019

Total Synthesis of Meayamycin and O-Acyl Analogues

scientific article published on 19 October 2020

Triarylaminium Radical Cation Promoted Coupling of Catharanthine with Vindoline: Diastereospecific Synthesis of Anhydrovinblastine and Reaction Scope

scientific article published on 03 September 2019

Vinblastine 20' Amides: Synthetic Analogues That Maintain or Improve Potency and Simultaneously Overcome Pgp-Derived Efflux and Resistance