Search filters

Authors whose works are in public domain in at least one jurisdiction

List of works by Thierry Durroux

A Broad G Protein-Coupled Receptor Internalization Assay that Combines SNAP-Tag Labeling, Diffusion-Enhanced Resonance Energy Transfer, and a Highly Emissive Terbium Cryptate

scientific article published on 9 November 2015

A Fluorescent Ligand-Binding Alternative Using Tag-lite® Technology ⬇️

scientific article published on October 25, 2010

BRET and Time-resolved FRET strategy to study GPCR oligomerization: from cell lines toward native tissues.

scientific article

Background calcium permeable channels in glomerulosa cells from adrenal gland

scientific article published on August 1, 1992

Building a new conceptual framework for receptor heteromers

scientific article

Characterization of K+ and Ca2+ ionic currents in glomerulosa cells from human adrenal glands

scientific article published on 01 June 1994

Chemoselective Acylation of Hydrazinopeptides to Access Fluorescent Probes for Time-Resolved FRET Assays on GPCRs

scientific article published on 01 January 2019

Comparison of vasopressin and oxytocin receptors in the rat uterus and vascular tissue

scientific article published on 01 July 1996

Context-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3

scientific article published on 15 May 2019

Design and validation of a homogeneous time-resolved fluorescence cell-based assay targeting the ligand-gated ion channel 5-HT3A.

scientific article published on 18 May 2015

Design of peptide oxytocin antagonists with strikingly higher affinities and selectivities for the human oxytocin receptor than atosiban

scientific article published in October 2005

Distribution of signaling molecules involved in vasopressin-induced Ca2+ mobilization in rat hepatocyte multiplets

scientific article published on 01 May 1999

Effects of Adrenocorticotropin on Action Potential and Calcium Currents in Cultured Rat and Bovine Glomerulosa Cells* ⬇️

scientific article published on October 1, 1991

Expression of human vasopressin and oxytocin receptors in Escherichia coli.

scientific article

Fluorescent agonists and antagonists for vasopressin/oxytocin G protein-coupled receptors: usefulness in ligand screening assays and receptor studies.

scientific article published on September 2008

Fluorescent ligands to investigate GPCR binding properties and oligomerization.

scientific article

Fluorescent pseudo-peptide linear vasopressin antagonists: design, synthesis, and applications

scientific article published on 01 April 1999

From the Promiscuous Asenapine to Potent Fluorescent Ligands Acting at a Series of Aminergic G-Protein-Coupled Receptors

scientific article published on 8 December 2017

Leukotriene BLT2 receptor monomers activate the G(i2) GTP-binding protein more efficiently than dimers

scientific article

Membrane-delimited G protein-mediated coupling between V1a vasopressin receptor and dihydropyridine binding sites in rat glomerulosa cells

scientific article published in November 1996

Multicolor time-resolved Förster resonance energy transfer microscopy reveals the impact of GPCR oligomerization on internalization processes

scientific article published on 17 February 2015

Natural amines inhibit activation of human plasmacytoid dendritic cells through CXCR4 engagement

scientific article published on 09 February 2017

Oligomerization of a G protein-coupled receptor in neurons controlled by its structural dynamics.

scientific article published on 10 July 2018

Original Fluorescent Ligand-Based Assays Open New Perspectives in G-Protein Coupled Receptor Drug Screening.

scientific article

Oxytocin and Vasopressin V1a and V2 Receptors Form Constitutive Homo- and Heterodimers during Biosynthesis

scientific article published on 23 December 2002

Oxytocin and vasopressin agonists and antagonists as research tools and potential therapeutics

scientific article

Past, present and future of vasopressin and oxytocin receptor oligomers, prototypical GPCR models to study dimerization processes.

scientific article

Peptide and non-peptide agonists and antagonists for the vasopressin and oxytocin V1a, V1b, V2 and OT receptors: research tools and potential therapeutic agents

scientific article

Pharmacological evidence for a metabotropic glutamate receptor heterodimer in neuronal cells

scientific article

Pharmacology of oxytocin and vasopressin receptors in the central and peripheral nervous system.

scientific article

Principles: a model for the allosteric interactions between ligand binding sites within a dimeric GPCR.

scientific article

Probing the existence of G protein-coupled receptor dimers by positive and negative ligand-dependent cooperative binding.

scientific article published on 22 August 2006

Selective fluorescent nonpeptidic antagonists for vasopressin V₂ GPCR: application to ligand screening and oligomerization assays

scientific article published on 05 October 2012

Selective nonpeptidic fluorescent ligands for oxytocin receptor: design, synthesis, and application to time-resolved FRET binding assay

scientific article published on 12 February 2015

Structural bases of vasopressin/oxytocin receptor function ⬇️

scientific article published on February 1, 1998

Structural insights into biased G protein-coupled receptor signaling revealed by fluorescence spectroscopy ⬇️

scientific article published on April 9, 2012

Subtlety of the structure-affinity and structure-efficacy relationships around a nonpeptide oxytocin receptor agonist.

scientific article published in February 2010

Synthesis and characterization of fluorescent antagonists and agonists for human oxytocin and vasopressin V(1)(a) receptors.

scientific article published in June 2002

The constitutively active V2 receptor mutants conferring NSIAD are weakly sensitive to agonist and antagonist regulation

scientific article

The oligomeric state sets GABA(B) receptor signalling efficacy

scientific journal article

Time resolved FRET strategy with fluorescent ligands to analyze receptor interactions in native tissues: application to GPCR oligomerization.

scientific article published in January 2011

Time-Resolved FRET-Based Assays to Characterize G Protein-Coupled Receptor Hetero-oligomer Pharmacology

scientific article published on 01 January 2019

Time-resolved FRET between GPCR ligands reveals oligomers in native tissues.

scientific article

Time-resolved FRET binding assay to investigate hetero-oligomer binding properties: proof of concept with dopamine D1/D3 heterodimer.

scientific article published on 11 November 2014

Time-resolved FRET strategy to screen GPCR ligand library

scientific article published on January 2015

Toward efficient drug screening by homogeneous assays based on the development of new fluorescent vasopressin and oxytocin receptor ligands.

scientific article published on 12 September 2007

Untangling dopamine-adenosine receptor-receptor assembly in experimental parkinsonism in rats

scientific article

V1b vasopressin receptor trafficking and signaling : role of arrestins, G proteins and Src kinase.

scientific article

Vasoactive intestinal polypeptide and carbachol act synergistically to induce the hydrolysis of inositol containing phospholipids in the rat superior cervical ganglion

scientific article published on 01 March 1987

Vasopressin regulates adrenal functions by acting through different vasopressin receptor subtypes.

scientific article

Visualization of cell surface vasopressin V1a receptors in rat hepatocytes with a fluorescent linear antagonist

scientific article published on 01 March 1999

Paulina is supported by:

About Paulina

Help