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List of works by Saïd Yous

Antagonists of the adenosine A2A receptor based on a 2-arylbenzoxazole scaffold: Investigation of the C5- and C7-positions to enhance affinity

scientific article published on 5 December 2017

Antioxidant activity of benzoxazolinonic and benzothiazolinonic derivatives in the LDL oxidation model.

scientific article published on 15 September 2009

Antioxidant activity of melatonin and a pinoline derivative on linoleate model system.

scientific article published in August 2005

Antioxydant activity of β-carboline derivatives in the LDL oxidation model

scientific article published on 30 March 2011

Bitopic fluorescent antagonists of the A2A adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners

scientific article

Carbazole scaffolds in cancer therapy: a review from 2012 to 2018

scientific article published on 01 December 2019

Comparison of 3D structures and AT(1) binding properties of pyrazolidine-3,5-diones and tetrahydropyridazine-3,6-diones with parent antihypertensive drug irbesartan.

scientific article published in October 2002

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Part II.

scientific article published on 18 March 2009

Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3.

scientific article published on 17 March 2008

Design and synthesis of fused tetrahydroisoquinoline-iminoimidazolines

scientific article published on 19 October 2015

Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3

scientific article published on 15 February 2011

Design and synthesis of naphthalenic dimers as selective MT1 melatoninergic ligands

scientific article published on March 2003

Design of experiments for enantiomeric separation in supercritical fluid chromatography

scientific article published on 28 December 2015

Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A2A receptor.

scientific article published in December 2017

Design, synthesis and pharmacological evaluation of new series of naphthalenic analogues as melatoninergic (MT1/MT2) and serotoninergic 5-HT2C dual ligands (I).

scientific article published on 20 January 2012

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands

scientific article

Dual CD system in capillary electrophoresis for direct separation of the four stereoisomers of agonist and antagonist melatoninergic ligands.

scientific article published in May 2010

Enantiomeric resolution of new aromatase inhibitors by liquid chromatography on cellulose chiral stationary phases.

scientific article published in March 2005

Enantioseparation and thermodynamic study of naphthalene derivatives, new melatoninergic agonists, on coated amylose [tris(S)-1-phenylethylcarbamate] stationary phase. Transposition to preparative scale.

scientific article

Enhanced detection for determination of enantiomeric purity of novel agomelatine analogs by EKC using single and dual cyclodextrin systems

scientific article published on 28 July 2014

Exposure to glycol ethers in a population of French men evaluated by measurement of urinary alkoxycarboxylic acids.

scientific article

Homology modeling of MT1 and MT2 receptors

scientific article published on 14 December 2007

Homology modelling of the serotoninergic 5-HT2c receptor

scientific article

Increased susceptibility of low-density lipoprotein to ex vivo oxidation in mice transgenic for human apolipoprotein B treated with 1 melatonin-related compound is not associated with atherosclerosis progression

scientific article published in September 2005

Interactions of bexarotene (LGD1069, Targretin) with the coagulation system

scientific article published on 13 January 2011

Investigations of new lead structures for the design of novel cyclooxygenase-2 inhibitors

scientific article published in June 2002

Lipid-lowering properties of 6-benzoyl-2(3H)-benzothiazolone and structurally related compounds

scientific article published in December 2005

Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives

scientific article published on 29 December 2015

New melatonin (MT1/MT2) ligands: design and synthesis of (8,9-dihydro-7H-furo[3,2-f]chromen-1-yl) derivatives

scientific article published on 3 January 2014

New naphthalenic ligands of melatoninergic receptors

scientific article published on 01 July 1992

New phenylaniline derivatives as modulators of amyloid protein precursor metabolism

scholarly article by Marion Gay published in May 2018

New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation

scientific article published on 3 January 2017

New substrate analogues of human serotonin N-acetyltransferase produce in situ specific and potent inhibitors

scientific article (publication date: 2004)

Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARgamma agonists

scientific article published on 02 August 2006

Novel conformationally constrained analogues of agomelatine as new melatoninergic ligands.

scientific article published on 24 December 2012

Novel naphthalenic ligands with high affinity for the melatonin receptor

scientific article (publication date: 17 April 1992)

Old and new inhibitors of quinone reductase 2.

scientific article published on 04 May 2010

Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands

scientific article published on 23 February 2011

Preparative HPLC separation of methoxytetralins, ligands for melatonin receptors, containing two chiral centers with polysaccharide chiral stationary phases. Determination of enantiomeric purity.

scientific article published in July 2005

Quantification of the water/lipid affinity of melatonin and a pinoline derivative in lipid models

scientific article published on 01 April 2007

Quantitative structure-activity relationships studies of antioxidant hexahydropyridoindoles and flavonoid derivatives

scientific article

Rexinoid bexarotene modulates triglyceride but not cholesterol metabolism via gene-specific permissivity of the RXR/LXR heterodimer in the liver

scientific article

Structural basis of ligand recognition at the human MT1 melatonin receptor

scientific article published on 24 April 2019

Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT1/MT2) and serotoninergic (5-HT2C) dual ligands

scientific article published on 12 October 2017

Synthesis and evaluation of benzoxazolinonic imidazoles and derivatives as non-steroidal aromatase inhibitors

scientific article

Synthesis and pharmacological evaluation of a series of the agomelatine analogues as melatonin MT1 /MT2 agonist and 5-HT2C antagonist

scientific article published on 12 September 2013

Synthesis and pharmacological evaluation of analgesic 6-substituted 2(3H)-benzothiazolones

scientific article (publication date: 2001)

Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II).

scientific article published on 13 December 2014

Synthesis of 3-phenylnaphthalenic derivatives as new selective MT(2) melatoninergic ligands.

scientific article published on 27 August 2008

Synthesis of nitroindole derivatives with high affinity and selectivity for melatoninergic binding sites MT(3).

scientific article

Targeting peroxisome proliferator-activated receptors (PPARs): development of modulators.

scientific article published on 27 February 2012

The RXR Agonist Bexarotene Improves Cholesterol Homeostasis and Inhibits Atherosclerosis Progression in a Mouse Model of Mixed Dyslipidemia

article

Three-Dimensional Quantitative Structure–Activity Relationship ofMT3 Melatonin Binding Site Ligands: A Comparative Molecular Field Analysis

Three-dimensional quantitative structure-activity relationships of cyclo-oxygenase-2 (COX-2) inhibitors: a comparative molecular field analysis.

scientific article published in September 2001

XFEL structures of the human MT2 melatonin receptor reveal the basis of subtype selectivity

scientific article published on 24 April 2019

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