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List of works by Michael J Stocks

A practical method for targeted library design balancing lead-like properties with diversity

scientific article

Antagonists of the P2X(7) receptor. From lead identification to drug development.

scientific article published on May 2009

Antitumour benzothiazoles. Part 32: DNA adducts and double strand breaks correlate with activity; synthesis of 5F203 hydrogels for local delivery

scientific article published on 3 October 2015

CXCL17 is an allosteric inhibitor of CXCR4 through a mechanism of action involving glycosaminoglycans

scientific article published in 2024

Class 1 PI3K Clinical Candidates and Recent Inhibitor Design Strategies: A Medicinal Chemistry Perspective

scientific article published on 24 December 2018

Correction to Synthesis and Evaluation of the First Fluorescent Antagonists of the Human P2Y2 Receptor Based on AR-C118925.

scientific article published on 24 April 2018

Design and Elaboration of a Tractable Tricyclic Scaffold To Synthesize Druglike Inhibitors of Dipeptidyl Peptidase-4 (DPP-4), Antagonists of the C-C Chemokine Receptor Type 5 (CCR5), and Highly Potent and Selective Phosphoinositol-3 Kinase δ (PI3Kδ)

scientific article published on 27 January 2017

Design driven HtL: The discovery and synthesis of new high efficacy β₂-agonists.

scientific article published on 20 May 2011

Discovery of AZD-2098 and AZD-1678, Two Potent and Bioavailable CCR4 Receptor Antagonists.

scientific article

Discovery of AZD3199, An Inhaled Ultralong Acting β2 Receptor Agonist with Rapid Onset of Action.

scientific article published on 8 February 2014

Drug-like Antagonists of P2Y Receptors-From Lead Identification to Drug Development

scientific article

Efficient and regiospecific one-pot synthesis of substituted 1,2,4-triazoles.

scientific article published in August 2004

From UTP to AR-C118925, the discovery of a potent non nucleotide antagonist of the P2Y2 receptor.

scientific article published on 21 September 2017

In Silico and in Vitro-Guided Identification of Inhibitors of Alkylquinolone-Dependent Quorum Sensing in Pseudomonas aeruginosa

scientific article published on 28 January 2018

Ipratropium is 'luminally recycled' by an inter-play between apical uptake and efflux transporters in Calu-3 bronchial epithelial cell layers.

scientific article published on 27 August 2017

Linifanib--a multi-targeted receptor tyrosine kinase inhibitor and a low molecular weight gelator

scientific article published in April 2015

Organocatalytic enantioselective one-pot four-component ugi-type multicomponent reaction for the synthesis of epoxy-tetrahydropyrrolo[3,4-b]pyridin-5-ones

scientific article published on 28 August 2012

Preparation and structural analysis of (±)-cis-ethyl 2-sulfanylidenedecahydro-1,6-naphthyridine-6-carboxylate and (±)-trans-ethyl 2-oxooctahydro-1H-pyrrolo[3,2-c]pyridine-5-carboxylate

scientific article published on 19 November 2014

Pseudomonas aeruginosa Quorum Sensing Systems as Drug Discovery Targets: Current Position and Future Perspectives

scientific article published on 27 July 2018

Self-Assembling Benzothiazole-Based Gelators: A Mechanistic Understanding of in Vitro Bioactivation and Gelation.

scientific article published on 5 March 2018

Synthesis and Evaluation of the First Fluorescent Antagonists of the Human P2Y2 Receptor Based on AR-C118925.

scientific article published on 20 March 2018

Synthesis of New DPP-4 Inhibitors Based on a Novel Tricyclic Scaffold

scientific article published on 13 January 2015

The Discovery of MMP7 Inhibitors Exploiting a Novel Selectivity Trigger ⬇️

scientific article published on February 18, 2011

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