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List of works by Pablo Martín-Gago

A PDE6δ-KRas Inhibitor Chemotype with up to Seven H-Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2.

scientific article

A tetradecapeptide somatostatin dicarba-analog: Synthesis, structural impact and biological activity.

scientific article published on 3 December 2013

Arylfluorosulfate-Based Electrophiles for Covalent Protein Labeling: A New Addition to the Arsenal.

scientific article published on 26 October 2018

Covalent Protein Labeling at Glutamic Acids

scientific article published on 13 April 2017

Development of Pyridazinone Chemotypes Targeting the PDEδ Prenyl Binding Site

scientific article published on 3 November 2016

Fine-tuning the π-π aromatic interactions in peptides: somatostatin analogues containing mesityl alanine.

scientific article published on 9 December 2011

Identification of pyrazolopyridazinones as PDEδ inhibitors

scientific article

Insights into structure-activity relationships of somatostatin analogs containing mesitylalanine.

scientific article published on 25 November 2013

PDEδ inhibition impedes the proliferation and survival of human colorectal cancer cell lines harboring oncogenic KRas.

scientific article published on 4 December 2018

Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine

scientific article

SSTR1- and SSTR3-Selective Somatostatin Analogues

scientific article published on 21 January 2011

Stereoconvergent arylations and alkenylations of unactivated alkyl electrophiles: catalytic enantioselective synthesis of secondary sulfonamides and sulfones

scientific article

Structure-based development of PDEδ inhibitors

scientific article published on 17 November 2016

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