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List of works by Peter S Kutchukian

Correction to "Stitched α-Helical Peptides via Bis Ring-Closing Metathesis".

scientific article published on 2 July 2015

Efficient search of chemical space: navigating from fragments to structurally diverse chemotypes

scientific article

Enforced presentation of an extrahelical guanine to the lesion recognition pocket of human 8-oxoguanine glycosylase, hOGG1.

scientific article

FOG: Fragment Optimized Growth algorithm for the de novo generation of molecules occupying druglike chemical space

scientific article

Fragment library design: using cheminformatics and expert chemists to fill gaps in existing fragment libraries

scientific article published on January 2015

Inside the mind of a medicinal chemist: the role of human bias in compound prioritization during drug discovery

scientific article

Introduction of all-hydrocarbon i,i+3 staples into alpha-helices via ring-closing olefin metathesis

scientific article published on 01 July 2010

Iterative Focused Screening with Biological Fingerprints Identifies Selective Asc-1 Inhibitors Distinct from Traditional High Throughput Screening

scientific article published on 29 December 2016

Large scale meta-analysis of fragment-based screening campaigns: privileged fragments and complementary technologies

scientific article

Linking High-Throughput Screens to Identify MoAs and Novel Inhibitors of Mycobacterium tuberculosis Dihydrofolate Reductase.

scientific article published on 14 August 2017

Mapping targetable sites on human telomerase RNA pseudoknot/template domain using 2'-OMe RNA-interacting polynucleotide (RIPtide) microarrays

scientific article

Rethinking molecular similarity: comparing compounds on the basis of biological activity.

scientific article published on 31 May 2012

Stitched α-helical peptides via bis ring-closing metathesis

scientific article published on 21 August 2014

Structure of the stapled p53 peptide bound to Mdm2

scientific article