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List of works by Tristan A. Reekie

A Raney-cobalt-mediated tandem reductive cyclization route to the 1,5-methanoazocino[4,3-b]indole framework of the uleine and Strychnos alkaloids

scientific article published on 20 November 2012

A Three-Step Synthesis of Tetrasubstituted NH-Pyrroles

scientific article published on 26 April 2016

A systematic exploration of the effects of flexibility and basicity on sigma (σ) receptor binding in a series of substituted diamines.

scientific article published in October 2016

Application of a Raney-cobalt-mediated tandem reductive cyclization protocol to total syntheses of the Aspidosperma alkaloids (±)-limaspermidine and (±)-1-acetylaspidoalbidine

scientific article published on 30 October 2012

Body temperature and cardiac changes induced by peripherally administered oxytocin, vasopressin and the non-peptide oxytocin receptor agonist WAY 267,464: a biotelemetry study in rats.

scientific article

Comparative Evaluation of Three TSPO PET Radiotracers in a LPS-Induced Model of Mild Neuroinflammation in Rats

scientific article published on August 2016

Conformationally rigid derivatives of WAY-267,464: Synthesis and pharmacology at the human oxytocin and vasopressin-1a receptors.

scientific article published on 23 October 2017

Determination and reduction of translocator protein (TSPO) ligand rs6971 discrimination

scientific article published on 15 November 2016

Discovery and pharmacological evaluation of a novel series of adamantyl cyanoguanidines as P2X7 receptor antagonists.

scientific article

Flexible analogues of WAY-267,464: Synthesis and pharmacology at the human oxytocin and vasopressin 1a receptors

scientific article published on 13 December 2015

Intramolecular cycloaddition reactions of cis-1,2-dihydrocatechol derivatives incorporating C3-tethered diazoketones, nitrile oxides, and azides: stereocontrolled routes to enantiomerically pure spiro[5.5]undecanes and related systems

scientific article published on 01 July 2013

Investigation of pyrazolo-sulfonamides as putative small molecule oxytocin receptor agonists

scientific article

Investigations of amide bond variation and biaryl modification in analogues of α7 nAChR agonist SEN12333.

scientific article published on 9 July 2014

Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists

scientific article published on 31 March 2020

Pharmacological evaluation of a novel series of urea, thiourea and guanidine derivatives as P2X7 receptor antagonists

scientific article published on 04 April 2017

RANEY® cobalt--an underutilised reagent for the selective cleavage of C-X and N-O bonds

scientific article published in October 2014

Rapid Antibacterial Activity of Cannabichromenic Acid against Methicillin-Resistant Staphylococcus aureus

scientific article published on 16 August 2020

Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores

scientific article

Ring-opened aminothienopyridazines as novel tau aggregation inhibitors

scientific article published on 05 May 2017

Structural Optimization and Pharmacological Evaluation of Inhibitors Targeting Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases (DYRK) and CDC-like kinases (CLK) in Glioblastoma.

scientific article

Structure-activity relationship studies of SEN12333 analogues: determination of the optimal requirements for binding affinities at α7 nAChRs through incorporation of known structural motifs.

scientific article published on 14 March 2015

The Formation of Seven-Membered Heterocycles under Mild Pictet-Spengler Conditions: A Route to Pyrazolo[3,4]benzodiazepines

scientific article published on 13 May 2016

WAY 267,464, a non-peptide oxytocin receptor agonist, impairs social recognition memory in rats through a vasopressin 1A receptor antagonist action.

scientific article published on 13 March 2015

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