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List of works by Stamatia Vassiliou

A novel and efficient synthesis of 3,4-dihydroxyphenylacetic ester and amide derivatives/conjugates and assessment of their antioxidant activity

scientific article published on 18 June 2017

A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases

scientific article published on 22 February 2007

An effective one-pot synthesis of 3-benzylfurans and their potential utility as versatile precursors of 3,4-dibenzyltetrahydrofuran lignans. formal synthesis of (+/-)-burseran

scientific article published on 01 June 2001

Computer-aided optimization of phosphinic inhibitors of bacterial ureases.

scientific article published on August 2010

Cyclic peptides with a phosphinic bond as potent inhibitors of a zinc bacterial collagenase

scientific article published on 01 August 1994

Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues

scientific article

Mapping the pathway toward thiophosphinic pseudopeptides. Synthesis of suitably protected PG-Phe-Ψ[P(S)(OX)CH2]-Gly-OY analogues as thiophosphinyl dipeptide isosters (TDI), a comparative study for selective deprotection and further elongation

scientific article published on 02 October 2013

Novel organophosphorus scaffolds of urease inhibitors obtained by substitution of Morita-Baylis-Hillman adducts with phosphorus nucleophiles.

scientific article

Phosphinic pseudo-tripeptides as potent inhibitors of matrix metalloproteinases: a structure-activity study

scientific article published on 01 July 1999

Protection of the Hydroxyphosphinyl Function of Phosphinic Dipeptides by Adamantyl. Application to the Solid-Phase Synthesis of Phosphinic Peptides

scientific article published on 01 September 1996

RXP 407, a phosphinic peptide, is a potent inhibitor of angiotensin I converting enzyme able to differentiate between its two active sites

scientific article published on April 1999

Structure of astacin with a transition-state analogue inhibitor

scientific article

Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases.

scientific article

The M18 aspartyl aminopeptidase of the human malaria parasite Plasmodium falciparum.

scientific article published on 20 August 2007