List of works - Marc P Baggelaar

2-Arachidonoylglycerol: A signaling lipid with manifold actions in the brain

scientific article published on 08 May 2018

A natural substrate-based fluorescence assay for inhibitor screening on diacylglycerol lipase α.

scientific article published on 15 February 2015

A palmitoyl transferase chemical–genetic system to map ZDHHC-specific S-acylation

scientific article published in 2024

ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction

scientific article published on 01 October 2019

ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction

scientific article published on 07 November 2019

Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474.

scientific article

Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity.

scientific article published on 03 January 2017

Catalytic asymmetric total synthesis of (S)-(-)-zearalenone, a novel lipoxygenase inhibitor

scientific article published on 20 June 2013

Chemical Proteomic Analysis of Serine Hydrolase Activity in Niemann-Pick Type C Mouse Brain

scientific article published on 03 July 2018

Chemical Proteomics Maps Brain Region Specific Activity of Endocannabinoid Hydrolases

scientific article published on 20 January 2017

Chiral disubstituted piperidinyl ureas: a class of dual diacylglycerol lipase-α and ABHD6 inhibitors

scientific article published on 10 March 2017

Competitive ABPP of Serine Hydrolases: A Case Study on DAGL-Alpha

scientific article published in January 2017

Comprehensive Analysis of Structure-Activity Relationships of α-Ketoheterocycles as sn-1-Diacylglycerol Lipase α Inhibitors

scientific article

Development of an acid ceramidase activity-based probe

scientific article published on 01 April 2015

Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-α in brain

scientific article published on 31 October 2013

Discovery of glycine sulfonamides as dual inhibitors of sn-1-diacylglycerol lipase α and α/β-hydrolase domain 6.

scientific article published on 23 July 2014

Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons

scientific article published on July 2015

Mapping in vivo target interaction profiles of covalent inhibitors using chemical proteomics with label-free quantification

scientific article published on 22 March 2018

Novel activity-based probes for N-acylethanolamine acid amidase

scientific article published on 16 October 2017

Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition

scientific article

Recent advancements in mass spectrometry-based tools to investigate newly synthesized proteins

Site-Specific Activity-Based Protein Profiling Using Phosphonate Handles

The novel, orally available and peripherally restricted selective cannabinoid CB2 receptor agonist LEI-101 prevents cisplatin-induced nephrotoxicity

scientific article published on 23 September 2015

Total Synthesis of the Triglycosyl Phenolic Glycolipid PGL-tb1 fromMycobacterium tuberculosis

scientific article published on 19 October 2012

Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding.

scientific article

List of works by Marc P Baggelaar

2-Arachidonoylglycerol: A signaling lipid with manifold actions in the brain

A natural substrate-based fluorescence assay for inhibitor screening on diacylglycerol lipase α.

A palmitoyl transferase chemical–genetic system to map ZDHHC-specific S-acylation

ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction

ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction

Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474.

Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity.

Catalytic asymmetric total synthesis of (S)-(-)-zearalenone, a novel lipoxygenase inhibitor

Chemical Proteomic Analysis of Serine Hydrolase Activity in Niemann-Pick Type C Mouse Brain

Chemical Proteomics Maps Brain Region Specific Activity of Endocannabinoid Hydrolases

Chiral disubstituted piperidinyl ureas: a class of dual diacylglycerol lipase-α and ABHD6 inhibitors

Competitive ABPP of Serine Hydrolases: A Case Study on DAGL-Alpha

Comprehensive Analysis of Structure-Activity Relationships of α-Ketoheterocycles as sn-1-Diacylglycerol Lipase α Inhibitors

Development of an acid ceramidase activity-based probe

Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-α in brain

Discovery of glycine sulfonamides as dual inhibitors of sn-1-diacylglycerol lipase α and α/β-hydrolase domain 6.

Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons

Mapping in vivo target interaction profiles of covalent inhibitors using chemical proteomics with label-free quantification

Novel activity-based probes for N-acylethanolamine acid amidase

Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition

Recent advancements in mass spectrometry-based tools to investigate newly synthesized proteins

Site-Specific Activity-Based Protein Profiling Using Phosphonate Handles

The novel, orally available and peripherally restricted selective cannabinoid CB2 receptor agonist LEI-101 prevents cisplatin-induced nephrotoxicity

Total Synthesis of the Triglycosyl Phenolic Glycolipid PGL-tb1 fromMycobacterium tuberculosis

Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding.