List of works - Antonio J Moreno-Vargas

6-Azido hyacinthacine A2 gives a straightforward access to the first multivalent pyrrolizidine architectures

scientific article published in August 2014

Allenyl sulfones and allenyl sulfides in the synthesis of 3-pyrrolines. A novel nucleophilic [3 + 2] cycloaddition on allenyl sulfones giving rearranged cycloadducts

scientific article published on 01 November 2009

Azabicyclic vinyl sulfones for residue-specific dual protein labelling

scientific article published on 18 March 2019

Discovery of a Potent α-Galactosidase Inhibitor by in Situ Analysis of a Library of Pyrrolizidine-(Thio)urea Hybrid Molecules Generated via Click Chemistry

scientific article published on 01 August 2018

Exploiting the ring strain in bicyclo[2.2.1]heptane systems for the stereoselective preparation of highly functionalized cyclopentene, dihydrofuran, pyrroline, and pyrrolidine scaffolds

scientific article published on 08 November 2011

Exploring a Multivalent Approach to α-L-Fucosidase Inhibition

Glycosidase inhibitors as potential HIV entry inhibitors?

scientific article published in August 2004

Mechanistic Insight into the Binding of Multivalent Pyrrolidines to α-Mannosidases

scientific article published on 7 August 2017

Mixtures of Monomeric and Dimeric Surfactants: Hydrophobic Chain Length and Spacer Group Length Effects on Non Ideality

scientific article published on 03 September 2008

Monosaccharides and Analogues from Simple Achiral Unsaturated Compounds ⬇️

scientific article published on January 1, 2011

New leads for selective inhibitors of alpha-L-fucosidases. Synthesis and glycosidase inhibitory activities of [(2R,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]furan derivatives.

scientific article

Polyhydroxyamino-Piperidine-Type Iminosugars and Pipecolic Acid Analogues from aD-Mannose-Derived Aldehyde

Rapid discovery of potent α-fucosidase inhibitors by in situ screening of a library of (pyrrolidin-2-yl)triazoles

scientific article

Stable Pyrrole-Linked Bioconjugates through Tetrazine-Triggered Azanorbornadiene Fragmentation

scientific article published on 18 February 2020

Strain-promoted retro-Dieckmann-type condensation on [2.2.2]- and [2.2.1]bicyclic systems: a fragmentation reaction for the preparation of functionalized heterocycles and carbocycles

scientific article

Synthesis and anti-HIV activity of trivalent CD4-mimetic miniproteins.

scientific article published on 24 March 2007

Synthesis and conformational analysis of novel trimeric maleimide cross-linking reagents.

scientific article

Synthesis and inhibitory activities of novel C-3 substituted azafagomines: a new type of selective inhibitors of α-L-fucosidases.

scientific article

Synthesis of Pyrrolidine 3,4-Diol Derivatives with Anticancer Activity on Pancreatic Tumor Cells

Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues.

scientific article published in July 2003

Synthesis, biological evaluation, WAC and NMR studies of S-galactosides and non-carbohydrate ligands of cholera toxin based on polyhydroxyalkylfuroate moieties.

scientific article published on 21 November 2013

Three dimensional structure of a bacterial α-l-fucosidase with a 5-membered iminocyclitol inhibitor

scientific article

Total Asymmetric Synthesis of Monosaccharides and Analogues ⬇️

scientific article published on January 1, 2011

List of works by Antonio J Moreno-Vargas

6-Azido hyacinthacine A2 gives a straightforward access to the first multivalent pyrrolizidine architectures

Allenyl sulfones and allenyl sulfides in the synthesis of 3-pyrrolines. A novel nucleophilic [3 + 2] cycloaddition on allenyl sulfones giving rearranged cycloadducts

Azabicyclic vinyl sulfones for residue-specific dual protein labelling

Discovery of a Potent α-Galactosidase Inhibitor by in Situ Analysis of a Library of Pyrrolizidine-(Thio)urea Hybrid Molecules Generated via Click Chemistry

Exploiting the ring strain in bicyclo[2.2.1]heptane systems for the stereoselective preparation of highly functionalized cyclopentene, dihydrofuran, pyrroline, and pyrrolidine scaffolds

Exploring a Multivalent Approach to α-L-Fucosidase Inhibition

Glycosidase inhibitors as potential HIV entry inhibitors?

Mechanistic Insight into the Binding of Multivalent Pyrrolidines to α-Mannosidases

Mixtures of Monomeric and Dimeric Surfactants: Hydrophobic Chain Length and Spacer Group Length Effects on Non Ideality

Monosaccharides and Analogues from Simple Achiral Unsaturated Compounds ⬇️

New leads for selective inhibitors of alpha-L-fucosidases. Synthesis and glycosidase inhibitory activities of [(2R,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]furan derivatives.

Polyhydroxyamino-Piperidine-Type Iminosugars and Pipecolic Acid Analogues from aD-Mannose-Derived Aldehyde

Rapid discovery of potent α-fucosidase inhibitors by in situ screening of a library of (pyrrolidin-2-yl)triazoles

Stable Pyrrole-Linked Bioconjugates through Tetrazine-Triggered Azanorbornadiene Fragmentation

Strain-promoted retro-Dieckmann-type condensation on [2.2.2]- and [2.2.1]bicyclic systems: a fragmentation reaction for the preparation of functionalized heterocycles and carbocycles

Synthesis and anti-HIV activity of trivalent CD4-mimetic miniproteins.

Synthesis and conformational analysis of novel trimeric maleimide cross-linking reagents.

Synthesis and inhibitory activities of novel C-3 substituted azafagomines: a new type of selective inhibitors of α-L-fucosidases.

Synthesis of Pyrrolidine 3,4-Diol Derivatives with Anticancer Activity on Pancreatic Tumor Cells

Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues.

Synthesis, biological evaluation, WAC and NMR studies of S-galactosides and non-carbohydrate ligands of cholera toxin based on polyhydroxyalkylfuroate moieties.

Three dimensional structure of a bacterial α-l-fucosidase with a 5-membered iminocyclitol inhibitor

Total Asymmetric Synthesis of Monosaccharides and Analogues ⬇️