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List of works by Terry W. Moore

A "cross-stitched" peptide with improved helicity and proteolytic stability

scientific article published on 01 May 2018

A Cell-Permeable Stapled Peptide Inhibitor of the Estrogen Receptor/Coactivator Interaction.

scientific article

A set of time-resolved fluorescence resonance energy transfer assays for the discovery of inhibitors of estrogen receptor-coactivator binding

scientific article

Antiviral atropisomers: conformational energy surfaces by NMR for host-directed myxovirus blockers

scientific article

Asymmetric synthesis of host-directed inhibitors of myxoviruses.

scientific article published on 30 January 2013

Curcumin analogue UBS109 prevents bone loss in breast cancer bone metastasis mouse model: involvement in osteoblastogenesis and osteoclastogenesis

scientific article published on 11 April 2014

Discovering Small‐Molecule Estrogen Receptor α/Coactivator Binding Inhibitors: High‐Throughput Screening, Ligand Development, and Models for Enhanced Potency ⬇️

scientific article published on April 4, 2011

Estrogen receptor alpha/co-activator interaction assay: TR-FRET

scientific article published on January 2015

Inhibition of the NF-κB signaling pathway by the curcumin analog, 3,5-Bis(2-pyridinylmethylidene)-4-piperidone (EF31): anti-inflammatory and anti-cancer properties.

scientific article

Isoquinoline Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-Derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability

scientific article published on 14 November 2019

Liver S9 Fraction-Derived Metabolites of Curcumin Analogue UBS109.

scientific article

Minireview: Not picking pockets: nuclear receptor alternate-site modulators (NRAMs)

scientific article

N-Substituted Pyrrole-Based Heterocycles as Broad-Spectrum Filoviral Entry Inhibitors

scholarly article published on 6 August 2024

Non-electrophilic modulators of the canonical Keap1/Nrf2 pathway

scientific article

Novel curcumin analogue UBS109 potently stimulates osteoblastogenesis and suppresses osteoclastogenesis: involvement in Smad activation and NF-κB inhibition.

scientific article

Probing the Topological Tolerance of Multimeric Protein Interactions: Evaluation of an Estrogen/Synthetic Ligand for FK506 Binding Protein Conjugate ⬇️

scientific article published on October 20, 2010

Probing the structural requirements of non-electrophilic naphthalene-based Nrf2 activators.

scientific article

Recent structural advances in constrained helical peptides

scientific article published on 11 October 2018

Replacement of a Naphthalene Scaffold in Kelch-like ECH-Associated Protein 1 (KEAP1)/Nuclear Factor (Erythroid-derived 2)-like 2 (NRF2) Inhibitors

scientific article published on 31 August 2018

SAR Study on Estrogen Receptor α/β Activity of (Iso)flavonoids: Importance of Prenylation, C-Ring (Un)Saturation, and Hydroxyl Substituents

scientific article published on 18 September 2020

Selective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast Cancer

scientific article published on 17 December 2015

Stapled Peptides with γ-Methylated Hydrocarbon Chains for the Estrogen Receptor/Coactivator Interaction

scientific article published on March 2016

Steroid receptor/coactivator binding inhibitors: An update

scientific article published on 01 June 2019

Synthetic curcumin analog EF31 inhibits the growth of head and neck squamous cell carcinoma xenografts

scientific article published on 25 April 2012

Synthetic curcumin analog UBS109 inhibits the growth of head and neck squamous cell carcinoma xenografts.

scientific article published on May 2014

Time-Gated Detection of Cystathionine γ-Lyase Activity and Inhibition with a Selective, Luminogenic Hydrogen Sulfide Sensor.

scientific article published on 12 October 2016

Time-Gated Luminescence Detection of Enzymatically Produced Hydrogen Sulfide: Design, Synthesis, and Application of a Lanthanide-Based Probe.

scientific article published on 27 December 2017

Using Tumor Explants for Imaging Mass Spectrometry Visualization of Unlabeled Peptides and Small Molecules

scientific article published on 17 May 2018

Visualizing cancer and response to therapy in vivo using Cy5.5-labeled factor VIIa and anti-tissue factor antibody

scientific article

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