Search filters

List of works by Élie Besserer-Offroy

Angiotensin II cyclic analogs as tools to investigate AT1R biased signaling mechanisms

scientific article published on 20 April 2018

Apelin-13 Regulates Vasopressin-Induced Aquaporin-2 Expression and Trafficking in Kidney Collecting Duct Cells

scientific article published on 01 January 2019

C-Terminal modifications of apelin-13 significantly change ligand binding, receptor signaling, and hypotensive action

scientific article published on 24 February 2015

Cell-penetrating pepducins targeting the neurotensin receptor type 1 relieve pain

scientific article published on 06 March 2020

Conjugation of a brain-penetrant peptide with neurotensin provides antinociceptive properties

scientific article

Data set describing the in vitro biological activity of JMV2009, a novel silylated neurotensin(8-13) analog

scientific article published on 20 June 2020

Design, synthesis, and biological evaluation of CXCR4 ligands

scientific article published on 18 October 2016

Discovery and Structure-Activity Relationship of a Bioactive Fragment of ELABELA that Modulates Vascular and Cardiac Functions.

scientific article

Elucidation of the structure-activity relationships of apelin: influence of unnatural amino acids on binding, signaling, and plasma stability

scientific article published on 13 December 2011

Identification of 2-({[1-(4-Fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)tricyclo[3.3.1.13,7]decane-2-carboxylic Acid (NTRC-844) as a Selective Antagonist for the Rat Neurotensin Receptor Type 2.

scientific article published on 30 June 2016

In Search of the Optimal Macrocyclization Site for Neurotensin

scientific article published on 29 January 2018

Label-free cell signaling pathway deconvolution of angiotensin type 1 receptor reveals time-resolved G-protein activity and distinct AngII and AngIIIIV responses

scientific article published on 28 June 2018

Pain relief devoid of opioid side effects following central action of a silylated neurotensin analog

scientific article published on 10 June 2020

Stereoselective Synthesis of β-(5-Arylthiazolyl) α-Amino Acids and Use in Neurotensin Analogues

Structural Optimization and Characterization of Potent Analgesic Macrocyclic Analogues of Neurotensin (8-13)

scientific article published on 13 August 2018

Structural basis of ligand selectivity and disease mutations in cysteinyl leukotriene receptors

scientific article published on 06 December 2019

Structural insights on ligand recognition at the human leukotriene B4 receptor 1

scientific article published on 20 May 2021

Structure-Activity Relationship and Signaling of New Chimeric CXCR4 Agonists

scientific article published on 19 July 2016

Structure-Based Virtual Screening of Ultra-Large Library Yields Potent Antagonists for a Lipid GPCR

scientific article published on 03 December 2020

Structure-activity relationship of novel macrocyclic biased apelin receptor agonists.

scientific article

Structure-based mechanism of cysteinyl leukotriene receptor inhibition by antiasthmatic drugs

scientific article published on 09 October 2019

Synthesis and Characterization in Vitro and in Vivo of (l)-(Trimethylsilyl)alanine Containing Neurotensin Analogues.

scientific article published on 8 September 2015

The hypotensive effect of activated apelin receptor is correlated with β-arrestin recruitment.

scientific article

The signaling signature of the neurotensin type 1 receptor with endogenous ligands

scientific article published on 21 March 2017

Use of Molecular Modeling to Design Selective NTS2 Neurotensin Analogues.

scientific article published on 3 April 2017

Paulina is supported by:

About Paulina

Help