List of works - Robert A. Batey

1H-Imidazol-1-yl 1,2,3,4-tetrahydroisoquinolin-2-yl ketone.

scientific article published on 18 September 2004

A Lanthanide(III) Triflate Mediated Macrolactonization/Solid-Phase Synthesis Approach for Depsipeptide Synthesis

scientific article published on 13 April 2015

A hetero Diels-Alder approach to the synthesis of chromans (3,4-dihydrobenzopyrans) using oxonium ion chemistry: the oxa-Povarov reaction

scientific article published on 31 January 2013

A mild protocol for allylation and highly diastereoselective syn or anti crotylation of aldehydes in biphasic and aqueous media utilizing potassium allyl- and crotyltrifluoroborates

scientific article published on 01 October 2002

A novel diquinolonium displays preclinical anti-cancer activity and induces caspase-independent cell death

scientific article

A novel inhibitor of glucose uptake sensitizes cells to FAS-induced cell death

scientific article

A room-temperature protocol for the rhodium(I)-catalyzed addition of arylboron compounds to sulfinimines

scientific article published on 01 April 2005

A short total synthesis of the marine sponge pyrrole-2-aminoimidazole alkaloid (±)-agelastatin A.

scientific article

A small-molecule inhibitor of D-cyclin transactivation displays preclinical efficacy in myeloma and leukemia via phosphoinositide 3-kinase pathway.

scientific article published on 6 December 2010

Activators of cylindrical proteases as antimicrobials: identification and development of small molecule activators of ClpP protease

scientific article published in September 2011

Acyldepsipeptide Analogs Dysregulate Human Mitochondrial ClpP Protease Activity and Cause Apoptotic Cell Death

scientific article published on 28 June 2018

Allylation and crotylation of ketones and aldehydes using potassium organotrifluoroborate salts under Lewis acid and montmorillonite K10 catalyzed conditions

scientific article published on 01 June 2009

Allylation of Imines and Their Derivatives with Organoboron Reagents: Stereocontrolled Synthesis of Homoallylic Amines

Amidation reactions from the direct coupling of metal carboxylate salts with amines

scientific article published on 13 January 2014

An Alumino-Mannich Reaction of Organoaluminum Reagents, Silylated Amines, and Aldehydes

scientific article published on 26 March 2018

An Approach to the 9-Oxo-10-oxabicyclo[5.3.0]dec-2-ene Core of the Guaianolide and Pseudoguaianolide Sesquiterpenes via a Domino Electrocyclic Ring Opening / Carboxylic Acid Trapping of a gem-Dibromocyclopropane

article

An organotrifluoroborate-based convergent total synthesis of the potent cancer cell growth inhibitory depsipeptides kitastatin and respirantin

scientific article published on 14 April 2014

Carbamoyl-SubstitutedN-Heterocyclic Carbene Complexes of Palladium(II): Application to Sonogashira Cross-Coupling Reactions

article

Chelation of intracellular iron with the antifungal agent ciclopirox olamine induces cell death in leukemia and myeloma cells.

scientific article published on 9 July 2009

Copper(II)-catalyzed ether synthesis from aliphatic alcohols and potassium organotrifluoroborate salts.

scientific article

Copper- and palladium-catalyzed intramolecular aryl guanidinylation: an efficient method for the synthesis of 2-aminobenzimidazoles

scientific article published on 01 January 2003

Copper-catalyzed domino annulation approaches to the synthesis of benzoxazoles under microwave-accelerated and conventional thermal conditions

scientific article

Copper-catalyzed nondecarboxylative cross coupling of alkenyltrifluoroborate salts with carboxylic acids or carboxylates: synthesis of enol esters

scientific article published on 04 June 2013

DABO Boronate Promoted Conjugate Allylation of α,β-Unsaturated Aldehydes Using Copper(II) Catalysis

scientific article published on 14 July 2016

Development and Characterization of Potent Cyclic Acyldepsipeptide Analogues with Increased Antimicrobial Activity

scientific article

Effect of noncompetitive proteasome inhibition on bortezomib resistance

scientific article

Enamide synthesis by copper-catalyzed cross-coupling of amides and potassium alkenyltrifluoroborate salts

scientific article published on 01 January 2008

Enantioselective palladium(II)-catalyzed formal [3,3]-sigmatropic rearrangement of 2-allyloxypyridines and related heterocycles.

scientific article published in January 2010

Functional characterization of a PROTAC directed against BRAF mutant V600E

scientific article published on 10 August 2020

Hetero Diels-Alder reactions of nitrosoamidines: an efficient method for the synthesis of functionalized guanidines

scientific article published on 01 March 2004

Heterocycle formation via palladium-catalyzed intramolecular oxidative C-H bond functionalization: an efficient strategy for the synthesis of 2-aminobenzothiazoles

scientific article published on 01 July 2009

Indium-promoted chemo- and diastereoselective allylation of α,β-epoxy ketones with potassium allyltrifluoroborate

scientific article published on 11 November 2010

Intramolecular hetero Diels-Alder (Povarov) approach to the synthesis of the alkaloids luotonin A and camptothecin

scientific article published on 01 December 2004

Lanthanide(III)-Catalyzed Synthesis of trans-Diaminocyclopentenones from Substituted Furfurals and Secondary Amines via a Domino Ring-Opening/4π-Electrocyclization Pathway

article

Ligand- and Base-Free Copper(II)-Catalyzed C−N Bond Formation: Cross-Coupling Reactions of Organoboron Compounds with Aliphatic Amines and Anilines ⬇️

scientific article published on November 13, 2003

Mild Double Allylboration Reactions of Nitriles and Acid Anhydrides Using Potassium Allyltrifluoroborate

scientific article published on 15 January 2013

Mild lanthanide(III) catalyzed formation of 4,5-diaminocyclopent-2-enones from 2-furaldehyde and secondary amines: a domino condensation/ring-opening/electrocyclization process

scientific article published on 09 July 2007

Organoboron-based allylation approach to the total synthesis of the medium-ring dilactone (+)-antimycin A(1b)

scientific article published on 25 July 2014

Palladium-catalyzed [3,3] sigmatropic rearrangement of (allyloxy)iminodiazaphospholidines: allylic transposition of C--O and C--N functionality

scientific article published on 01 March 2004

Palladium-catalyzed allylic transposition of (allyloxy) iminodiazaphospholidines: a formal [3,3]-aza-phospha-oxa-Cope sigmatropic rearrangement for the stereoselective synthesis of allylic amines

scientific article published in October 2005

Parallel synthesis of a library of benzoxazoles and benzothiazoles using ligand-accelerated copper-catalyzed cyclizations of ortho-halobenzanilides

scientific article published in March 2006

Peptide Heterocycle Conjugates: A Diverted Edman Degradation Protocol for the Synthesis of N-Terminal 2-Iminohydantoins

scientific article published in April 2003

Peptide-heterocycle hybrid molecules: solid-phase synthesis of a 400-member library of N-terminal 2-iminohydantoin peptides

scientific article

Peptide-heterocycle hybrid molecules: solid-phase-supported synthesis of substituted N-terminal 5-aminotetrazole peptides via electrocyclization of peptidic imidoylazides

scientific article

Phase-transfer-catalyzed alkylation of guanidines by alkyl halides under biphasic conditions: a convenient protocol for the synthesis of highly functionalized guanidines.

scientific article published in March 2003

RNA-Puzzles Round III: 3D RNA structure prediction of five riboswitches and one ribozyme

scientific article

Regio- and stereoselective allylation and crotylation of indoles at C2 through the use of potassium organotrifluoroborate salts

scientific article published on 06 December 2012

Sequential O-Arylation/Lanthanide(III)-Catalyzed [3,3]-Sigmatropic Rearrangement of Bromo-Substituted Allylic Alcohols

Stereocontrolled Microwave-Assisted Domino [3,3]-Sigmatropic Reactions: A Winstein-Overman Rearrangement for the Formation of Differentiated Contiguous C-N Bonds

scientific article published on 30 March 2020

Stereocontrolled Synthesis of Contiguous C(sp3)−C(aryl) Bonds by Lanthanide(III)-Catalyzed Domino Aryl-Claisen [3,3]-Sigmatropic Rearrangements

scientific article published on 01 October 2010

Structure-based de novo design of ligands using a three-dimensional model of the insulin receptor.

scientific article published on March 2004

Synthesis and reactivity of N-alkyl carbamoylimidazoles: development of N-methyl carbamoylimidazole as a methyl isocyanate equivalent

scientific article published on 29 October 2012

Terminal alkyne addition to diazodicarboxylates: synthesis of hydrazide linked alkynes (ynehydrazides)

scientific article published on 04 January 2012

The antiparasitic agent ivermectin induces chloride-dependent membrane hyperpolarization and cell death in leukemia cells

scientific article published on 19 July 2010

The role of ClpP protease in bacterial pathogenesis and human diseases.

scientific article

The ubiquitin-activating enzyme E1 as a therapeutic target for the treatment of leukemia and multiple myeloma

scientific article

Total Synthesis of (+)-Prunustatin A: Utility of Organotrifluoroborate-Mediated Prenylation and Shiina MNBA Esterification and Macrolactonization To Avoid a Competing Thorpe-Ingold Effect Accelerated Transesterification

scientific article published on 30 August 2018

Total synthesis and antibacterial testing of the A54556 cyclic acyldepsipeptides isolated from Streptomyces hawaiiensis.

scientific article

Total synthesis of the alkaloids martinelline and martinellic acid via a hetero Diels-Alder multicomponent coupling reaction

scientific article published on 01 August 2002

Total synthesis of the cytotoxic enehydrazide natural products hydrazidomycins A and B by a carbazate addition/Peterson olefination approach

scientific article published on 04 June 2013

List of works by Robert A. Batey

1H-Imidazol-1-yl 1,2,3,4-tetrahydroisoquinolin-2-yl ketone.

A Lanthanide(III) Triflate Mediated Macrolactonization/Solid-Phase Synthesis Approach for Depsipeptide Synthesis

A hetero Diels-Alder approach to the synthesis of chromans (3,4-dihydrobenzopyrans) using oxonium ion chemistry: the oxa-Povarov reaction

A mild protocol for allylation and highly diastereoselective syn or anti crotylation of aldehydes in biphasic and aqueous media utilizing potassium allyl- and crotyltrifluoroborates

A novel diquinolonium displays preclinical anti-cancer activity and induces caspase-independent cell death

A novel inhibitor of glucose uptake sensitizes cells to FAS-induced cell death

A room-temperature protocol for the rhodium(I)-catalyzed addition of arylboron compounds to sulfinimines

A short total synthesis of the marine sponge pyrrole-2-aminoimidazole alkaloid (±)-agelastatin A.

A small-molecule inhibitor of D-cyclin transactivation displays preclinical efficacy in myeloma and leukemia via phosphoinositide 3-kinase pathway.

Activators of cylindrical proteases as antimicrobials: identification and development of small molecule activators of ClpP protease

Acyldepsipeptide Analogs Dysregulate Human Mitochondrial ClpP Protease Activity and Cause Apoptotic Cell Death

Allylation and crotylation of ketones and aldehydes using potassium organotrifluoroborate salts under Lewis acid and montmorillonite K10 catalyzed conditions

Allylation of Imines and Their Derivatives with Organoboron Reagents: Stereocontrolled Synthesis of Homoallylic Amines

Amidation reactions from the direct coupling of metal carboxylate salts with amines

An Alumino-Mannich Reaction of Organoaluminum Reagents, Silylated Amines, and Aldehydes

An Approach to the 9-Oxo-10-oxabicyclo[5.3.0]dec-2-ene Core of the Guaianolide and Pseudoguaianolide Sesquiterpenes via a Domino Electrocyclic Ring Opening / Carboxylic Acid Trapping of a gem-Dibromocyclopropane

An organotrifluoroborate-based convergent total synthesis of the potent cancer cell growth inhibitory depsipeptides kitastatin and respirantin

Carbamoyl-SubstitutedN-Heterocyclic Carbene Complexes of Palladium(II): Application to Sonogashira Cross-Coupling Reactions

Chelation of intracellular iron with the antifungal agent ciclopirox olamine induces cell death in leukemia and myeloma cells.

Copper(II)-catalyzed ether synthesis from aliphatic alcohols and potassium organotrifluoroborate salts.

Copper- and palladium-catalyzed intramolecular aryl guanidinylation: an efficient method for the synthesis of 2-aminobenzimidazoles

Copper-catalyzed domino annulation approaches to the synthesis of benzoxazoles under microwave-accelerated and conventional thermal conditions

Copper-catalyzed nondecarboxylative cross coupling of alkenyltrifluoroborate salts with carboxylic acids or carboxylates: synthesis of enol esters

DABO Boronate Promoted Conjugate Allylation of α,β-Unsaturated Aldehydes Using Copper(II) Catalysis

Development and Characterization of Potent Cyclic Acyldepsipeptide Analogues with Increased Antimicrobial Activity

Effect of noncompetitive proteasome inhibition on bortezomib resistance

Enamide synthesis by copper-catalyzed cross-coupling of amides and potassium alkenyltrifluoroborate salts

Enantioselective palladium(II)-catalyzed formal [3,3]-sigmatropic rearrangement of 2-allyloxypyridines and related heterocycles.

Functional characterization of a PROTAC directed against BRAF mutant V600E

Hetero Diels-Alder reactions of nitrosoamidines: an efficient method for the synthesis of functionalized guanidines

Heterocycle formation via palladium-catalyzed intramolecular oxidative C-H bond functionalization: an efficient strategy for the synthesis of 2-aminobenzothiazoles

Indium-promoted chemo- and diastereoselective allylation of α,β-epoxy ketones with potassium allyltrifluoroborate

Intramolecular hetero Diels-Alder (Povarov) approach to the synthesis of the alkaloids luotonin A and camptothecin

Lanthanide(III)-Catalyzed Synthesis of trans-Diaminocyclopentenones from Substituted Furfurals and Secondary Amines via a Domino Ring-Opening/4π-Electrocyclization Pathway

Ligand- and Base-Free Copper(II)-Catalyzed C−N Bond Formation: Cross-Coupling Reactions of Organoboron Compounds with Aliphatic Amines and Anilines ⬇️

Mild Double Allylboration Reactions of Nitriles and Acid Anhydrides Using Potassium Allyltrifluoroborate

Mild lanthanide(III) catalyzed formation of 4,5-diaminocyclopent-2-enones from 2-furaldehyde and secondary amines: a domino condensation/ring-opening/electrocyclization process

Organoboron-based allylation approach to the total synthesis of the medium-ring dilactone (+)-antimycin A(1b)

Palladium-catalyzed [3,3] sigmatropic rearrangement of (allyloxy)iminodiazaphospholidines: allylic transposition of C--O and C--N functionality

Palladium-catalyzed allylic transposition of (allyloxy) iminodiazaphospholidines: a formal [3,3]-aza-phospha-oxa-Cope sigmatropic rearrangement for the stereoselective synthesis of allylic amines

Parallel synthesis of a library of benzoxazoles and benzothiazoles using ligand-accelerated copper-catalyzed cyclizations of ortho-halobenzanilides

Peptide Heterocycle Conjugates: A Diverted Edman Degradation Protocol for the Synthesis of N-Terminal 2-Iminohydantoins

Peptide-heterocycle hybrid molecules: solid-phase synthesis of a 400-member library of N-terminal 2-iminohydantoin peptides

Peptide-heterocycle hybrid molecules: solid-phase-supported synthesis of substituted N-terminal 5-aminotetrazole peptides via electrocyclization of peptidic imidoylazides

Phase-transfer-catalyzed alkylation of guanidines by alkyl halides under biphasic conditions: a convenient protocol for the synthesis of highly functionalized guanidines.

RNA-Puzzles Round III: 3D RNA structure prediction of five riboswitches and one ribozyme

Regio- and stereoselective allylation and crotylation of indoles at C2 through the use of potassium organotrifluoroborate salts

Sequential O-Arylation/Lanthanide(III)-Catalyzed [3,3]-Sigmatropic Rearrangement of Bromo-Substituted Allylic Alcohols

Stereocontrolled Microwave-Assisted Domino [3,3]-Sigmatropic Reactions: A Winstein-Overman Rearrangement for the Formation of Differentiated Contiguous C-N Bonds

Stereocontrolled Synthesis of Contiguous C(sp3)−C(aryl) Bonds by Lanthanide(III)-Catalyzed Domino Aryl-Claisen [3,3]-Sigmatropic Rearrangements

Structure-based de novo design of ligands using a three-dimensional model of the insulin receptor.

Synthesis and reactivity of N-alkyl carbamoylimidazoles: development of N-methyl carbamoylimidazole as a methyl isocyanate equivalent

Terminal alkyne addition to diazodicarboxylates: synthesis of hydrazide linked alkynes (ynehydrazides)

The antiparasitic agent ivermectin induces chloride-dependent membrane hyperpolarization and cell death in leukemia cells

The role of ClpP protease in bacterial pathogenesis and human diseases.

The ubiquitin-activating enzyme E1 as a therapeutic target for the treatment of leukemia and multiple myeloma

Total Synthesis of (+)-Prunustatin A: Utility of Organotrifluoroborate-Mediated Prenylation and Shiina MNBA Esterification and Macrolactonization To Avoid a Competing Thorpe-Ingold Effect Accelerated Transesterification

Total synthesis and antibacterial testing of the A54556 cyclic acyldepsipeptides isolated from Streptomyces hawaiiensis.

Total synthesis of the alkaloids martinelline and martinellic acid via a hetero Diels-Alder multicomponent coupling reaction

Total synthesis of the cytotoxic enehydrazide natural products hydrazidomycins A and B by a carbazate addition/Peterson olefination approach