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List of works by Ole A. Andersen

2.0A resolution crystal structures of the ternary complexes of human phenylalanine hydroxylase catalytic domain with tetrahydrobiopterin and 3-(2-thienyl)-L-alanine or L-norleucine...

scientific article

An efficient synthesis of argifin: a natural product chitinase inhibitor with chemotherapeutic potential.

scientific article

Analyzing Airway Inflammation with Chemical Biology: Dissection of Acidic Mammalian Chitinase Function with a Selective Drug-like Inhibitor

scientific article

Bisdionin C-a rationally designed, submicromolar inhibitor of family 18 chitinases

scientific article

Cross-linking of protein crystals as an aid in the generation of binary protein-ligand crystal complexes, exemplified by the human PDE10a-papaverine structure

scientific article

Crystal structure of alkaline phosphatase from the Antarctic bacterium TAB5

scientific article

Crystal structure of the ternary complex of the catalytic domain of human phenylalanine hydroxylase with tetrahydrobiopterin and 3-(2-thienyl)-L-alanine, and its implications for the mechanism of catalysis and substrate activation

scientific article

Deamidation of labile asparagine residues in the autoregulatory sequence of human phenylalanine hydroxylase.

scientific article

Discovery and structure-activity relationship of potent and selective covalent inhibitors of transglutaminase 2 for Huntington's disease.

scientific article

First Synthesis of Argadin: A Nanomolar Inhibitor of Family-18 Chitinases

First Synthesis of Argadin: A Nanomolar Inhibitor of Family-18 Chitinases

Methylxanthine drugs are chitinase inhibitors: investigation of inhibition and binding modes.

scientific article published in September 2005

Natural product family 18 chitinase inhibitors

scientific article

SPPS of the natural product chitinase inhibitor argifin: library generation and biological evaluation

scientific article

Screening-based discovery and structural dissection of a novel family 18 chitinase inhibitor

scientific article published on 14 July 2006

Solid-phase synthesis of cyclic peptide chitinase inhibitors: SAR of the argifin scaffold.

scientific article published on 13 November 2008

Structural basis for enzymatic excision of N1-methyladenine and N3-methylcytosine from DNA

scientific article

Structure-Based Dissection of the Natural Product Cyclopentapeptide Chitinase Inhibitor Argifin

scientific article

Studies on the regulatory properties of the pterin cofactor and dopamine bound at the active site of human phenylalanine hydroxylase.

scientific article published in March 2003

Synthesis and structure-based dissection of cyclic peptide chitinase inhibitors: new leads for antifungal and anti-inflammatory drugs

The multiple roles of computational chemistry in fragment-based drug design

scientific article published on 17 June 2009