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List of works by Gino Giannaccini

1,2,3-Triazolo[1,5-a][1,4]- and 1,2,3-triazolo[1,5-a]-[1,5]benzodiazepine derivatives: synthesis and benzodiazepine receptor binding

scientific article published in April 1998

1,2,3-Triazolo[1,5-a]quinoxalines: synthesis and binding to benzodiazepine and adenosine receptors

1,2,3-Triazolo[4,5-d]pyridazines

1,8-Naphthyridin-4-one derivatives as new ligands of A2A adenosine receptors

scientific article published in October 2005

1-Aminocyclopentane-1,2,4-tricarboxylic acids screening on glutamatergic and serotonergic systems

scientific article published on 12 September 2007

A 3H-flunitrazepam binding inhibitor is present in psychiatric patients' sera

scientific article

A link between oxytocin and serotonin in humans: Supporting evidence from peripheral markers

article

A multidisciplinary approach to study the effects of balneotherapy and mud-bath therapy treatments on fibromyalgia

scientific article

A novel class of highly potent and selective A1 adenosine antagonists: structure-affinity profile of a series of 1,8-naphthyridine derivatives.

scientific article published in July 2000

A proteomic approach to study parathyroid glands

scientific article published on 21 December 2010

A proteomic profile of washing fluid from the colorectal tract to search for potential biomarkers of colon cancer

article

A relationship between oxytocin and anxiety of romantic attachment

scientific article

ATP, calcium and magnesium levels in platelets of patients with primary fibromyalgia

scientific article published on 2 July 2008

Absence of NK 1 Receptors in Human Blood Lymphocytes and Granulocytes

Adenosine receptors: synthesis, structure-activity relationships and biological activity of new 6-amino purine derivatives

Alpha(1)-adrenoceptor antagonists. 4. Pharmacophore-based design, synthesis, and biological evaluation of new imidazo-, benzimidazo-, and indoloarylpiperazine derivatives

scientific article published in August 2002

Alpha1-adrenoceptor antagonists. 6. Structural optimization of pyridazinone-arylpiperazines. Study of the influence on affinity and selectivity of cyclic substituents at the pyridazinone ring and alkoxy groups at the arylpiperazine moiety

scientific article published in July 2003

Alteration of serotonin transporter density and activity in fibromyalgia

scientific article published on January 2006

Alterations of the dopamine transporter in resting lymphocytes of patients with different psychotic disorders

scientific article published on 11 November 2009

Altered amino acid homeostasis in subjects affected by fibromyalgia

scientific article published on 10 March 2009

Apparent absence of aging and gender effects on serotonin 1A receptors in human neocortex and hippocampus

scientific article published in May 1997

Autoradiographic distribution of neuropeptide Y binding sites in the brain of the carp Cyprinus carpio L. (Cyprinidae, Teleostei).

scientific article published in April 2003

Autoradiographic distribution of peripheral benzodiazepine receptors in the retina of the albino rabbit, Lepus cunicula

scientific article published on 01 February 2000

Autoradiographic localization and binding study of benzodiazepines receptor sites in carp brain (Cyprinus carpio L.).

scientific article

Barbiturate enhancement of [3H]flunitrazepam binding to purified benzodiazepine/gaba receptor from rat brain

scientific article published on 01 January 1987

Benzodiazepine agonists reverse the effects of noise exposure on central benzodiazepine receptors and cardiac responsiveness.

scientific article published in January 1995

Binding of 3H-WIN-35,428 and 125I-RTI-121 to human platelet membranes

scientific article

Binding of [3H] muscimol to the retina of rabbit and turtle

scientific article published on 01 January 1989

Binding of beta 1-adrenoceptor antagonist [3H]CGP 26505 in rat cerebral cortex and sinus atrial node

scientific article published in October 1996

Binding of the benzodiazepine ligand [3H]-RO 15-1788 to membrane preparations of the rabbit and turtle retina

scientific article published on 01 February 1992

Binding of the benzodiazepine ligand [3H]-Ro 15-1788 to brain membrane of the saltwater fish Mullus surmuletus

scientific article

Changes in peripheral benzodiazepine receptors in patients with bipolar disorder

scientific article published on June 2005

Characterization of adenosine receptors in Mullus surmuletus

scientific article published in 1996

Characterization of sulfonylurea receptors in isolated human pancreatic islets

scientific article published on 01 November 1998

Chiral 1,4-benzodiazepin-2-ones: relationship between stereochemistry and pharmacological activity.

scientific article

Clozapine effects on adenylyl cyclase activity and serotonin type 1A receptors in human brain post-mortem

scientific article

Clozapine, norclozapine plasma levels, their sum and ratio in 50 psychotic patients: influence of patient-related variables

scientific article

Common alterations in the serotonin transporter in platelets and lymphocytes of psychotic patients

scientific article published in January 2006

Comparative proteomic analysis of malignant pleural mesothelioma evidences an altered expression of nuclear lamin and filament-related proteins

scientific article published on 12 February 2014

Conformationally restrained analogues of sympathomimetic catecholamines. Synthesis and adrenergic activity of 5,6- and 6,7-dihydroxy-3,4-dihydrospiro[naphthalen-1(2H)-2',5'-morpholines].

scientific article published in January 2002

Conformationally restrained β-blocking oxime ethers: synthesis and β-adrenergic properties of diastereoisomeric anti and syn 2-(5′-isoxazolidinyl)-ethanolamines

Correlation between platelet alpha(2)-adrenoreceptors and symptom severity in major depression.

scientific article

Correlation between the sites labelled by [3H]-8 hydroxy-2-(di-N-propylamino)tetralin and [3H]-imipramine in human platelets

Decreased density of peripheral benzodiazepine receptors in psychiatric patients after a suicide attempt

scientific article published on 12 July 2005

Decreased density of the platelet serotonin transporter in pathological gamblers

scientific article published on 2 May 2008

Decreased elastase activity in circulating granulocytes of systemic sclerosis patients: a possible pathogenetic role

scientific article published on 01 November 2005

Decreased inhibitory activity of PKC in OCD patients after six months of treatment

scientific article published in October 2002

Decreased lymphocyte 3H-paroxetine binding in obsessive-compulsive disorder

scientific article published in January 2003

Decreased lymphocyte dopamine transporter in romantic lovers

scientific article published on 29 December 2016

Design, synthesis, and alpha(1)-adrenoceptor binding properties of new arylpiperazine derivatives bearing a flavone nucleus as the terminal heterocyclic molecular portion

scientific article published in March 2004

Detection of potential markers of primary fibromyalgia syndrome in human saliva

scientific article published on 14 September 2009

Discovery of N-hydroxyindole-based inhibitors of human lactate dehydrogenase isoform A (LDH-A) as starvation agents against cancer cells.

scientific article published on 18 February 2011

Distribution of serotonin receptor of type 6 (5-HT₆) in human brain post-mortem. A pharmacology, autoradiography and immunohistochemistry study.

scientific article published on 26 January 2012

Effect of aging and sex on the [3H]-paroxetine binding to human platelets.

scientific article published in July 1998

Effect of noise exposure on rat cardiac peripheral benzodiazepine receptors.

scientific article

Effect of valproate and antidepressant drugs on clozapine metabolism in patients with psychotic mood disorders

scientific article published on 29 March 2018

Effects of chestnut hydrolysable tannin enrichment in the artificial diet of forager bees, <i>Apis mellifera</i>

scientific article published on 26 August 2021

Effects of postmortem delay on serotonin and (+)8-OH-DPAT-mediated inhibition of adenylyl cyclase activity in rat and human brain tissues.

scientific article published in January 1999

Ethyl 8-fluoro-6-(3-nitrophenyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate as novel, highly potent, and safe antianxiety agent

scientific article published on 19 July 2008

Evaluation of formalin-fixed paraffin-embedded tissues in the proteomic analysis of parathyroid glands

scientific article published on 8 June 2011

Fine-needle aspiration of thyroid nodules: proteomic analysis to identify cancer biomarkers

scientific article

First evidence of TRPV5 and TRPV6 channels in human parathyroid glands: possible involvement in neoplastic transformation.

scientific article published on 28 August 2014

Gender and age-related variation in adenylyl cyclase activity in the human prefrontal cortex, hippocampus and dorsal raphe nuclei

scientific article published on 01 January 2000

HPLC resolution of C5 chiral 4,5-dihydro-1,4-benzodiazepines: stereochemical characterization and enantioselective GABAA receptor binding

scientific article published on 01 March 1997

Human serotonin transporter expression during megakaryocytic differentiation of MEG-01 cells

scientific article

Immunohistochemical distribution of neuropeptide Y in the mesencephalon and rhombencephalon of carp, Cyprinus carpio L. (Cyprinidae: Teleostei)

scientific article published on 01 June 2004

In vitro effects of lead ions on peripheral benzodiazepine receptors and adenylyl cyclase activity in the mantle of Mytilus galloprovincialis.

scientific article published on February 2004

Increased density of the platelet serotonin transporter in autism

scientific article published in September 2000

Influence of chemical pollution on brain adenosine receptors of Mugil cephalus

article by Gino Giannaccini et al published October 1998 in Environmental Pollution

Is GRP78/BiP a potential salivary biomarker in patients with rheumatoid arthritis?

scientific article published on 4 January 2010

Jealousy and subthreshold psychopathology: a serotonergic link

scientific article published in January 2003

Lack of stereoselectivity of 8-hydroxy-2(di-N-propylamino)tetralin-mediated inhibition of forskolin-stimulated adenylyl cyclase activity in human pre- and post-synaptic brain regions

scientific article published on 01 March 2000

Male axillary extracts modify the affinity of the platelet serotonin transporter and impulsiveness in women

scientific article published on 27 March 2010

Modified RP-LC of Phenylthiocarbamyl Amino Acid Adducts in Plasma Acetonitrile Extracts Using Multiple Internal Standards and Photo-Diode UV Detection

article published in 2010

N'-Phenylindol-3-ylglyoxylohydrazide derivatives: synthesis, structure-activity relationships, molecular modeling studies, and pharmacological action on brain benzodiazepine receptors.

scientific article published in September 1998

N-Hydroxyindole-based inhibitors of lactate dehydrogenase against cancer cell proliferation

scientific article published on 8 September 2011

N-n-Propyl-substituted 3-(dimethylphenyl)piperidines display novel discriminative properties between dopamine receptor subtypes: synthesis and receptor binding studies

scientific article published in December 1998

Neuropeptide Y in the Brain and Retina of the Adult Teleost Gilthead Seabream (Sparus aurata L.)

scientific article published on 16 January 2008

New 1,2,3-triazolo[1,5-a]quinoxalines: synthesis and binding to benzodiazepine and adenosine receptors. II.

scientific article

New 4-(4-methyl-phenyl)phthalazin-1(2H)-one derivatives and their effects on α1-receptors

scientific article published on 20 March 2006

New insight into benign tumours of major salivary glands by proteomic approach

scientific article

New insight into the central benzodiazepine receptor-ligand interactions: design, synthesis, biological evaluation, and molecular modeling of 3-substituted 6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and related compounds

scientific article published on 27 July 2011

Novel 3-aralkyl-7-(amino-substituted)-1,2,3-triazolo[4,5-d]pyrimidines with high affinity toward A1 adenosine receptors

scientific article published in February 1998

Partial characterization of 3H-imipramine and 3H-paroxetine binding sites from calf striatum cerebral membranes

Peripheral benzodiazepine receptors on platelets of fibromyalgic patients

scientific article published on 13 July 2006

Peripheral-type benzodiazepine receptors in human blood cells of patients affected by migraine without aura

scientific article published on 01 October 2000

Peripheral-type benzodiazepine receptors in human mononuclear cells of patients affected by osteoarthritis, rheumatoid arthritis or psoriasic arthritis

scientific article

Pharmacological characterization of the serotonin transporter in young and elderly subjects.

scientific article published in January 2001

Phosphonomethylphosphorylmethyl(oxy)-analogues of geranylgeranyl diphosphate as stable and selective geranylgeranyl protein transferase inhibitors

Plasma Oxytocin Levels in Untreated Adult Obsessive-Compulsive Disorder Patients

Plasma clomipramine levels in adult patients with obsessive-compulsive disorder.

scientific article

Plasma fluvoxamine levels and OCD symptoms/response in adult patients

article

Plasma redox and inflammatory patterns during major depressive episodes: a cross-sectional investigation in elderly patients with mood disorders

scientific article published on 19 May 2020

Platelet [3H]paroxetine binding in patients with OCD-related disorders

article

Platelet alpha2-adrenoreceptors in obsessive-compulsive disorder

scientific article published in January 2004

Platelet peripheral benzodiazepine receptors are decreased in Parkinson's disease

scientific article published on 01 January 1991

Platelet proteome and clopidogrel response in patients with stable angina undergoing percutaneous coronary intervention

scientific article

Platelet serotonin transporter in patients with diarrhea-predominant irritable bowel syndrome both before and after treatment with alosetron

scientific article published in December 2003

Presence and characterization of the dopamine transporter in human resting lymphocytes

scientific article published on 22 November 2007

Presence and characterization of the serotonin transporter in human resting lymphocytes

scientific article published in August 1998

Presence of D4 dopamine receptors in human prefrontal cortex: a postmortem study

scientific article

Proteome analysis of whole saliva: a new tool for rheumatic diseases--the example of Sjögren's syndrome

scientific article published on May 2007

Proteomic analysis of saliva: a unique tool to distinguish primary Sjögren's syndrome from secondary Sjögren's syndrome and other sicca syndromes

scientific article

Proteomic approach used in the diagnosis of Riedel's thyroiditis: a case report

scientific article

Psychopharmacology and ethnicity: A comparative study on Senegalese and Italian men

scientific article published on 23 April 2019

Purification and characterization of the serotonin transporter from human brain

scholarly article by A. Rotondo et al published September 1994 in European Neuropsychopharmacology

RP-LC of Phenylthiocarbamyl Amino Acid Adducts in Plasma Acetonitrile Extracts: Use of Multiple Internal Standards and Variable Wavelength UV Detection

scientific article published on 01 January 2012

Regulation of the platelet serotonin transporter by protein kinase C in the young and elderly

scientific article published on 01 February 1999

Rosiglitazone reverses salbutamol-induced β(2) -adrenoceptor tolerance in airway smooth muscle

scientific article published on January 2011

Search for peripheral biomarkers in patients affected by acutely psychotic bipolar disorder: a proteomic approach

scientific article published on 19 February 2014

Serotonin receptor of type 6 (5-HT6) in human prefrontal cortex and hippocampus post-mortem: an immunohistochemical and immunofluorescence study.

scientific article published on 3 December 2012

Serotonin transporter (SERT) and translocator protein (TSPO) expression in the obese ob/ob mouse

scientific article

Sex-Related Differences in Plasma Oxytocin Levels in Humans

Short-term effects of 3,4-methylen-dioxy-metamphetamine (MDMA) on 5-HT(1A) receptors in the rat hippocampus

scientific article published on 31 May 2007

Simultaneous Plasma Level Analysis of Clomipramine, N-desmethylclomipramine, and Fluvoxamine by Reversed-Phase Liquid Chromatography

scientific article published on 01 April 2000

Simultaneous analysis of clozapine, clomipramine and their metabolites by reversed-phase liquid chromatography.

scientific article published in April 2001

Solubilization and characterization of [3H]Imipramine and [3H]Paroxetine binding sites from calf striatum

scientific article published on 01 October 1994

Solubilization of rat kidney benzodiazepine binding sites ⬇️

scientific article published on 01 March 1983

Species comparison of adenosine receptor subtypes in brain and testis

scientific article published on 7 November 2007

Specific inhibition of benzodiazepine receptor binding by some N-(indol-3-ylglyoxylyl) amino acid derivatives: stereoselective interactions

scientific article published on 01 December 1989

Stable analogues of geranylgeranyl diphosphate possessing improved geranylgeranyl versus farnesyl protein transferase inhibitory selectivity.

scientific article

Stable propylphosphonic acid analogues of geranylgeranyl diphosphate possessing inhibitory activity on geranylgeranyl protein transferase

scientific article published in November 2004

Stress-related changes of benzodiazepine binding inhibitory activity (B.B.I.A.) in humans

scientific article published in January 1990

Studies of peripheral benzodiazepine receptors in mussels: comparison between a polluted and a nonpolluted site

scientific article

Study on affinity profile toward native human and bovine adenosine receptors of a series of 1,8-naphthyridine derivatives

scientific article

Substituted 1,2,3-triazolo[1,5-a]quinazolines: synthesis and binding to benzodiazepine and adenosine receptors

scientific article published on 01 March 2000

Synthesis and 5-HT2A, 5-HT1A and alpha1-binding affinities of 2-[2-Hydroxy-3-(pyridin-3-yl-methyl)amino]-, 2-[2-hydroxy-3-(2-pyridin-2-yl-ethyl)amino]- and 2-[2-hydroxy-3-(4-N-methyl-piperazin-1-yl)-amino]propoxybenzaldehyde-O-(substituted) benzyl o

scientific article published in March 2007

Synthesis and biological activity of new 1,4-benzodioxan-arylpiperazine derivatives. Further validation of a pharmacophore model for alpha(1)-adrenoceptor antagonists

scientific article published in February 2002

Synthesis and biological affinity of new imidazo- and indol-arylpiperazine derivatives: further validation of a pharmacophore model for alpha(1)-adrenoceptor antagonists

scientific article published on 24 July 2008

Synthesis and α-adrenergic and I1-imidazoline activity of 3-phenylpiperidines dimethyl-substituted on the phenyl ring

Synthesis and β-adrenergic properties of tetrahydronaphthalene analogs of dichloroisoproterenol

Synthesis of Stable Analogues of Geranylgeranyl Diphosphate Possessing a (Z,E,E)-Geranylgeranyl Side Chain, Docking Analysis, and Biological Assays for Prenyl Protein Transferase Inhibition

scientific article published on 01 February 2006

Synthesis of aniline-type analogues of farnesyl diphosphate and their biological assays for prenyl protein transferase inhibitory activity

scientific article published in December 2003

Synthesis of new piperazine–pyridazinone derivatives and their binding affinity toward α1-, α2-adrenergic and 5-HT1A serotoninergic receptors

scientific article published on 20 December 2005

Synthesis of new pyridazinone derivatives and their affinity towards alpha1-alpha2-adrenoceptors

scientific article

Synthesis of sulfonamide-containing N-hydroxyindole-2-carboxylates as inhibitors of human lactate dehydrogenase-isoform 5

scientific article published on 17 October 2011

Synthesis, biological evaluation, and pharmacophore generation of new pyridazinone derivatives with affinity toward alpha(1)- and alpha(2)-adrenoceptors

scientific article published in June 2001

Synthesis, molecular docking and binding studies of selective serotonin transporter inhibitors

scholarly article by Susanna Nencetti et al published March 2011 in European Journal of Medicinal Chemistry

Synthesis, structure-activity relationships, and molecular modeling studies of N-(indol-3-ylglyoxylyl)benzylamine derivatives acting at the benzodiazepine receptor.

scientific article published in December 1996

The complex interactions amongst serotonin, insulin, leptin and glycolipid metabolic parameters in human obesity

scientific article published on 14 September 2020

The expression of platelet serotonin transporter (SERT) in human obesity

scientific article

The serotonin transporter from human brain: purification and partial characterization.

scientific article published in March 1996

The trace element content of top-soil and wild edible mushroom samples collected in Tuscany, Italy

scientific article published on 29 February 2012

Thermal balneotherapy induces changes of the platelet serotonin transporter in healthy subjects

scholarly article by Donatella Marazziti et al published October 2007 in Progress in Neuro-Psychopharmacology & Biological Psychiatry

Triazole-substituted N-hydroxyindol-2-carboxylates as inhibitors of isoform 5 of human lactate dehydrogenase (hLDH5)

Tricyclic heteroaromatic systems. [1]benzopyranopyrrol-4-ones and [1]benzopyrano-1,2,3-triazol-4-ones as benzodiazepine receptor ligands. Synthesis and structure-activity relationships

scientific article published in September 1990

Tubby protein in human lymphocytes from normal weight and obese subjects

scientific article

Variously substituted (phosphonoacetamido)oxy analogues of geranylgeranyl diphosphate (GGdP) as GGdP-transferase (GGTase) inhibitors and antiproliferative agents.

scientific article published on May 2005

X-ray analysis, theoretical studies and α-adrenergic biopharmacological properties of 1-(2,5-dimethoxyphenyl)-2-aminoethanol and its morpholine analogue

[(3)H]-YM-09151-2 binding sites in human brain postmortem.

scientific article published on 18 June 2009

[35S]TBPS binding to purified benzodiazepine-GABA-ionophore receptor complex: the effect of GABA on the modulation exerted by benzodiazepine site ligands

scientific article published on 01 January 1989

[3H] muscimol receptors sites in the carp (Cyprinus carpio L.) brain: binding assay and autoradiographic distribution

scientific article

[3H]-ketanserin binding sites in different psychiatric disorders

scientific article

[3H]PK11195 binding sites in human neutrophils: effect of fMLP stimulation and modulation in rheumatic diseases

scientific article published in January 2004

[3H]ketanserin binding in human brain postmortem.

scientific article published in June 1997

alpha(1)-Adrenoceptor antagonists. Rational design, synthesis and biological evaluation of new trazodone-like compounds

scientific article published in February 2002

alpha1-Adrenoceptor antagonists. 5. Pyridazinone-arylpiperazines. Probing the influence on affinity and selectivity of both ortho-alkoxy groups at the arylpiperazine moiety and cyclic substituents at the pyridazinone nucleus

scientific article published in January 2003

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