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List of works by Gianluca Papeo

A straightforward total synthesis of (-)-chaetominine.

scientific article published in August 2009

A submarine journey: the pyrrole-imidazole alkaloids.

scientific article

Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases

scientific article

Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy

scientific article

Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515 ⬇️

scientific article published on 13 March 2019

Improved synthesis of polyfluorinated L-lysine for 19F NMR-based screening

scientific article published on 22 November 2008

Insights into PARP Inhibitors' Selectivity Using Fluorescence Polarization and Surface Plasmon Resonance Binding Assays

scientific article published on 10 June 2014

Italian chemists' contributions to named reactions in organic synthesis: an historical perspective.

scientific article published on 04 September 2013

MutT Homolog 1 (MTH1): The Silencing of a Target

scientific article

Oxindole alkaloids. A novel non-biomimetic entry to (−)-Horsfiline

PARP inhibitors in cancer therapy: an update.

scientific article published on 05 February 2013

Poly(ADP-ribose) polymerase inhibition in cancer therapy: are we close to maturity?

scientific article published on October 2009

Synthesis of 3 10-helix-inducing constrained analogues of L-proline.

scientific article published in July 2004

Synthesis of a β-Carboline Scaffold Properly Functionalized for the Generation of Libraries of Bioactive Compounds

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