List of works - Adyary Fallarero

1,4-Substituted 4-(1H)-pyridylene-hydrazone-type inhibitors of AChE, BuChE, and amyloid-β aggregation crossing the blood-brain barrier

scientific article

Activity-based assay for human mono-ADP-ribosyltransferases ARTD7/PARP15 and ARTD10/PARP10 aimed at screening and profiling inhibitors.

scientific article published on 26 February 2013

Alpha- and β-casein components of host milk induce biofilm formation in the mastitis bacterium Streptococcus uberis

scientific article published on 12 November 2010

Automating a 96-well microtitre plate model for Staphylococcus aureus biofilms: an approach to screening of natural antimicrobial compounds

scientific article

Combining biofilm matrix measurements with biomass and viability assays in susceptibility assessments of antimicrobials against Staphylococcus aureus biofilms

scientific article

Coumarins permeability in Caco-2 cell model

scientific article published in February 2009

Effect of high concentration of Co (II) on Enterobacter liquefaciens strain C-1: a bacterium highly resistant to heavy metals with an unknown genome

scientific article published in May 2004

Effective Antibiofilm Polyketides against Staphylococcus aureus from the Pyranonaphthoquinone Biosynthetic Pathways of Streptomyces Species ⬇️

scientific article published on 20 July 2015

Effects of the aqueous extract of Bryothamnion triquetrum on chemical hypoxia and aglycemia-induced damage in GT1-7 mouse hypothalamic immortalized cells.

scientific article published on 29 June 2005

Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.

scientific article

GT1-7 cell-based cytoxicity screening assay on 96-well microplates as a platform for the safety assessment of genetically modified Gerbera hybrida extracts

scientific article published in January 2009

High-throughput screening with a miniaturized radioligand competition assay identifies new modulators of human α2-adrenoceptors.

scientific article

Homogeneous screening assay for human tankyrase.

scientific article

How to translate a bioassay into a screening assay for natural products: general considerations and implementation of antimicrobial screens.

scientific article

Identification and characterization of diarylimidazoles as hybrid inhibitors of butyrylcholinesterase and amyloid beta fibril formation

scientific article

Identification of Privileged Antichlamydial Natural Products by a Ligand-Based Strategy.

scientific article

Inhibition of acetylcholinesterase by coumarins: the case of coumarin 106.

scientific article

Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with beta-amyloid, acetylcholine, and butyrylcholine esterases

scientific article published on 15 January 2010

Liposomes-in-hydrogel delivery system with mupirocin: in vitro antibiofilm studies and in vivo evaluation in mice burn model.

scientific article

Living cells of Staphylococcus aureus immobilized onto the capillary surface in electrochromatography: a tool for screening of biofilms

scientific article published on 28 May 2008

Miniaturization and validation of the Ellman's reaction based acetylcholinesterase inhibitory assay into 384-well plate format and screening of a chemical library

scientific article

Molecular Docking Guided Comparative GFA, G/PLS, SVM and ANN Models of Structurally Diverse Dual Binding Site Acetylcholinesterase Inhibitors.

scientific article published on 4 August 2011

New derivatives of dehydroabietic acid target planktonic and biofilm bacteria in Staphylococcus aureus and effectively disrupt bacterial membrane integrity

scientific article published on 21 July 2015

Potency determinations of acetylcholinesterase inhibitors using Ellman’s reaction-based assay in screening: Effect of assay variants

scientific article published on 17 September 2010

Printed paper-based arrays as substrates for biofilm formation.

scientific article

Pros and cons of using resazurin staining for quantification of viable Staphylococcus aureus biofilms in a screening assay.

scientific article published on 8 May 2009

Revisiting an agar-based plate method: what the static biofilm method can offer for biofilm research

scientific article published on 01 December 2014

Screening and structural analysis of flavones inhibiting tankyrases

scientific article

Staphylococcus aureus biofilm susceptibility to small and potent β(2,2)-amino acid derivatives.

scientific article published on 21 November 2013

Studies on the toxicity of Punica granatum L. (Punicaceae) whole fruit extracts ⬇️

scientific article published on December 1, 2003

Systematic exploration of natural and synthetic flavonoids for the inhibition of Staphylococcus aureus biofilms

scientific article

The exploration of thienothiazines as selective butyrylcholinesterase inhibitors ⬇️

scientific article published on June 6, 2012

Towards fabrication of 3D printed medical devices to prevent biofilm formation

scientific article

List of works by Adyary Fallarero

1,4-Substituted 4-(1H)-pyridylene-hydrazone-type inhibitors of AChE, BuChE, and amyloid-β aggregation crossing the blood-brain barrier

Activity-based assay for human mono-ADP-ribosyltransferases ARTD7/PARP15 and ARTD10/PARP10 aimed at screening and profiling inhibitors.

Alpha- and β-casein components of host milk induce biofilm formation in the mastitis bacterium Streptococcus uberis

Automating a 96-well microtitre plate model for Staphylococcus aureus biofilms: an approach to screening of natural antimicrobial compounds

Combining biofilm matrix measurements with biomass and viability assays in susceptibility assessments of antimicrobials against Staphylococcus aureus biofilms

Coumarins permeability in Caco-2 cell model

Effect of high concentration of Co (II) on Enterobacter liquefaciens strain C-1: a bacterium highly resistant to heavy metals with an unknown genome

Effective Antibiofilm Polyketides against Staphylococcus aureus from the Pyranonaphthoquinone Biosynthetic Pathways of Streptomyces Species ⬇️

Effects of the aqueous extract of Bryothamnion triquetrum on chemical hypoxia and aglycemia-induced damage in GT1-7 mouse hypothalamic immortalized cells.

Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.

GT1-7 cell-based cytoxicity screening assay on 96-well microplates as a platform for the safety assessment of genetically modified Gerbera hybrida extracts

High-throughput screening with a miniaturized radioligand competition assay identifies new modulators of human α2-adrenoceptors.

Homogeneous screening assay for human tankyrase.

How to translate a bioassay into a screening assay for natural products: general considerations and implementation of antimicrobial screens.

Identification and characterization of diarylimidazoles as hybrid inhibitors of butyrylcholinesterase and amyloid beta fibril formation

Identification of Privileged Antichlamydial Natural Products by a Ligand-Based Strategy.

Inhibition of acetylcholinesterase by coumarins: the case of coumarin 106.

Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with beta-amyloid, acetylcholine, and butyrylcholine esterases

Liposomes-in-hydrogel delivery system with mupirocin: in vitro antibiofilm studies and in vivo evaluation in mice burn model.

Living cells of Staphylococcus aureus immobilized onto the capillary surface in electrochromatography: a tool for screening of biofilms

Miniaturization and validation of the Ellman's reaction based acetylcholinesterase inhibitory assay into 384-well plate format and screening of a chemical library

Molecular Docking Guided Comparative GFA, G/PLS, SVM and ANN Models of Structurally Diverse Dual Binding Site Acetylcholinesterase Inhibitors.

New derivatives of dehydroabietic acid target planktonic and biofilm bacteria in Staphylococcus aureus and effectively disrupt bacterial membrane integrity

Potency determinations of acetylcholinesterase inhibitors using Ellman’s reaction-based assay in screening: Effect of assay variants

Printed paper-based arrays as substrates for biofilm formation.

Pros and cons of using resazurin staining for quantification of viable Staphylococcus aureus biofilms in a screening assay.

Revisiting an agar-based plate method: what the static biofilm method can offer for biofilm research

Screening and structural analysis of flavones inhibiting tankyrases

Staphylococcus aureus biofilm susceptibility to small and potent β(2,2)-amino acid derivatives.

Studies on the toxicity of Punica granatum L. (Punicaceae) whole fruit extracts ⬇️

Systematic exploration of natural and synthetic flavonoids for the inhibition of Staphylococcus aureus biofilms

The exploration of thienothiazines as selective butyrylcholinesterase inhibitors ⬇️

Towards fabrication of 3D printed medical devices to prevent biofilm formation