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List of works by Paula Morales

(R)-N-(1-Methyl-2-hydroxyethyl)-13-(S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes

scientific article published on 21 September 2018

A Molecular Modeling Approach to Identify Novel Inhibitors of the Major Facilitator Superfamily of Efflux Pump Transporters

scientific article published on 15 March 2019

A critical review of both the synthesis approach and the receptor profile of the 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide and analogue derivatives.

scientific article published on 6 May 2016

An Overview on Medicinal Chemistry of Synthetic and Natural Derivatives of Cannabidiol

scientific article

An Update on Non-CB1, Non-CB2 Cannabinoid Related G-Protein-Coupled Receptors

scientific article published in October 2017

Antichagasic and trichomonacidal activity of 1-substituted 2-benzyl-5-nitroindazolin-3-ones and 3-alkoxy-2-benzyl-5-nitro-2H-indazoles.

scientific article

Antitumor Cannabinoid Chemotypes: Structural Insights

scientific article published on 31 May 2019

Biological characterization of PM226, a chromenoisoxazole, as a selective CB2 receptor agonist with neuroprotective profile.

scientific article published on 21 March 2016

CBD: A New Hope?

scientific article published on 29 April 2019

Cannabidiol skews biased agonism at cannabinoid CB1 and CB2 receptors with smaller effect in CB1-CB2 heteroreceptor complexes

article

Cannabinoid Ligands Targeting TRP Channels

scientific article published on 01 January 2018

Cannabinoid receptor 2 (CB2) agonists and antagonists: a patent update

scientific article published on 24 May 2016

Chromenopyrazole, a Versatile Cannabinoid Scaffold with in Vivo Activity in a Model of Multiple Sclerosis

scientific article published on 16 June 2016

Chromenopyrazoles: non-psychoactive and selective CB₁ cannabinoid agonists with peripheral antinociceptive properties

scientific article

Corrigendum to "Biological characterization of PM226, a chromenoisoxazole, as a selective CB2 receptor agonist with neuroprotective profile" [Pharmacol. Res. 110 (August 2016) (2016) 205-215].

scientific article published on 19 April 2017

Description of a bivalent cannabinoid ligand with hypophagic properties

scientific article

Design and structural characterisation of monomeric water-soluble α-helix and β-hairpin peptides: State-of-the-art

scientific article published on 20 November 2018

Emerging strategies targeting CB2 cannabinoid receptor: Biased agonism and allosterism

scientific article published on 26 July 2018

Identification of Novel GPR55 Modulators Using Cell-Impedance-Based Label-Free Technology.

scientific article published on 20 January 2016

Increased expression of cannabinoid CB2 and serotonin 5-HT1A heteroreceptor complexes in a model of newborn hypoxic-ischemic brain damage

scientific article published on 07 February 2019

Methods for the Development of In Silico GPCR Models

scientific article published on 14 July 2017

Molecular Targets of the Phytocannabinoids: A Complex Picture

scientific article published on January 2017

New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking

scientific article

Potential metabolic and behavioural roles of the putative endocannabinoid receptors GPR18, GPR55 and GPR119 in feeding

scientific article published on 01 January 2019

Selective, nontoxic CB(2) cannabinoid o-quinone with in vivo activity against triple-negative breast cancer.

scientific article published on 20 February 2015

Structural Insights into CB1 Receptor Biased Signaling

article

Structural Insights into β-arrestin/CB1 Receptor Interaction: NMR and CD Studies on Model Peptides

scientific article published on 30 October 2020

Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands

scientific article published on 16 April 2018

Synthesis, pharmacological evaluation and docking studies of pyrrole structure-based CB2 receptor antagonists.

scientific article published on 15 July 2015

Synthetic cannabinoid quinones: preparation, in vitro antiproliferative effects and in vivo prostate antitumor activity.

scientific article published on 2 October 2013

Targeting Cannabinoid CB2 Receptors in the Central Nervous System. Medicinal Chemistry Approaches with Focus on Neurodegenerative Disorders

scientific article

Towards A Molecular Understanding of The Cannabinoid Related Orphan Receptor GPR18: A Focus on Its Constitutive Activity

scientific article published on 09 May 2019

Towards a better understanding of the cannabinoid-related orphan receptors GPR3, GPR6, and GPR12.

scientific article published in February 2018