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List of works by Keith D. Combrink

1,2-Benzisothiazol-3-one 1,1-dioxide inhibitors of human mast cell tryptase.

scientific article

Discovery and early clinical evaluation of BMS-605339, a potent and orally efficacious tripeptidic acylsulfonamide NS3 protease inhibitor for the treatment of hepatitis C virus infection

scientific article

Discovery and structure-based optimization of adenain inhibitors.

scientific article published on 20 June 2014

In vivo optimization of 2,3-diaminopyrazine Rho Kinase inhibitors for the treatment of glaucoma

scientific article published on 19 March 2014

New C25 carbamate rifamycin derivatives are resistant to inactivation by ADP-ribosyl transferases.

scientific article

Oral efficacy of a respiratory syncytial virus inhibitor in rodent models of infection

scientific article

Orally active fusion inhibitor of respiratory syncytial virus

scientific article published on February 2004

Respiratory syncytial virus fusion inhibitors. Part 3: Water-soluble benzimidazol-2-one derivatives with antiviral activity in vivo

scientific article

Respiratory syncytial virus fusion inhibitors. Part 4: optimization for oral bioavailability

scientific article published in December 2006

Respiratory syncytial virus fusion inhibitors. Part 5: Optimization of benzimidazole substitution patterns towards derivatives with improved activity.

scientific article

Respiratory syncytial virus fusion inhibitors. Part 6: an examination of the effect of structural variation of the benzimidazol-2-one heterocycle moiety.

scientific article

Respiratory syncytial virus fusion inhibitors. Part 7: structure-activity relationships associated with a series of isatin oximes that demonstrate antiviral activity in vivo.

scientific article

Salicylamide inhibitors of influenza virus fusion

scientific article

Structure-based design and optimization of potent inhibitors of the adenoviral protease

scientific article

Synthesis and antibacterial evaluation of a novel series of rifabutin-like spirorifamycins

scientific article published on 12 December 2006

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